Friday, July 10, 2026

Drug profile · INN

mesalazine

mesalazine (ASACOL) is a arachidonate 5-lipoxygenase inhibitor. Associated with Ferring Pharmaceuticals.

TGA: approved PMDA: approved NMPA: clinical trials
Patents linked 0
Pipeline programs 15
News articles 0
Drug details — mesalazine

Quick answer

mesalazine (ASACOL) is a arachidonate 5-lipoxygenase inhibitor. Associated with Ferring Pharmaceuticals.

Key facts

INN mesalazine
Brand ASACOL
Mechanism Arachidonate 5-lipoxygenase inhibitor
Target Polyunsaturated fatty acid 5-lipoxygenase

Mechanism of action

Arachidonate 5-lipoxygenase inhibitor

Primary target: Polyunsaturated fatty acid 5-lipoxygenase

Approval history

Authority Status Date
TGA approved
PMDA approved
NMPA clinical trials

Pipeline programs

  1. Asacol® Phase 3 · Tillotts Pharma AG · Active Ulcerative Colitis
  2. Delayed and extended release mesalazine Phase 3 · Takeda · Colitis, Ulcerative
  3. MMX Mesalamine/Mesalazine (Low Dose) Phase 3 · Takeda · Ulcerative Colitis
  4. SPD476 (mesalazine) Phase 3 · Takeda · Colitis, Ulcerative
  5. SPD476-302 Phase 3 · Takeda · Ulcerative Colitis
  6. SPD476-314 Phase 3 · Takeda · Diverticulitis
  7. mesalazine (Asacol®) Phase 3 · Cardiff Oncology · Ulcerative Colitis
  8. Pentasa Sachet depotgranulat for Lynch syndrome, which is increa… Phase 2 · George Institute for · Lynch syndrome, which is increasing the risk of developing c

Related & competitor drugs

  1. meclofenamate sodium Arachidonate 5-lipoxygenase inhibitor
  2. mesalamine Arachidonate 5-lipoxygenase inhibitor
  3. zileuton Arachidonate 5-lipoxygenase inhibitor
  4. balsalazide disodium Cyclooxygenase inhibitor
  5. olsalazine sodium Arachidonate 5-lipoxygenase inhibitor
  6. sulfasalazine Arachidonate 5-lipoxygenase inhibitor

Frequently asked questions

What is mesalazine?

mesalazine (ASACOL) is a arachidonate 5-lipoxygenase inhibitor. Associated with Ferring Pharmaceuticals.

What is the brand name for mesalazine?

ASACOL is a marketed brand name for mesalazine. Check FDA Drugs@FDA for the current US label holder and prescribing information.