Wednesday, July 22, 2026

pharma · Asthma · Respiratory Syncytial Virus Infections

GSK Glaxo Smith

GSK Glaxo Smith drug portfolio — 143 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

637 r Aulnois, Saint Amand les Eaux, 59 59230, FR, SAINT-AMAND LES EAUX HQ
30 Employees
NMPA registrant Type
Company details
Status
Public
HQ
637 r Aulnois, Saint Amand les Eaux, 59 59230, FR, SAINT-AMAND LES EAUX
Employees
30
Programs
4
Drugs
143
Patents
0
Intelligence · Drug Pipeline

GSK Glaxo Smith pipeline

Portfolio lens on 143 drugs and development assets — regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

GSK Glaxo Smith drug portfolio — 143 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

143 compounds
  1. Development asset linked to GSK Glaxo Smith in public FDA and regional records.

  2. US regulatory status: approved. Molecular target: Fatty-acid amide hydrolase 1.

    Target
    Fatty-acid amide hydrolase 1
    Mechanism
    Cyclooxygenase inhibitor
  3. US regulatory status: approved. Molecular target: DNA polymerase catalytic subunit.

    Target
    DNA polymerase catalytic subunit
    Mechanism
    Human herpesvirus 1 DNA polymerase inhibitor
  4. adalimumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Tumor necrosis factor.

    Target
    Tumor necrosis factor
    Mechanism
    TNF-alpha inhibitor
  5. adefovir dipivoxil

    Antiinfectives for systemic use (J05)

    US regulatory status: approved. Molecular target: DNA polymerase/reverse transcriptase.

    Target
    DNA polymerase/reverse transcriptase
    Mechanism
    DNA polymerase/reverse transcriptase inhibitor
  6. albiglutide

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Glucagon-like peptide 1 receptor.

    Target
    Glucagon-like peptide 1 receptor
    Mechanism
    Glucagon-like peptide 1 receptor agonist
  7. US regulatory status: approved. Molecular target: Beta-2 adrenergic receptor.

    Target
    Beta-2 adrenergic receptor
    Mechanism
    Beta-2 adrenergic receptor agonist
  8. US regulatory status: approved. Molecular target: Beta-2 adrenergic receptor.

    Target
    Beta-2 adrenergic receptor
    Mechanism
    Beta-2 adrenergic receptor agonist
  9. US regulatory status: approved.

  10. US regulatory status: approved. Molecular target: Interleukin-2 receptor.

    Target
    Interleukin-2 receptor
    Mechanism
    Interleukin-2 receptor agonist
  11. US regulatory status: approved. Molecular target: 5-hydroxytryptamine receptor 3A.

    Target
    5-hydroxytryptamine receptor 3A
    Mechanism
    Serotonin 3a (5-HT3a) receptor antagonist
  12. US regulatory status: approved. Molecular target: Bacterial penicillin-binding protein.

    Target
    Bacterial penicillin-binding protein
    Mechanism
    Bacterial penicillin-binding protein inhibitor
  13. US regulatory status: approved. Molecular target: Histamine H1 receptor.

    Target
    Histamine H1 receptor
    Mechanism
    Histamine H1 receptor antagonist
  14. Various (V09) compound in GSK Glaxo Smith's portfolio. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  15. aprepitant

    Alimentary tract and metabolism (A04)

    US regulatory status: approved. Molecular target: Substance-P receptor.

    Target
    Substance-P receptor
    Mechanism
    Neurokinin 1 receptor antagonist
  16. asenapine

    Nervous system (N05)

    US regulatory status: approved. Mechanism: Serotonin 2a (5-HT2a) receptor antagonist.

    Mechanism
    Serotonin 2a (5-HT2a) receptor antagonist
  17. US regulatory status: approved. Molecular target: Cyclooxygenase.

    Target
    Cyclooxygenase
    Mechanism
    Cyclooxygenase inhibitor
  18. US regulatory status: approved. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  19. belantamab mafodotin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in GSK Glaxo Smith's portfolio. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tumor necrosis factor receptor superfamily member 17 binding agent
  20. US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  21. belimumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Tumor necrosis factor ligand superfamily member 13B.

    Target
    Tumor necrosis factor ligand superfamily member 13B
    Mechanism
    Tumor necrosis factor ligand superfamily member 13B inhibitor
  22. benralizumab

    Respiratory system (R03)

    US regulatory status: approved. Molecular target: Interleukin-5 receptor subunit alpha.

    Target
    Interleukin-5 receptor subunit alpha
    Mechanism
    Interleukin-5 receptor subunit alpha inhibitor
  23. bevacizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Vascular endothelial growth factor A, long form.

    Target
    Vascular endothelial growth factor A, long form
    Mechanism
    Vascular endothelial growth factor A inhibitor
  24. bortezomib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  25. budesonide

    Alimentary tract and metabolism (A07)

    US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  26. US regulatory status: approved.

  27. capecitabine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  28. US regulatory status: approved. Molecular target: Sodium channel alpha subunit.

    Target
    Sodium channel alpha subunit
    Mechanism
    Sodium channel alpha subunit blocker
  29. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  30. carfilzomib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  31. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  32. Development asset linked to GSK Glaxo Smith in public FDA and regional records. Molecular target: Substance-P receptor.

    Target
    Substance-P receptor
    Mechanism
    Neurokinin 1 receptor antagonist
  33. US regulatory status: approved. Molecular target: Ferriprotoporphyrin IX.

    Target
    Ferriprotoporphyrin IX
    Mechanism
    Ferriprotoporphyrin IX binding agent
  34. US regulatory status: approved. Molecular target: Bacterial DNA gyrase.

    Target
    Bacterial DNA gyrase
    Mechanism
    Bacterial DNA gyrase inhibitor
  35. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  36. US regulatory status: approved. Molecular target: GABA-A receptor; anion channel.

    Target
    GABA-A receptor; anion channel
    Mechanism
    GABA-A receptor; anion channel positive allosteric modulator
  37. covid-19 mrna vaccine

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in GSK Glaxo Smith's portfolio. Molecular target: Spike glycoprotein.

    Target
    Spike glycoprotein
    Mechanism
    Spike glycoprotein vaccine antigen
  38. dabrafenib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in GSK Glaxo Smith's portfolio. Mechanism: Serine/threonine-protein kinase B-raf inhibitor.

    Mechanism
    Serine/threonine-protein kinase B-raf inhibitor
  39. daprodustat

    Blood and blood forming organs (B03)

    US regulatory status: approved. Molecular target: Hypoxia-inducible factor prolyl hydroxylase.

    Target
    Hypoxia-inducible factor prolyl hydroxylase
    Mechanism
    Hypoxia-inducible factor prolyl hydroxylase inhibitor
  40. daratumumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1.

    Target
    ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
    Mechanism
    Lymphocyte differentiation antigen CD38 inhibitor
  41. denosumab

    Musculo-skeletal system (M05)

    US regulatory status: approved. Molecular target: Tumor necrosis factor ligand superfamily member 11.

    Target
    Tumor necrosis factor ligand superfamily member 11
    Mechanism
    Tumor necrosis factor ligand superfamily member 11 inhibitor
  42. depemokimab

    Respiratory system (R03)

    Respiratory system (R03) compound in GSK Glaxo Smith's portfolio. Molecular target: Interleukin-5.

    Target
    Interleukin-5
    Mechanism
    Interleukin-5 inhibitor
  43. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  44. dexamethasone phosphate

    Systemic hormonal preparations (H02)

    Systemic hormonal preparations (H02) compound in GSK Glaxo Smith's portfolio.

  45. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  46. docetaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  47. dostarlimab

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in GSK Glaxo Smith's portfolio. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 antagonist
  48. US regulatory status: approved. Molecular target: Steroid 5-alpha-reductase.

    Target
    Steroid 5-alpha-reductase
    Mechanism
    Steroid 5-alpha-reductase inhibitor
  49. eltrombopag

    Blood and blood forming organs (B02)

    US regulatory status: approved. Mechanism: Thrombopoietin receptor agonist.

    Mechanism
    Thrombopoietin receptor agonist
  50. US regulatory status: approved. Molecular target: Thrombopoietin receptor.

    Target
    Thrombopoietin receptor
    Mechanism
    Thrombopoietin receptor agonist
  51. enzalutamide

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  52. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  53. US regulatory status: approved. Molecular target: KCNQ (Kv7) potassium channel.

    Target
    KCNQ (Kv7) potassium channel
    Mechanism
    KCNQ (Kv7) potassium channel opener
  54. florbetaben (18f)

    Various (V09)

    Various (V09) compound in GSK Glaxo Smith's portfolio. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  55. US regulatory status: approved. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  56. US regulatory status: approved. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  57. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  58. US regulatory status: approved. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  59. Development asset linked to GSK Glaxo Smith in public FDA and regional records.

  60. fluticasone furoate

    Respiratory system (R03)

    US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  61. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  62. formoterol

    Respiratory system (R03)

    Respiratory system (R03) compound in GSK Glaxo Smith's portfolio. Mechanism: Beta-2 adrenergic receptor agonist.

    Mechanism
    Beta-2 adrenergic receptor agonist
  63. US regulatory status: approved. Molecular target: Sulfonylurea receptor 1, Kir6.2.

    Target
    Sulfonylurea receptor 1, Kir6.2
    Mechanism
    Sulfonylurea receptor 1, Kir6.2 blocker
  64. herpes zoster vaccine (recombinant, adjuvanted)

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in GSK Glaxo Smith's portfolio. Molecular target: Envelope glycoprotein E.

    Target
    Envelope glycoprotein E
    Mechanism
    Envelope glycoprotein E vaccine antigen
  65. Development asset linked to GSK Glaxo Smith in public FDA and regional records. Mechanism: Mu opioid receptor agonist.

    Mechanism
    Mu opioid receptor agonist
  66. insulin glargine

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  67. insulin human

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  68. isatuximab

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in GSK Glaxo Smith's portfolio. Molecular target: ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1.

    Target
    ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
    Mechanism
    Lymphocyte differentiation antigen CD38 inhibitor
  69. lamivudine

    Antiinfectives for systemic use (J05)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  70. US regulatory status: approved. Molecular target: Sodium channel alpha subunit.

    Target
    Sodium channel alpha subunit
    Mechanism
    Sodium channel alpha subunit blocker
  71. lapatinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in GSK Glaxo Smith's portfolio. Mechanism: Receptor protein-tyrosine kinase erbB-2 inhibitor.

    Mechanism
    Receptor protein-tyrosine kinase erbB-2 inhibitor
  72. lenalidomide

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: CRL4(CRBN) E3 ubiquitin ligase.

    Target
    CRL4(CRBN) E3 ubiquitin ligase
    Mechanism
    CRL4(CRBN) E3 ubiquitin ligase inhibitor
  73. Development asset linked to GSK Glaxo Smith in public FDA and regional records.

  74. luspatercept

    Blood and blood forming organs (B03)

    Blood and blood forming organs (B03) compound in GSK Glaxo Smith's portfolio. Molecular target: Transforming growth factor beta.

    Target
    Transforming growth factor beta
    Mechanism
    Transforming growth factor beta inhibitor
  75. US regulatory status: approved. Molecular target: Transforming growth factor beta.

    Target
    Transforming growth factor beta
    Mechanism
    Transforming growth factor beta inhibitor
  76. US regulatory status: approved. Molecular target: Acetylcholinesterase.

    Target
    Acetylcholinesterase
    Mechanism
    Acetylcholinesterase inhibitor
  77. mepolizumab

    Respiratory system (R03)

    US regulatory status: approved. Molecular target: Interleukin-5.

    Target
    Interleukin-5
    Mechanism
    Interleukin-5 inhibitor
  78. Development asset linked to GSK Glaxo Smith in public FDA and regional records. Molecular target: Tyrosine-protein kinase JAK1.

    Target
    Tyrosine-protein kinase JAK1
    Mechanism
    Tyrosine-protein kinase JAK1 inhibitor
  79. Development asset linked to GSK Glaxo Smith in public FDA and regional records. Mechanism: Cysteinyl leukotriene receptor 1 antagonist.

    Mechanism
    Cysteinyl leukotriene receptor 1 antagonist
  80. US regulatory status: approved. Molecular target: Isoleucine--tRNA ligase.

    Target
    Isoleucine--tRNA ligase
    Mechanism
    Isoleucyl-tRNA synthetase inhibitor
  81. niraparib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in GSK Glaxo Smith's portfolio. Molecular target: Poly [ADP-ribose] polymerase 2.

    Target
    Poly [ADP-ribose] polymerase 2
    Mechanism
    Poly [ADP-ribose] polymerase-1 inhibitor
  82. Development asset linked to GSK Glaxo Smith in public FDA and regional records. Molecular target: Poly [ADP-ribose] polymerase 2.

    Target
    Poly [ADP-ribose] polymerase 2
    Mechanism
    Poly [ADP-ribose] polymerase 2 inhibitor
  83. nirogacestat

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in GSK Glaxo Smith's portfolio. Molecular target: Gamma-secretase.

    Target
    Gamma-secretase
    Mechanism
    Gamma-secretase inhibitor
  84. orlistat

    Alimentary tract and metabolism (A08)

    US regulatory status: approved. Molecular target: Gastric triacylglycerol lipase.

    Target
    Gastric triacylglycerol lipase
    Mechanism
    Pancreatic lipase inhibitor
  85. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  86. pazopanib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in GSK Glaxo Smith's portfolio. Mechanism: Vascular endothelial growth factor receptor inhibitor.

    Mechanism
    Vascular endothelial growth factor receptor inhibitor
  87. pembrolizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  88. US regulatory status: approved. Molecular target: Dihydrofolate reductase.

    Target
    Dihydrofolate reductase
    Mechanism
    Thymidylate synthase inhibitor
  89. pioglitazone

    Alimentary tract and metabolism (A10)

    Alimentary tract and metabolism (A10) compound in GSK Glaxo Smith's portfolio. Mechanism: Peroxisome proliferator-activated receptor gamma agonist.

    Mechanism
    Peroxisome proliferator-activated receptor gamma agonist
  90. US regulatory status: approved. Molecular target: Peroxisome proliferator-activated receptor gamma.

    Target
    Peroxisome proliferator-activated receptor gamma
    Mechanism
    Peroxisome proliferator-activated receptor gamma agonist
  91. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  92. pomalidomide

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: CRL4(CRBN) E3 ubiquitin ligase.

    Target
    CRL4(CRBN) E3 ubiquitin ligase
    Mechanism
    CRL4(CRBN) E3 ubiquitin ligase inhibitor
  93. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  94. retigabine

    Nervous system (N03)

    Nervous system (N03) compound in GSK Glaxo Smith's portfolio. Molecular target: KCNQ (Kv7) potassium channel.

    Target
    KCNQ (Kv7) potassium channel
    Mechanism
    KCNQ (Kv7) potassium channel opener
  95. Development asset linked to GSK Glaxo Smith in public FDA and regional records. Mechanism: Vascular endothelial growth factor receptor 2 inhibitor.

    Mechanism
    Vascular endothelial growth factor receptor 2 inhibitor
  96. rosiglitazone

    Alimentary tract and metabolism (A10)

    Alimentary tract and metabolism (A10) compound in GSK Glaxo Smith's portfolio. Molecular target: Peroxisome proliferator-activated receptor gamma.

    Target
    Peroxisome proliferator-activated receptor gamma
    Mechanism
    Peroxisome proliferator-activated receptor gamma agonist
  97. rotavirus vaccine

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in GSK Glaxo Smith's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  98. rotavirus vaccine, live

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in GSK Glaxo Smith's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  99. salmeterol

    Respiratory system (R03)

    Respiratory system (R03) compound in GSK Glaxo Smith's portfolio. Mechanism: Beta-2 adrenergic receptor agonist.

    Mechanism
    Beta-2 adrenergic receptor agonist
  100. Development asset linked to GSK Glaxo Smith in public FDA and regional records.

  101. shingles (herpes zoster) vaccine (live)

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in GSK Glaxo Smith's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  102. Development asset linked to GSK Glaxo Smith in public FDA and regional records. Mechanism: Adrenergic receptor alpha-1 antagonist.

    Mechanism
    Adrenergic receptor alpha-1 antagonist
  103. topotecan

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in GSK Glaxo Smith's portfolio. Mechanism: DNA topoisomerase I, mitochondrial inhibitor.

    Mechanism
    DNA topoisomerase I, mitochondrial inhibitor
  104. US regulatory status: approved. Molecular target: DNA topoisomerase 1.

    Target
    DNA topoisomerase 1
    Mechanism
    DNA topoisomerase I, mitochondrial inhibitor
  105. ulipristal acetate

    Genito-urinary system and sex hormones (G03)

    US regulatory status: approved. Molecular target: Progesterone receptor.

    Target
    Progesterone receptor
    Mechanism
    Progesterone receptor modulator
  106. umeclidinium

    Respiratory system (R03)

    Respiratory system (R03) compound in GSK Glaxo Smith's portfolio. Mechanism: Muscarinic acetylcholine receptor M3 antagonist.

    Mechanism
    Muscarinic acetylcholine receptor M3 antagonist
  107. US regulatory status: approved. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  108. zanamivir

    Antiinfectives for systemic use (J05)

    US regulatory status: approved. Molecular target: Neuraminidase.

    Target
    Neuraminidase
    Mechanism
    Neuraminidase inhibitor