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Celgene

Celgene drug portfolio — 80 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Summit, USA HQ
2,104 Employees
EMA registrant Type
Company details
Status
Public
HQ
Summit, USA
Employees
2,104
Programs
45
Drugs
91
Patents
0
Intelligence · Drug Pipeline

Celgene pipeline

Portfolio lens on 80 drugs and development assets — regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

Celgene drug portfolio — 80 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

80 compounds
  1. abiraterone

    Antineoplastic and immunomodulating agents (L02)

    Antineoplastic and immunomodulating agents (L02) compound in Celgene's portfolio. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Steroid 5-alpha-reductase inhibitor
  2. US regulatory status: approved. Molecular target: DNA polymerase catalytic subunit.

    Target
    DNA polymerase catalytic subunit
    Mechanism
    Human herpesvirus 1 DNA polymerase inhibitor
  3. Development asset linked to Celgene in public FDA and regional records.

  4. apixaban

    Blood and blood forming organs (B01)

    US regulatory status: approved. Molecular target: Coagulation factor X.

    Target
    Coagulation factor X
    Mechanism
    Coagulation factor X inhibitor
  5. Development asset linked to Celgene in public FDA and regional records.

  6. azacitidine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA (cytosine-5)-methyltransferase 1.

    Target
    DNA (cytosine-5)-methyltransferase 1
    Mechanism
    DNA (cytosine-5)-methyltransferase 3A inhibitor
  7. Development asset linked to Celgene in public FDA and regional records.

  8. bortezomib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  9. busulfan

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  10. Development asset linked to Celgene in public FDA and regional records.

  11. Development asset linked to Celgene in public FDA and regional records.

  12. Development asset linked to Celgene in public FDA and regional records.

  13. carfilzomib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  14. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  15. Development asset linked to Celgene in public FDA and regional records.

  16. Development asset linked to Celgene in public FDA and regional records.

  17. Development asset linked to Celgene in public FDA and regional records.

  18. Development asset linked to Celgene in public FDA and regional records.

  19. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  20. Development asset linked to Celgene in public FDA and regional records.

  21. Development asset linked to Celgene in public FDA and regional records.

  22. Development asset linked to Celgene in public FDA and regional records.

  23. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  24. US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Progesterone receptor agonist
  25. daratumumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1.

    Target
    ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
    Mechanism
    Lymphocyte differentiation antigen CD38 inhibitor
  26. dexamethasone phosphate

    Systemic hormonal preparations (H02)

    Systemic hormonal preparations (H02) compound in Celgene's portfolio.

  27. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  28. docetaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  29. doxorubicin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Celgene's portfolio. Mechanism: DNA topoisomerase II alpha inhibitor.

    Mechanism
    DNA topoisomerase II alpha inhibitor
  30. doxorubicin hydrochloride

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA topoisomerase II alpha inhibitor
  31. edoxaban

    Blood and blood forming organs (B01)

    US regulatory status: approved. Mechanism: Coagulation factor X inhibitor.

    Mechanism
    Coagulation factor X inhibitor
  32. elotuzumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: SLAM family member 7.

    Target
    SLAM family member 7
    Mechanism
    SLAM family member 7 inhibitor
  33. US regulatory status: approved. Molecular target: T cell surface glycoprotein CD3.

    Target
    T cell surface glycoprotein CD3
    Mechanism
    T cell surface glycoprotein CD3 binding agent
  34. US regulatory status: approved. Molecular target: Isocitrate dehydrogenase [NADP], mitochondrial.

    Target
    Isocitrate dehydrogenase [NADP], mitochondrial
    Mechanism
    Isocitrate dehydrogenase [NADP], mitochondrial inhibitor
  35. enzalutamide

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  36. US regulatory status: approved. Molecular target: DNA topoisomerase II.

    Target
    DNA topoisomerase II
    Mechanism
    DNA topoisomerase II inhibitor
  37. Development asset linked to Celgene in public FDA and regional records.

  38. fedratinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Celgene's portfolio. Molecular target: Tyrosine-protein kinase JAK2.

    Target
    Tyrosine-protein kinase JAK2
    Mechanism
    Tyrosine-protein kinase JAK2 inhibitor
  39. filgrastim

    Antineoplastic and immunomodulating agents (L03)

    US regulatory status: approved. Molecular target: Granulocyte colony-stimulating factor receptor.

    Target
    Granulocyte colony-stimulating factor receptor
    Mechanism
    Granulocyte colony stimulating factor receptor agonist
  40. Development asset linked to Celgene in public FDA and regional records.

  41. US regulatory status: approved. Molecular target: DNA polymerase (alpha/delta/epsilon).

    Target
    DNA polymerase (alpha/delta/epsilon)
    Mechanism
    DNA polymerase (alpha/delta/epsilon) inhibitor
  42. Development asset linked to Celgene in public FDA and regional records.

  43. US regulatory status: approved. Molecular target: Muscarinic acetylcholine receptor M1.

    Target
    Muscarinic acetylcholine receptor M1
    Mechanism
    Muscarinic acetylcholine receptor M1 antagonist
  44. hydroxycarbamide

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Celgene's portfolio. Molecular target: Ribonucleoside-diphosphate reductase RR1.

    Target
    Ribonucleoside-diphosphate reductase RR1
    Mechanism
    Ribonucleoside-diphosphate reductase RR1 inhibitor
  45. idecabtagene vicleucel

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Celgene's portfolio. Molecular target: Tumor necrosis factor receptor superfamily member 17.

    Target
    Tumor necrosis factor receptor superfamily member 17
    Mechanism
    Tumor necrosis factor receptor superfamily member 17 binding agent
  46. Development asset linked to Celgene in public FDA and regional records.

  47. Development asset linked to Celgene in public FDA and regional records.

  48. Development asset linked to Celgene in public FDA and regional records.

  49. Development asset linked to Celgene in public FDA and regional records.

  50. ivosidenib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Isocitrate dehydrogenase [NADP] cytoplasmic.

    Target
    Isocitrate dehydrogenase [NADP] cytoplasmic
    Mechanism
    Isocitrate dehydrogenase [NADP] cytoplasmic inhibitor
  51. ixazomib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Celgene's portfolio. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteasome inhibitor
  52. lenalidomide

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: CRL4(CRBN) E3 ubiquitin ligase.

    Target
    CRL4(CRBN) E3 ubiquitin ligase
    Mechanism
    CRL4(CRBN) E3 ubiquitin ligase inhibitor
  53. lisocabtagene maraleucel

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Celgene's portfolio. Molecular target: B-lymphocyte antigen CD19.

    Target
    B-lymphocyte antigen CD19
    Mechanism
    B-lymphocyte antigen CD19 binding agent
  54. luspatercept

    Blood and blood forming organs (B03)

    Blood and blood forming organs (B03) compound in Celgene's portfolio. Molecular target: Transforming growth factor beta.

    Target
    Transforming growth factor beta
    Mechanism
    Transforming growth factor beta inhibitor
  55. US regulatory status: approved. Molecular target: Transforming growth factor beta.

    Target
    Transforming growth factor beta
    Mechanism
    Transforming growth factor beta inhibitor
  56. Development asset linked to Celgene in public FDA and regional records.

  57. Development asset linked to Celgene in public FDA and regional records.

  58. Development asset linked to Celgene in public FDA and regional records.

  59. ozanimod

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Sphingosine 1-phosphate receptor 5.

    Target
    Sphingosine 1-phosphate receptor 5
    Mechanism
    Sphingosine 1-phosphate receptor Edg-1 modulator
  60. US regulatory status: approved. Molecular target: Sphingosine 1-phosphate receptor 1.

    Target
    Sphingosine 1-phosphate receptor 1
    Mechanism
    Sphingosine 1-phosphate receptor Edg-1 modulator
  61. pegfilgrastim

    Antineoplastic and immunomodulating agents (L03)

    US regulatory status: approved. Molecular target: Granulocyte colony-stimulating factor receptor.

    Target
    Granulocyte colony-stimulating factor receptor
    Mechanism
    Granulocyte colony stimulating factor receptor agonist
  62. Development asset linked to Celgene in public FDA and regional records.

  63. pembrolizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  64. Development asset linked to Celgene in public FDA and regional records.

  65. pomalidomide

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: CRL4(CRBN) E3 ubiquitin ligase.

    Target
    CRL4(CRBN) E3 ubiquitin ligase
    Mechanism
    CRL4(CRBN) E3 ubiquitin ligase inhibitor
  66. Development asset linked to Celgene in public FDA and regional records.

  67. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  68. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  69. Development asset linked to Celgene in public FDA and regional records.

  70. Development asset linked to Celgene in public FDA and regional records.

  71. rituximab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: B-lymphocyte antigen CD20.

    Target
    B-lymphocyte antigen CD20
    Mechanism
    B-lymphocyte antigen CD20 binding agent
  72. ruxolitinib

    Dermatologicals (D11)

    US regulatory status: approved. Mechanism: Tyrosine-protein kinase JAK2 inhibitor.

    Mechanism
    Tyrosine-protein kinase JAK2 inhibitor
  73. Development asset linked to Celgene in public FDA and regional records.

  74. Development asset linked to Celgene in public FDA and regional records.

  75. Development asset linked to Celgene in public FDA and regional records.

  76. Development asset linked to Celgene in public FDA and regional records.

  77. Development asset linked to Celgene in public FDA and regional records.