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Anaxis Pharma

Anaxis Pharma drug portfolio — 200 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Melbourne, AU HQ
2017 Founded
7 Employees
TGA registrant Type
Company details
Status
Public
HQ
Melbourne, AU
Founded
2017
Employees
7
Programs
10
Drugs
582
Patents
0
Intelligence · Drug Pipeline

Anaxis Pharma pipeline

Portfolio lens on 200 drugs and development assets — regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

Anaxis Pharma drug portfolio — 200 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

200 compounds
  1. abemaciclib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Cyclin-dependent kinase 4.

    Target
    Cyclin-dependent kinase 4
    Mechanism
    Cyclin-dependent kinase 6 inhibitor
  2. abiraterone

    Antineoplastic and immunomodulating agents (L02)

    Antineoplastic and immunomodulating agents (L02) compound in Anaxis Pharma's portfolio. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Steroid 5-alpha-reductase inhibitor
  3. abiraterone acetate

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Steroid 17-alpha-hydroxylase/17,20 lyase.

    Target
    Steroid 17-alpha-hydroxylase/17,20 lyase
    Mechanism
    Cytochrome P450 17A1 inhibitor
  4. acalabrutinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tyrosine-protein kinase BTK.

    Target
    Tyrosine-protein kinase BTK
    Mechanism
    Tyrosine-protein kinase BTK inhibitor
  5. US regulatory status: approved. Molecular target: Tyrosine-protein kinase BTK.

    Target
    Tyrosine-protein kinase BTK
    Mechanism
    Tyrosine-protein kinase BTK inhibitor
  6. US regulatory status: approved. Molecular target: Fatty-acid amide hydrolase 1.

    Target
    Fatty-acid amide hydrolase 1
    Mechanism
    Cyclooxygenase inhibitor
  7. US regulatory status: approved. Molecular target: Carbonic anhydrase 1.

    Target
    Carbonic anhydrase 1
    Mechanism
    Carbonic anhydrase XII inhibitor
  8. US regulatory status: approved. Molecular target: Retinoid receptor.

    Target
    Retinoid receptor
    Mechanism
    Retinoid receptor agonist
  9. US regulatory status: approved. Molecular target: DNA polymerase catalytic subunit.

    Target
    DNA polymerase catalytic subunit
    Mechanism
    Human herpesvirus 1 DNA polymerase inhibitor
  10. US regulatory status: approved. Molecular target: DNA polymerase catalytic subunit.

    Target
    DNA polymerase catalytic subunit
    Mechanism
    Human herpesvirus 1 DNA polymerase inhibitor
  11. adalimumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Tumor necrosis factor.

    Target
    Tumor necrosis factor
    Mechanism
    TNF-alpha inhibitor
  12. US regulatory status: approved. Molecular target: Tumor necrosis factor.

    Target
    Tumor necrosis factor
    Mechanism
    TNF-alpha inhibitor
  13. US regulatory status: approved. Molecular target: Tumor necrosis factor.

    Target
    Tumor necrosis factor
    Mechanism
    TNF-alpha inhibitor
  14. aflibercept

    Sensory organs (S01)

    US regulatory status: approved. Molecular target: Placenta growth factor.

    Target
    Placenta growth factor
    Mechanism
    Placenta growth factor inhibitor
  15. US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  16. US regulatory status: approved. Molecular target: Beta-2 adrenergic receptor.

    Target
    Beta-2 adrenergic receptor
    Mechanism
    Beta-2 adrenergic receptor agonist
  17. US regulatory status: approved. Molecular target: Beta-2 adrenergic receptor.

    Target
    Beta-2 adrenergic receptor
    Mechanism
    Beta-2 adrenergic receptor agonist
  18. US regulatory status: approved.

  19. alogliptin

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Mechanism: Dipeptidyl peptidase IV inhibitor.

    Mechanism
    Dipeptidyl peptidase IV inhibitor
  20. US regulatory status: approved. Molecular target: GABA-A receptor; anion channel.

    Target
    GABA-A receptor; anion channel
    Mechanism
    GABA-A receptor; anion channel positive allosteric modulator
  21. US regulatory status: approved. Molecular target: Prostaglandin E2 receptor EP1 subtype.

    Target
    Prostaglandin E2 receptor EP1 subtype
    Mechanism
    Prostanoid EP1 receptor agonist
  22. US regulatory status: approved. Molecular target: Adrenergic receptor alpha.

    Target
    Adrenergic receptor alpha
    Mechanism
    Adrenergic receptor alpha antagonist
  23. amifampridine

    Nervous system (N07)

    US regulatory status: approved. Molecular target: Voltage-gated potassium channel.

    Target
    Voltage-gated potassium channel
    Mechanism
    Voltage-gated potassium channel blocker
  24. US regulatory status: approved. Mechanism: Reactive metabolite scavenging agent.

    Mechanism
    Reactive metabolite scavenging agent
  25. amikacin

    Antiinfectives for systemic use (J01)

    Antiinfectives for systemic use (J01) compound in Anaxis Pharma's portfolio.

  26. US regulatory status: approved. Molecular target: Dopamine receptors; D2 & D3.

    Target
    Dopamine receptors; D2 & D3
    Mechanism
    Serotonin (5-HT) receptor antagonist
  27. amlodipine

    Cardiovascular system (C09)

    Cardiovascular system (C09) compound in Anaxis Pharma's portfolio. Mechanism: Voltage-gated L-type calcium channel blocker.

    Mechanism
    Voltage-gated L-type calcium channel blocker
  28. amlodipine besilate

    Cardiovascular system (C09)

    Cardiovascular system (C09) compound in Anaxis Pharma's portfolio. Molecular target: Voltage-gated L-type calcium channel.

    Target
    Voltage-gated L-type calcium channel
    Mechanism
    Voltage-gated L-type calcium channel blocker
  29. US regulatory status: approved. Molecular target: Voltage-gated L-type calcium channel.

    Target
    Voltage-gated L-type calcium channel
    Mechanism
    Voltage-gated L-type calcium channel blocker
  30. US regulatory status: approved. Molecular target: Bacterial penicillin-binding protein.

    Target
    Bacterial penicillin-binding protein
    Mechanism
    Bacterial penicillin-binding protein inhibitor
  31. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter releasing agent
  32. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter releasing agent
  33. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter releasing agent
  34. US regulatory status: approved. Molecular target: Ergosterol.

    Target
    Ergosterol
    Mechanism
    Ergosterol sequestering agent
  35. anidulafungin

    Antiinfectives for systemic use (J02)

    US regulatory status: approved. Molecular target: 1,3-beta-glucan synthase.

    Target
    1,3-beta-glucan synthase
    Mechanism
    1,3-beta-glucan synthase inhibitor
  36. US regulatory status: approved. Molecular target: Histamine H1 receptor.

    Target
    Histamine H1 receptor
    Mechanism
    Histamine H1 receptor antagonist
  37. Various (V09) compound in Anaxis Pharma's portfolio. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  38. apalutamide

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  39. apixaban

    Blood and blood forming organs (B01)

    US regulatory status: approved. Molecular target: Coagulation factor X.

    Target
    Coagulation factor X
    Mechanism
    Coagulation factor X inhibitor
  40. aprepitant

    Alimentary tract and metabolism (A04)

    US regulatory status: approved. Molecular target: Substance-P receptor.

    Target
    Substance-P receptor
    Mechanism
    Neurokinin 1 receptor antagonist
  41. aprocitentan

    Cardiovascular system (C02)

    US regulatory status: approved. Molecular target: Endothelin receptor, ET-A/ET-B.

    Target
    Endothelin receptor, ET-A/ET-B
    Mechanism
    Endothelin receptor, ET-A/ET-B antagonist
  42. arginine

    Various (V03)

    Various (V03) compound in Anaxis Pharma's portfolio.

  43. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Dopamine transporter inhibitor
  44. Development asset linked to Anaxis Pharma in public FDA and regional records.

  45. asenapine

    Nervous system (N05)

    US regulatory status: approved. Mechanism: Serotonin 2a (5-HT2a) receptor antagonist.

    Mechanism
    Serotonin 2a (5-HT2a) receptor antagonist
  46. US regulatory status: approved. Molecular target: Cyclooxygenase.

    Target
    Cyclooxygenase
    Mechanism
    Cyclooxygenase inhibitor
  47. atezolizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death 1 ligand 1.

    Target
    Programmed cell death 1 ligand 1
    Mechanism
    Programmed cell death 1 ligand 1 inhibitor
  48. US regulatory status: approved. Molecular target: Cytochrome b.

    Target
    Cytochrome b
    Mechanism
    Cytochrome b inhibitor
  49. atropine

    Sensory organs (S01)

    US regulatory status: approved. Molecular target: Muscarinic acetylcholine receptor M1.

    Target
    Muscarinic acetylcholine receptor M1
    Mechanism
    Muscarinic acetylcholine receptor M1 antagonist
  50. atropine sulfate

    Sensory organs (S01)

    US regulatory status: approved. Molecular target: Muscarinic acetylcholine receptor M1.

    Target
    Muscarinic acetylcholine receptor M1
    Mechanism
    Muscarinic acetylcholine receptor M3 antagonist
  51. aumolertinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Anaxis Pharma's portfolio. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  52. axicabtagene ciloleucel

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Anaxis Pharma's portfolio. Molecular target: B-lymphocyte antigen CD19.

    Target
    B-lymphocyte antigen CD19
    Mechanism
    B-lymphocyte antigen CD19 binding agent
  53. azacitidine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA (cytosine-5)-methyltransferase 1.

    Target
    DNA (cytosine-5)-methyltransferase 1
    Mechanism
    DNA (cytosine-5)-methyltransferase 3A inhibitor
  54. aztreonam

    Antiinfectives for systemic use (J01)

    US regulatory status: approved. Molecular target: Bacterial penicillin-binding protein.

    Target
    Bacterial penicillin-binding protein
    Mechanism
    Bacterial penicillin-binding protein inhibitor
  55. US regulatory status: approved. Molecular target: GABA-B receptor.

    Target
    GABA-B receptor
    Mechanism
    GABA-B receptor agonist
  56. Development asset linked to Anaxis Pharma in public FDA and regional records.

  57. US regulatory status: approved. Molecular target: Histone deacetylase.

    Target
    Histone deacetylase
    Mechanism
    Histone deacetylase inhibitor
  58. Development asset linked to Anaxis Pharma in public FDA and regional records.

  59. Development asset linked to Anaxis Pharma in public FDA and regional records. Molecular target: Cyclooxygenase.

    Target
    Cyclooxygenase
    Mechanism
    Cyclooxygenase inhibitor
  60. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  61. berotralstat

    Blood and blood forming organs (B06)

    Blood and blood forming organs (B06) compound in Anaxis Pharma's portfolio. Mechanism: Plasma kallikrein inhibitor.

    Mechanism
    Plasma kallikrein inhibitor
  62. Development asset linked to Anaxis Pharma in public FDA and regional records. Molecular target: Plasma kallikrein.

    Target
    Plasma kallikrein
    Mechanism
    Plasma kallikrein inhibitor
  63. bevacizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Vascular endothelial growth factor A, long form.

    Target
    Vascular endothelial growth factor A, long form
    Mechanism
    Vascular endothelial growth factor A inhibitor
  64. US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  65. Development asset linked to Anaxis Pharma in public FDA and regional records.

  66. bimekizumab

    Antineoplastic and immunomodulating agents (L04)

    Antineoplastic and immunomodulating agents (L04) compound in Anaxis Pharma's portfolio. Molecular target: Interleukin-17A.

    Target
    Interleukin-17A
    Mechanism
    Interleukin-17F inhibitor
  67. US regulatory status: approved. Molecular target: Interleukin-17A.

    Target
    Interleukin-17A
    Mechanism
    Interleukin 17A inhibitor
  68. bivalirudin

    Blood and blood forming organs (B01)

    US regulatory status: approved. Molecular target: Prothrombin.

    Target
    Prothrombin
    Mechanism
    Thrombin inhibitor
  69. bortezomib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  70. bosutinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Anaxis Pharma's portfolio. Molecular target: Tyrosine-protein kinase ABL1.

    Target
    Tyrosine-protein kinase ABL1
    Mechanism
    Tyrosine-protein kinase ABL inhibitor
  71. brentuximab vedotin

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  72. brexucabtagene autoleucel

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Anaxis Pharma's portfolio. Molecular target: B-lymphocyte antigen CD19.

    Target
    B-lymphocyte antigen CD19
    Mechanism
    B-lymphocyte antigen CD19 binding agent
  73. brigatinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: ALK tyrosine kinase receptor.

    Target
    ALK tyrosine kinase receptor
    Mechanism
    ALK tyrosine kinase receptor inhibitor
  74. US regulatory status: approved. Molecular target: DNA polymerase.

    Target
    DNA polymerase
    Mechanism
    DNA polymerase inhibitor
  75. brivaracetam

    Nervous system (N03)

    US regulatory status: approved. Molecular target: Synaptic vesicle glycoprotein 2A.

    Target
    Synaptic vesicle glycoprotein 2A
    Mechanism
    Synaptic vesicle glycoprotein 2A modulator
  76. Development asset linked to Anaxis Pharma in public FDA and regional records. Molecular target: Gamma-aminobutyric acid receptor subunit alpha-2.

    Target
    Gamma-aminobutyric acid receptor subunit alpha-2
    Mechanism
    GABA receptor alpha-2 subunit positive allosteric modulator
  77. Development asset linked to Anaxis Pharma in public FDA and regional records. Mechanism: Dopamine transporter inhibitor.

    Mechanism
    Dopamine transporter inhibitor
  78. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Dopamine transporter inhibitor
  79. busulfan

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  80. cabazitaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  81. cabozantinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Mechanism: Hepatocyte growth factor receptor inhibitor.

    Mechanism
    Hepatocyte growth factor receptor inhibitor
  82. caffeine

    Nervous system (N06)

    US regulatory status: approved. Molecular target: Adenosine receptor.

    Target
    Adenosine receptor
    Mechanism
    Adenosine receptor antagonist
  83. US regulatory status: approved. Molecular target: Vitamin D3 receptor.

    Target
    Vitamin D3 receptor
    Mechanism
    Vitamin D receptor agonist
  84. Development asset linked to Anaxis Pharma in public FDA and regional records. Molecular target: Vitamin D3 receptor.

    Target
    Vitamin D3 receptor
    Mechanism
    Vitamin D receptor agonist
  85. US regulatory status: approved. Molecular target: Vitamin D3 receptor.

    Target
    Vitamin D3 receptor
    Mechanism
    Vitamin D receptor agonist
  86. US regulatory status: approved.

  87. US regulatory status: approved. Mechanism: Dihydrofolate reductase inhibitor.

    Mechanism
    Dihydrofolate reductase inhibitor
  88. cannabidiol

    Nervous system (N03)

    US regulatory status: approved. Molecular target: Cannabinoid receptor 1.

    Target
    Cannabinoid receptor 1
    Mechanism
    Cannabinoid CB1 receptor negative allosteric modulator
  89. capecitabine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  90. capsaicin

    Nervous system (N01)

    US regulatory status: approved. Molecular target: Transient receptor potential cation channel subfamily V member 1.

    Target
    Transient receptor potential cation channel subfamily V member 1
    Mechanism
    Vanilloid receptor opener
  91. US regulatory status: approved. Molecular target: Angiotensin-converting enzyme.

    Target
    Angiotensin-converting enzyme
    Mechanism
    Angiotensin-converting enzyme inhibitor
  92. US regulatory status: approved. Molecular target: Sodium channel alpha subunit.

    Target
    Sodium channel alpha subunit
    Mechanism
    Sodium channel alpha subunit blocker
  93. Development asset linked to Anaxis Pharma in public FDA and regional records.

  94. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  95. carfilzomib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  96. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  97. US regulatory status: approved. Molecular target: Adrenergic receptor alpha-1.

    Target
    Adrenergic receptor alpha-1
    Mechanism
    Adrenergic receptor beta antagonist
  98. caspofungin

    Antiinfectives for systemic use (J02)

    Antiinfectives for systemic use (J02) compound in Anaxis Pharma's portfolio.

  99. cefepime

    Antiinfectives for systemic use (J01)

    Antiinfectives for systemic use (J01) compound in Anaxis Pharma's portfolio.

  100. ceftobiprole

    Antiinfectives for systemic use (J01)

    Antiinfectives for systemic use (J01) compound in Anaxis Pharma's portfolio. Molecular target: Bacterial penicillin-binding protein.

    Target
    Bacterial penicillin-binding protein
    Mechanism
    Bacterial penicillin-binding protein inhibitor
  101. cemiplimab

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Anaxis Pharma's portfolio. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  102. cetuximab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  103. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  104. US regulatory status: approved. Molecular target: Bacterial 70S ribosome.

    Target
    Bacterial 70S ribosome
    Mechanism
    Bacterial 70S ribosome inhibitor
  105. US regulatory status: approved. Molecular target: Cell membrane.

    Target
    Cell membrane
    Mechanism
    Cell membrane inhibitor
  106. chlormethine

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Anaxis Pharma's portfolio. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  107. US regulatory status: approved. Molecular target: Solute carrier family 12 member 3.

    Target
    Solute carrier family 12 member 3
    Mechanism
    Thiazide-sensitive sodium-chloride cotransporter inhibitor
  108. US regulatory status: approved. Molecular target: Solute carrier family 12 member 3.

    Target
    Solute carrier family 12 member 3
    Mechanism
    Thiazide-sensitive sodium-chloride cotransporter inhibitor
  109. cholic acid

    Alimentary tract and metabolism (A05)

    US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  110. cidofovir

    Antiinfectives for systemic use (J05)

    US regulatory status: approved. Molecular target: DNA polymerase catalytic subunit.

    Target
    DNA polymerase catalytic subunit
    Mechanism
    Human herpesvirus 1 DNA polymerase inhibitor
  111. US regulatory status: approved. Molecular target: Histamine H2 receptor.

    Target
    Histamine H2 receptor
    Mechanism
    Histamine H2 receptor antagonist
  112. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  113. Development asset linked to Anaxis Pharma in public FDA and regional records.

  114. cladribine

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  115. US regulatory status: approved. Molecular target: Bacterial 70S ribosome.

    Target
    Bacterial 70S ribosome
    Mechanism
    Bacterial 70S ribosome inhibitor
  116. US regulatory status: approved. Molecular target: GABA-A receptor; anion channel.

    Target
    GABA-A receptor; anion channel
    Mechanism
    GABA-A receptor; anion channel positive allosteric modulator
  117. US regulatory status: approved. Molecular target: D(2) dopamine receptor.

    Target
    D(2) dopamine receptor
    Mechanism
    Serotonin 2a (5-HT2a) receptor antagonist
  118. Development asset linked to Anaxis Pharma in public FDA and regional records. Mechanism: Opioid receptors; mu/kappa/delta agonist.

    Mechanism
    Opioid receptors; mu/kappa/delta agonist
  119. US regulatory status: approved. Molecular target: Opioid receptors; mu/kappa/delta.

    Target
    Opioid receptors; mu/kappa/delta
    Mechanism
    Opioid receptors; mu/kappa/delta agonist
  120. colchicine

    Musculo-skeletal system (M04)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  121. Development asset linked to Anaxis Pharma in public FDA and regional records.

  122. US regulatory status: approved. Molecular target: Anoctamin-1.

    Target
    Anoctamin-1
    Mechanism
    Cystic fibrosis transmembrane conductance regulator inhibitor
  123. US regulatory status: approved. Mechanism: Supplement.

    Mechanism
    Supplement
  124. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  125. cytarabine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA polymerase (alpha/delta/epsilon) inhibitor
  126. dabrafenib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Anaxis Pharma's portfolio. Mechanism: Serine/threonine-protein kinase B-raf inhibitor.

    Mechanism
    Serine/threonine-protein kinase B-raf inhibitor
  127. danicopan

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Complement factor D.

    Target
    Complement factor D
    Mechanism
    Complement factor D inhibitor
  128. Development asset linked to Anaxis Pharma in public FDA and regional records. Mechanism: Ryanodine receptor 3 antagonist.

    Mechanism
    Ryanodine receptor 3 antagonist
  129. US regulatory status: approved. Molecular target: Ryanodine receptor 1.

    Target
    Ryanodine receptor 1
    Mechanism
    Ryanodine receptor 3 antagonist
  130. daratumumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1.

    Target
    ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
    Mechanism
    Lymphocyte differentiation antigen CD38 inhibitor
  131. daridorexant

    Nervous system (N05)

    Nervous system (N05) compound in Anaxis Pharma's portfolio. Molecular target: Orexin receptor.

    Target
    Orexin receptor
    Mechanism
    Orexin receptor antagonist
  132. dasatinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Bcr/Abl fusion protein.

    Target
    Bcr/Abl fusion protein
    Mechanism
    SRC inhibitor
  133. US regulatory status: approved. Molecular target: Vasopressin receptor.

    Target
    Vasopressin receptor
    Mechanism
    Vasopressin receptor agonist
  134. US regulatory status: approved. Molecular target: Progesterone receptor.

    Target
    Progesterone receptor
    Mechanism
    Progesterone receptor agonist
  135. US regulatory status: approved. Molecular target: Mineralocorticoid receptor.

    Target
    Mineralocorticoid receptor
    Mechanism
    Mineralocorticoid receptor agonist
  136. deucravacitinib

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Non-receptor tyrosine-protein kinase TYK2.

    Target
    Non-receptor tyrosine-protein kinase TYK2
    Mechanism
    Tyrosine-protein kinase TYK2 negative allosteric modulator
  137. dexamethasone

    Systemic hormonal preparations (H02)

    US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  138. dexamethasone phosphate

    Systemic hormonal preparations (H02)

    Systemic hormonal preparations (H02) compound in Anaxis Pharma's portfolio.

  139. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  140. Development asset linked to Anaxis Pharma in public FDA and regional records. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Dopamine transporter releasing agent
  141. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter releasing agent
  142. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Dopamine transporter releasing agent
  143. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter releasing agent
  144. US regulatory status: approved.

  145. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  146. US regulatory status: approved. Molecular target: Sodium/potassium-transporting ATPase.

    Target
    Sodium/potassium-transporting ATPase
    Mechanism
    Sodium/potassium-transporting ATPase inhibitor
  147. US regulatory status: approved. Molecular target: Histamine H1 receptor.

    Target
    Histamine H1 receptor
    Mechanism
    Histamine H1 receptor antagonist
  148. Development asset linked to Anaxis Pharma in public FDA and regional records. Mechanism: Histamine H1 receptor antagonist.

    Mechanism
    Histamine H1 receptor antagonist
  149. US regulatory status: approved. Molecular target: Histamine H1 receptor.

    Target
    Histamine H1 receptor
    Mechanism
    Histamine H1 receptor antagonist
  150. Development asset linked to Anaxis Pharma in public FDA and regional records. Mechanism: Sodium channel alpha subunit blocker.

    Mechanism
    Sodium channel alpha subunit blocker
  151. Development asset linked to Anaxis Pharma in public FDA and regional records. Mechanism: Surfactant laxative.

    Mechanism
    Surfactant laxative
  152. Development asset linked to Anaxis Pharma in public FDA and regional records. Mechanism: Beta-1 adrenergic receptor agonist.

    Mechanism
    Beta-1 adrenergic receptor agonist
  153. doxorubicin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Anaxis Pharma's portfolio. Mechanism: DNA topoisomerase II alpha inhibitor.

    Mechanism
    DNA topoisomerase II alpha inhibitor
  154. dupilumab

    Dermatologicals (D11)

    US regulatory status: approved. Molecular target: Interleukin-4 receptor subunit alpha.

    Target
    Interleukin-4 receptor subunit alpha
    Mechanism
    Interleukin-4 receptor subunit alpha antagonist
  155. durvalumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death 1 ligand 1.

    Target
    Programmed cell death 1 ligand 1
    Mechanism
    Programmed cell death 1 ligand 1 inhibitor
  156. eculizumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Complement C5.

    Target
    Complement C5
    Mechanism
    Complement C5 inhibitor
  157. edaravone

    Nervous system (N07)

    US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  158. elacestrant

    Antineoplastic and immunomodulating agents (L02)

    Antineoplastic and immunomodulating agents (L02) compound in Anaxis Pharma's portfolio. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha degrader
  159. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha degrader
  160. empagliflozin

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Sodium/glucose cotransporter 2.

    Target
    Sodium/glucose cotransporter 2
    Mechanism
    Sodium/glucose cotransporter 2 inhibitor
  161. enoxaparin sodium

    Blood and blood forming organs (B01)

    US regulatory status: approved. Molecular target: Antithrombin-III.

    Target
    Antithrombin-III
    Mechanism
    Antithrombin-III activator
  162. ensifentrine

    Respiratory system (R03)

    US regulatory status: approved. Molecular target: Phosphodiesterase 3.

    Target
    Phosphodiesterase 3
    Mechanism
    Phosphodiesterase 4 inhibitor
  163. enzalutamide

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  164. epinephrine

    Cardiovascular system (C01)

    US regulatory status: approved. Molecular target: Adrenergic receptor.

    Target
    Adrenergic receptor
    Mechanism
    Adrenergic receptor agonist
  165. US regulatory status: approved. Molecular target: Vitamin D3 receptor.

    Target
    Vitamin D3 receptor
    Mechanism
    Vitamin D receptor agonist
  166. erlotinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Anaxis Pharma's portfolio. Mechanism: Epidermal growth factor receptor erbB1 inhibitor.

    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  167. US regulatory status: approved. Molecular target: Bacterial 70S ribosome.

    Target
    Bacterial 70S ribosome
    Mechanism
    Bacterial 70S ribosome inhibitor
  168. US regulatory status: approved. Molecular target: Bacterial 70S ribosome.

    Target
    Bacterial 70S ribosome
    Mechanism
    Bacterial 70S ribosome inhibitor
  169. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  170. Development asset linked to Anaxis Pharma in public FDA and regional records. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor modulator
  171. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  172. etanercept

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Tumor necrosis factor.

    Target
    Tumor necrosis factor
    Mechanism
    TNF-alpha inhibitor
  173. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist