Wednesday, July 8, 2026

Drug profile · INN

cetrorelix acetate

cetrorelix acetate (CETRORELIX ACETATE) is a gonadotropin-releasing hormone receptor antagonist. Associated with Teva Pharma GmbH. Route of administration: subcutaneous. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 20
Pipeline programs 3
News articles 0
Drug details — cetrorelix acetate
US status
approved
Class
Route
SUBCUTANEOUS
Patents
20
Programs
3
Data quality
0.89

Quick answer

cetrorelix acetate (CETRORELIX ACETATE) is a gonadotropin-releasing hormone receptor antagonist. Associated with Teva Pharma GmbH. Route of administration: subcutaneous. Current US regulatory status: approved.

Key facts

INN cetrorelix acetate
Brand CETRORELIX ACETATE
Mechanism Gonadotropin-releasing hormone receptor antagonist
Target Gonadotropin-releasing hormone receptor
Route SUBCUTANEOUS
Formulation POWDER

Mechanism of action

Gonadotropin-releasing hormone receptor antagonist

Primary target: Gonadotropin-releasing hormone receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. ICO-N-2013-03 Phase 2 · CERo Therapeutics · Breast cancer
  2. Cetrorelix Acetate Approved · United Therapeutics Europe · Infertility
  3. Generic cetrorelix acetate Unknown · NORTHWEST BIOTHERAPEUTICS · Infertility

Related & competitor drugs

  1. elagolix Gonadotropin-releasing hormone receptor antagonist
  2. ganirelix acetate Gonadotropin-releasing hormone receptor antagonist
  3. leuprolide acetate Gonadotropin-releasing hormone receptor agonist
  4. abarelix Gonadotropin-releasing hormone receptor antagonist
  5. degarelix acetate Gonadotropin-releasing hormone receptor antagonist
  6. elagolix sodium Gonadotropin-releasing hormone receptor antagonist
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Frequently asked questions

What is cetrorelix acetate?

cetrorelix acetate (CETRORELIX ACETATE) is a gonadotropin-releasing hormone receptor antagonist. Associated with Teva Pharma GmbH. Route of administration: subcutaneous. Current US regulatory status: approved.

What is the brand name for cetrorelix acetate?

CETRORELIX ACETATE is a marketed brand name for cetrorelix acetate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of cetrorelix acetate?

cetrorelix acetate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.