Wednesday, July 8, 2026

biotech · Non small cell lung cancer · oligometastatic hormone sensitive prostate cancer · CERO

CERo Therapeutics

CERo Therapeutics drug portfolio — 80 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

201 Haskins Way, 230, South San Francisco, California 94080, US HQ
17 Employees
Public company Type
CERO · NYSE Ticker
Company details
Status
Public
HQ
201 Haskins Way, 230, South San Francisco, California 94080, US
Employees
17
Programs
47
Drugs
84
Patents
14
Intelligence · Drug Pipeline

CERo Therapeutics pipeline

Portfolio lens on 80 drugs and development assets — regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

CERo Therapeutics drug portfolio — 80 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

80 compounds
  1. aflibercept

    Sensory organs (S01)

    US regulatory status: approved. Molecular target: Placenta growth factor.

    Target
    Placenta growth factor
    Mechanism
    Placenta growth factor inhibitor
  2. US regulatory status: approved. Molecular target: Phosphodiesterase 4.

    Target
    Phosphodiesterase 4
    Mechanism
    Phosphodiesterase 4 inhibitor
  3. US regulatory status: approved. Molecular target: Cyclooxygenase.

    Target
    Cyclooxygenase
    Mechanism
    Cyclooxygenase inhibitor
  4. atezolizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death 1 ligand 1.

    Target
    Programmed cell death 1 ligand 1
    Mechanism
    Programmed cell death 1 ligand 1 inhibitor
  5. avelumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death 1 ligand 1.

    Target
    Programmed cell death 1 ligand 1
    Mechanism
    Programmed cell death 1 ligand 1 other
  6. bevacizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Vascular endothelial growth factor A, long form.

    Target
    Vascular endothelial growth factor A, long form
    Mechanism
    Vascular endothelial growth factor A inhibitor
  7. binimetinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Dual specificity mitogen-activated protein kinase kinase 1.

    Target
    Dual specificity mitogen-activated protein kinase kinase 1
    Mechanism
    Dual specificity mitogen-activated protein kinase kinase 1 inhibitor
  8. brigatinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: ALK tyrosine kinase receptor.

    Target
    ALK tyrosine kinase receptor
    Mechanism
    ALK tyrosine kinase receptor inhibitor
  9. US regulatory status: approved.

  10. capecitabine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  11. Development asset linked to CERo Therapeutics in public FDA and regional records.

  12. Development asset linked to CERo Therapeutics in public FDA and regional records.

  13. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  14. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  15. cemiplimab

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in CERo Therapeutics's portfolio. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  16. US regulatory status: approved. Molecular target: Gonadotropin-releasing hormone receptor.

    Target
    Gonadotropin-releasing hormone receptor
    Mechanism
    Gonadotropin-releasing hormone receptor antagonist
  17. cetuximab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  18. Development asset linked to CERo Therapeutics in public FDA and regional records.

  19. choriogonadotropin alfa

    Genito-urinary system and sex hormones (G03)

    US regulatory status: approved. Molecular target: Lutropin-choriogonadotropic hormone receptor.

    Target
    Lutropin-choriogonadotropic hormone receptor
    Mechanism
    Luteinizing hormone/Choriogonadotropin receptor agonist
  20. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  21. clopidogrel

    Blood and blood forming organs (B01)

    Blood and blood forming organs (B01) compound in CERo Therapeutics's portfolio. Mechanism: Purinergic receptor P2Y12 antagonist.

    Mechanism
    Purinergic receptor P2Y12 antagonist
  22. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  23. denosumab

    Musculo-skeletal system (M05)

    US regulatory status: approved. Molecular target: Tumor necrosis factor ligand superfamily member 11.

    Target
    Tumor necrosis factor ligand superfamily member 11
    Mechanism
    Tumor necrosis factor ligand superfamily member 11 inhibitor
  24. docetaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  25. durvalumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death 1 ligand 1.

    Target
    Programmed cell death 1 ligand 1
    Mechanism
    Programmed cell death 1 ligand 1 inhibitor
  26. encorafenib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Serine/threonine-protein kinase B-raf.

    Target
    Serine/threonine-protein kinase B-raf
    Mechanism
    Serine/threonine-protein kinase B-raf inhibitor
  27. Development asset linked to CERo Therapeutics in public FDA and regional records.

  28. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  29. Development asset linked to CERo Therapeutics in public FDA and regional records.

  30. follitropin beta

    Genito-urinary system and sex hormones (G03)

    Genito-urinary system and sex hormones (G03) compound in CERo Therapeutics's portfolio. Molecular target: Follicle-stimulating hormone receptor.

    Target
    Follicle-stimulating hormone receptor
    Mechanism
    Follicle stimulating hormone receptor agonist
  31. fruquintinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Vascular endothelial growth factor receptor.

    Target
    Vascular endothelial growth factor receptor
    Mechanism
    Vascular endothelial growth factor receptor inhibitor
  32. US regulatory status: approved. Mechanism: DNA polymerase (alpha/delta/epsilon) inhibitor.

    Mechanism
    DNA polymerase (alpha/delta/epsilon) inhibitor
  33. Development asset linked to CERo Therapeutics in public FDA and regional records. Mechanism: Mu opioid receptor agonist.

    Mechanism
    Mu opioid receptor agonist
  34. Development asset linked to CERo Therapeutics in public FDA and regional records.

  35. Development asset linked to CERo Therapeutics in public FDA and regional records.

  36. Development asset linked to CERo Therapeutics in public FDA and regional records.

  37. ipilimumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Cytotoxic T-lymphocyte protein 4.

    Target
    Cytotoxic T-lymphocyte protein 4
    Mechanism
    Cytotoxic T-lymphocyte protein 4 inhibitor
  38. Development asset linked to CERo Therapeutics in public FDA and regional records. Mechanism: DNA topoisomerase I inhibitor.

    Mechanism
    DNA topoisomerase I inhibitor
  39. US regulatory status: approved. Molecular target: DNA topoisomerase 1.

    Target
    DNA topoisomerase 1
    Mechanism
    DNA topoisomerase I inhibitor
  40. Development asset linked to CERo Therapeutics in public FDA and regional records.

  41. lorlatinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: ALK tyrosine kinase receptor.

    Target
    ALK tyrosine kinase receptor
    Mechanism
    EML4-ALK inhibitor
  42. Development asset linked to CERo Therapeutics in public FDA and regional records. Molecular target: Polyunsaturated fatty acid 5-lipoxygenase.

    Target
    Polyunsaturated fatty acid 5-lipoxygenase
    Mechanism
    Arachidonate 5-lipoxygenase inhibitor
  43. Development asset linked to CERo Therapeutics in public FDA and regional records. Mechanism: Mitochondrial complex I (NADH dehydrogenase) inhibitor.

    Mechanism
    Mitochondrial complex I (NADH dehydrogenase) inhibitor
  44. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  45. Development asset linked to CERo Therapeutics in public FDA and regional records.

  46. nivolumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  47. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  48. paclitaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  49. panitumumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  50. pembrolizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  51. US regulatory status: approved. Molecular target: Dihydrofolate reductase.

    Target
    Dihydrofolate reductase
    Mechanism
    Thymidylate synthase inhibitor
  52. Development asset linked to CERo Therapeutics in public FDA and regional records.

  53. Development asset linked to CERo Therapeutics in public FDA and regional records.

  54. pioglitazone

    Alimentary tract and metabolism (A10)

    Alimentary tract and metabolism (A10) compound in CERo Therapeutics's portfolio. Mechanism: Peroxisome proliferator-activated receptor gamma agonist.

    Mechanism
    Peroxisome proliferator-activated receptor gamma agonist
  55. Development asset linked to CERo Therapeutics in public FDA and regional records.

  56. US regulatory status: approved. Mechanism: Supplement.

    Mechanism
    Supplement
  57. Development asset linked to CERo Therapeutics in public FDA and regional records.

  58. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  59. Development asset linked to CERo Therapeutics in public FDA and regional records.

  60. Development asset linked to CERo Therapeutics in public FDA and regional records.

  61. ramucirumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Vascular endothelial growth factor receptor 2.

    Target
    Vascular endothelial growth factor receptor 2
    Mechanism
    Vascular endothelial growth factor receptor 2 inhibitor
  62. Development asset linked to CERo Therapeutics in public FDA and regional records.

  63. Development asset linked to CERo Therapeutics in public FDA and regional records.

  64. sotorasib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: GTPase KRas.

    Target
    GTPase KRas
    Mechanism
    GTPase KRas inhibitor
  65. Development asset linked to CERo Therapeutics in public FDA and regional records.

  66. Development asset linked to CERo Therapeutics in public FDA and regional records.

  67. Development asset linked to CERo Therapeutics in public FDA and regional records.

  68. Development asset linked to CERo Therapeutics in public FDA and regional records.

  69. Development asset linked to CERo Therapeutics in public FDA and regional records.

  70. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha modulator
  71. tarlatamab

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in CERo Therapeutics's portfolio. Molecular target: Delta-like protein 3.

    Target
    Delta-like protein 3
    Mechanism
    Delta-like protein 3 binding agent
  72. temozolomide

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  73. Development asset linked to CERo Therapeutics in public FDA and regional records. Molecular target: Hepatocyte growth factor receptor.

    Target
    Hepatocyte growth factor receptor
    Mechanism
    Hepatocyte growth factor receptor inhibitor
  74. Development asset linked to CERo Therapeutics in public FDA and regional records.

  75. topotecan

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in CERo Therapeutics's portfolio. Mechanism: DNA topoisomerase I, mitochondrial inhibitor.

    Mechanism
    DNA topoisomerase I, mitochondrial inhibitor
  76. US regulatory status: approved. Molecular target: DNA topoisomerase 1.

    Target
    DNA topoisomerase 1
    Mechanism
    DNA topoisomerase I, mitochondrial inhibitor
  77. Development asset linked to CERo Therapeutics in public FDA and regional records.