Wednesday, July 8, 2026

Drug profile · INN

tamoxifen citrate

tamoxifen citrate (TAMOXIFEN CITRATE) is a estrogen receptor alpha modulator. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 4
News articles 0
Drug details — tamoxifen citrate
US status
approved
Class
Route
ORAL
Patents
0
Programs
4
Data quality
0.89

Quick answer

tamoxifen citrate (TAMOXIFEN CITRATE) is a estrogen receptor alpha modulator. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN tamoxifen citrate
Brand TAMOXIFEN CITRATE
Mechanism Estrogen receptor alpha modulator
Target Estrogen receptor
Route ORAL
Formulation SOLUTION

Mechanism of action

Estrogen receptor alpha modulator

Primary target: Estrogen receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. D8535C00001 Phase 3 · AstraZeneca · ER+/HER2- Early Breast Cancer
  2. Tamoxifen Phase 3 · Chinese Academy of · Breast Cancer Female
  3. ICO-N-2013-03 Phase 2 · CERo Therapeutics · Breast cancer
  4. TAMOXIFEN Approved · Disc Medicine · Breast cancer

Related & competitor drugs

  1. estradiol Estrogen receptor alpha agonist
  2. estradiol valerate Estrogen receptor alpha agonist
  3. estrogens, conjugated synthetic a Estrogen receptor agonist
  4. estropipate Estrogen receptor alpha agonist
  5. ethinyl estradiol Estrogen receptor alpha agonist
  6. fulvestrant Antineoplastic and immunomodulating agents (L02)

Frequently asked questions

What is tamoxifen citrate?

tamoxifen citrate (TAMOXIFEN CITRATE) is a estrogen receptor alpha modulator. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for tamoxifen citrate?

TAMOXIFEN CITRATE is a marketed brand name for tamoxifen citrate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of tamoxifen citrate?

tamoxifen citrate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.