Wednesday, July 8, 2026

Drug profile · INN

carvedilol

carvedilol (APO-CARVEDILOL) is a adrenergic receptor beta antagonist. Associated with Alphapharm Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

FDA: approved TGA: approved PMDA: approved
US status approved
Patents linked 20
Pipeline programs 17
News articles 0
Drug details — carvedilol
US status
approved
Class
Route
ORAL
Patents
20
Programs
17
Data quality
0.89

Quick answer

carvedilol (APO-CARVEDILOL) is a adrenergic receptor beta antagonist. Associated with Alphapharm Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN carvedilol
Brand APO-CARVEDILOL
Mechanism Adrenergic receptor beta antagonist
Target Adrenergic receptor alpha-1
Route ORAL
Formulation TABLET

Mechanism of action

Adrenergic receptor beta antagonist

Primary target: Adrenergic receptor alpha-1

Approval history

Authority Status Date
FDA approved
TGA approved
PMDA approved

Pipeline programs

  1. APHP230833 Phase 3 · PARItec · Heart failure
  2. D910DC00001 Phase 3 · AstraZeneca · Histologically or cytologically confirmed Locoregional Hepat
  3. D910VC00001 Phase 3 · AstraZeneca · Locoregional Hepatocellular Carcinoma (HCC)
  4. EMERALD-1 Phase 3 · AstraZeneca · Locoregional Hepatocellular Carcinoma (HCC)
  5. IBCSG 59-19 Phase 3 · Impact Therapeutics · Female or male patients with histologically confirmed HR-pos
  6. ASND0038 Phase 2 · Anaxis Pharma · Stage III-IVA Resectable Locoregionall Advanced Head and Nec
  7. Carvedilol Phase 2 · BRIGHT MINDS BIOSCIENCES · Cocaine-Related Disorders
  8. Carvedilol Phase 2 · NORTHWEST BIOTHERAPEUTICS · Post-Traumatic Stress Disorder

Related & competitor drugs

  1. doxazosin mesylate Adrenergic receptor alpha-1 antagonist
  2. midodrine hydrochloride Adrenergic receptor alpha-1 agonist
  3. phenylephrine hydrochloride Adrenergic receptor alpha-1 agonist
  4. prazosin hydrochloride Adrenergic receptor alpha-1 antagonist
  5. tamsulosin hydrochloride Adrenergic receptor alpha-1 antagonist
  6. terazosin hydrochloride Adrenergic receptor alpha-1 antagonist
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Frequently asked questions

What is carvedilol?

carvedilol (APO-CARVEDILOL) is a adrenergic receptor beta antagonist. Associated with Alphapharm Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for carvedilol?

APO-CARVEDILOL is a marketed brand name for carvedilol. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of carvedilol?

carvedilol has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.