Wednesday, July 8, 2026

Drug profile · INN

edoxaban

edoxaban (LIXIANA) is a coagulation factor x inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved EMA: approved PMDA: approved Blood and blood forming organs (B01) B01AF03
US status approved
Patents linked 20
Pipeline programs 12
News articles 0
Drug details — edoxaban
US status
approved
Class
Blood and blood forming organs (B01)
Route
ORAL
Patents
20
Programs
12
Data quality
0.84

Quick answer

edoxaban (LIXIANA) is a coagulation factor x inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN edoxaban
Brand LIXIANA
Mechanism Coagulation factor X inhibitor
Therapeutic class Blood and blood forming organs (B01)
Route ORAL
Formulation TABLET
ATC code B01AF03

Mechanism of action

Coagulation factor X inhibitor

Approval history

Authority Status Date
FDA approved
EMA approved
PMDA approved

Pipeline programs

  1. BB2121-MM-003 Phase 3 · Celgene · Multiple myeloma (MM) with at least 2 prior therapies includ
  2. D9604C00001 Phase 3 · AstraZeneca · Reversal of anticoagulation effect in patients on a FXa inhi
  3. Edoxaban Phase 3 · Daiichi Sankyo US · Cardiac Disease
  4. edoxaban tosylate(DU-176b) Phase 3 · Daiichi Sankyo US · Venous Thromboembolism
  5. CARTBCMA-HCB-01 Phase 2 · George Institute for · Multiple Myeloma
  6. EAE 115 Phase 2 · Createrna Science and · Multiple myeloma patients who received one prior line of the
  7. Bioequivalence clinical trial of two formulations of edoxaban. Phase 1 · Tillomed Laboratories · Healthy volunteers
  8. UECHUP-EDO/25-2 Phase 1 · Tillomed Laboratories · Healthy volunteers

Related & competitor drugs

  1. apixaban Blood and blood forming organs (B01)
  2. berotralstat Blood and blood forming organs (B06)
  3. bivalirudin Blood and blood forming organs (B01)
  4. c1 inhibitor (human) Blood and blood forming organs (B06)
  5. clopidogrel Blood and blood forming organs (B01)
  6. dabigatran etexilate Blood and blood forming organs (B01)

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Frequently asked questions

What is edoxaban?

edoxaban (LIXIANA) is a coagulation factor x inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for edoxaban?

LIXIANA is a marketed brand name for edoxaban. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of edoxaban?

edoxaban has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.