Wednesday, July 8, 2026

Drug profile · INN

dasatinib

dasatinib (DASATINIB ARX) is a src inhibitor. Associated with Alphapharm Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

FDA: approved EMA: approved TGA: approved Antineoplastic and immunomodulating agents (L01) L01EA02
US status approved
Patents linked 19
Pipeline programs 13
News articles 0
Drug details — dasatinib
US status
approved
Class
Antineoplastic and immunomodulating agents (L01)
Route
ORAL
Patents
19
Programs
13
Data quality
0.89

Quick answer

dasatinib (DASATINIB ARX) is a src inhibitor. Associated with Alphapharm Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN dasatinib
Brand DASATINIB ARX
Mechanism SRC inhibitor
Target Bcr/Abl fusion protein
Therapeutic class Antineoplastic and immunomodulating agents (L01)
Route ORAL
Formulation TABLET
ATC code L01EA02

Mechanism of action

SRC inhibitor

Primary target: Bcr/Abl fusion protein

Approval history

Authority Status Date
FDA approved
EMA approved
TGA approved

Pipeline programs

  1. CABL001A2001B Phase 3 · Novartis India · chronic myelogenous leukemia (CML) or Philadelphia Chromosom
  2. CABL001J12301 Phase 3 · Novartis India · Chronic Myeloid Leukemia
  3. HQP1351AG301 Phase 3 · Anaxis Pharma · Newly Diagnosed Philadelphia Chromosome-Positive Acute Lymph
  4. BCN04-DASA Phase 2 · George Institute for · Human immunodeficiency virus
  5. CA180-226 Phase 2 · Bristol-Myers Squibb Australia · Children and Adolescents with Newly Diagnosed Chronic Phase
  6. DASATINIB, Placebo Phase 2 · George Institute for · Asymptomatic patients with recent HIV-1 infection
  7. Dasatinib Phase 2 · Bristol Myers Squibb · Chronic Myeloid Leukemia
  8. Dasatinib Phase 2 · Takeda · Acute Lymphoblastic Leukemia

Related & competitor drugs

  1. abiraterone acetate Antineoplastic and immunomodulating agents (L02)
  2. anagrelide Antineoplastic and immunomodulating agents (L01)
  3. apremilast Antineoplastic and immunomodulating agents (L04)
  4. arsenic trioxide Antineoplastic and immunomodulating agents (L01)
  5. axitinib Antineoplastic and immunomodulating agents (L01)
  6. azacitidine Antineoplastic and immunomodulating agents (L01)
  1. US 20260152488

    AMIDE-SUBSTITUTED HETEROCYCLIC COMPOUNDS

    Expires Wed May 30 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. WO 2026112386

    COMPOSÉS D'OXOISOINDOLINYL PIPÉRIDINE-2,6-DIONE SUBSTITUÉS ET PROCÉDÉS DE DÉGRADATION DE PROTÉINES

    Expires Wed May 23 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. WO 2026112045

    NICOTINAMIDES PYRAZOLYLIQUES ET CARBOXAMIDES PYRIMIDINIQUES EN TANT QU'INHIBITEURS DE CAMK2

    Expires Wed May 23 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. WO 2026112047

    AMIDES DE PYRIDINE ET DE PYRIMIDINE EN TANT QU'INHIBITEURS DE CAMK2

    Expires Wed May 23 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  5. WO 2026107420

    DÉRIVÉS DE N-(4-(1H-BENZO[D[IMIDAZOL-6-YL)-PYRIDIN-2-YL)BENZAMIDE UTILES COMME INHIBITEURS DE CAMK2 POUR LE TRAITEMENT DE L'INSUFFISANCE CARDIAQUE

    Expires Wed May 16 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  6. WO 2026107418

    DÉRIVÉS DE N-(4-(1H-BENZO[D[IMIDAZOL-6-YL)-PYRIDIN-2-YL)BENZAMIDE UTILISÉS EN TANT QU'INHIBITEURS DE CAMK2 POUR LE TRAITEMENT D'UNE INSUFFISANCE CARDIAQUE

    Expires Wed May 16 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  7. WO 2026107421

    DÉRIVÉS DE 1H-BENZO[D]IMIDAZOLE UTILES COMME INHIBITEURS DE CAMK2 POUR LE TRAITEMENT DE L'INSUFFISANCE CARDIAQUE

    Expires Wed May 16 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  8. WO 2026107422

    DÉRIVÉS DE 6-(PYRIDIN-4-YL)-1H-BENZO[D]IMIDAZOLE UTILES COMME INHIBITEURS DE CAMK2 POUR LE TRAITEMENT DE L'INSUFFISANCE CARDIAQUE

    Expires Wed May 16 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  9. WO 2026107425

    DÉRIVÉS DE 5-(PYRIDIN-4-YL)-3H-IMIDAZO[4,5-B]PYRIDINE UTILES COMME INHIBITEURS DE CAMK2 POUR LE TRAITEMENT DE L'INSUFFISANCE CARDIAQUE

    Expires Wed May 16 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  10. WO 2026107424

    DÉRIVÉS DE N-(4-(IMIDAZO[4,5-B]PYRIDIN-5-YL)-2-PYRIDYL)BENZAMIDE UTILES COMME INHIBITEURS DE CAMK2 POUR LE TRAITEMENT DE L'INSUFFISANCE CARDIAQUE

    Expires Wed May 16 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  11. WO 2026096847

    MÉTHODES DE RÉGULATION DE L'INFLAMMATION ET DE L'AUTOPHAGIE À L'AIDE DE PIÈGES À LIGANDS ACTRIIB

    Expires Wed May 02 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  12. WO 2026080794

    COMPOSÉS CHIMIQUES UTILES POUR DÉGRADER DES PROTÉINES

    Expires Wed Apr 11 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  13. WO 2026075941

    DÉRIVÉS DE PYRIDAZINONE EN TANT QU'INHIBITEURS DE PAD4

    Expires Wed Apr 04 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  14. WO 2026039512

    INHIBITEURS DE KRAS

    Expires Wed Feb 14 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  15. WO 2026035787

    MACROCYLES DE PROTÉASE DE TRAITEMENT SPÉCIFIQUE DE L'UBIQUITINE (USP1)

    Expires Wed Feb 07 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  16. US 20260035358

    WEE1 DEGRADING COMPOUNDS AND USES THEREOF

    Expires Wed Jan 31 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  17. WO 2026011019

    COMPOSÉS PYRROLIDINYLE UTILISÉS EN TANT QU'INHIBITEURS DE CGAZ

    Expires Wed Jan 03 2046 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  18. US 8067423

    Polymorphs of dasatinib isopropyl alcohol and process for preparation thereof

    Expires Mon Nov 24 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  19. US 7973045

    Anhydrous form of dasatinib and process for preparation thereof

    Expires Mon Jun 30 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is dasatinib?

dasatinib (DASATINIB ARX) is a src inhibitor. Associated with Alphapharm Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for dasatinib?

DASATINIB ARX is a marketed brand name for dasatinib. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of dasatinib?

dasatinib has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.