Wednesday, July 8, 2026

Drug profile · INN

alseroxylon

alseroxylon (RAUWILOID) is a adrenergic receptor alpha antagonist. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 4
Pipeline programs 8
News articles 0
Drug details — alseroxylon
US status
approved
Class
Route
ORAL
Patents
4
Programs
8
Data quality
0.84

Quick answer

alseroxylon (RAUWILOID) is a adrenergic receptor alpha antagonist. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN alseroxylon
Brand RAUWILOID
Mechanism Adrenergic receptor alpha antagonist
Target Adrenergic receptor alpha
Route ORAL
Formulation TABLET

Mechanism of action

Adrenergic receptor alpha antagonist

Primary target: Adrenergic receptor alpha

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. MT-1186 Phase 3 · Tanabe Pharma · ALS
  2. AMX0035 Phase 2 · Amylyx Pharmaceuticals EMEA · ALS
  3. Riluzole Oral Soluble Film Phase 2 · Aquestive Therapeutics · ALS
  4. Talampanel Phase 2 · Teva Pharma · ALS
  5. Triheptanoin Phase 2 · Ultragenyx UK · ALS
  6. [11C]CPPC PET ligand Phase 2 · United Therapeutics Europe · ALS
  7. AMX0114 Phase 1 · Amylyx Pharmaceuticals EMEA · ALS
  8. MP-101-02 Phase 1 · Anaxis Pharma · Amyotrophic Lateral Sclerosis (ALS), Alzheimer’s Disease (AD

Related & competitor drugs

  1. brimonidine tartrate Adrenergic receptor alpha-2 agonist
  2. carvedilol Adrenergic receptor beta antagonist
  3. clonidine hydrochloride Adrenergic receptor alpha-2 agonist
  4. dexmedetomidine hydrochloride Adrenergic receptor alpha-2 agonist
  5. doxazosin mesylate Adrenergic receptor alpha-1 antagonist
  6. guanfacine hydrochloride Adrenergic receptor alpha-2 agonist

Related patents

  1. US 12246027

    Compositions of bile acids and phenylbutyrate compounds

    Expires Mon Mar 06 2045 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 12186330

    Compositions for improving cell viability and methods of use thereof

    Expires Mon Jan 02 2045 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 12138272

    Methods and compositions for treating amyotrophic lateral sclerosis

    Expires Mon Nov 07 2044 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. US 11559533

    Compositions of bile acids and phenylbutyrate compounds

    Expires Mon Jan 19 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is alseroxylon?

alseroxylon (RAUWILOID) is a adrenergic receptor alpha antagonist. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for alseroxylon?

RAUWILOID is a marketed brand name for alseroxylon. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of alseroxylon?

alseroxylon has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.