Saturday, July 11, 2026

Drug profile · INN

fedratinib

fedratinib (INREBIC) is a tyrosine-protein kinase jak2 inhibitor. Associated with Bristol-Myers Squibb Australia Pty Ltd.

EMA: approved TGA: approved Antineoplastic and immunomodulating agents (L01) L01EJ02
Patents linked 0
Pipeline programs 3
News articles 0
Drug details — fedratinib
Class
Antineoplastic and immunomodulating agents (L01)
Route
Patents
0
Programs
3
Data quality
0.83

Quick answer

fedratinib (INREBIC) is a tyrosine-protein kinase jak2 inhibitor. Associated with Bristol-Myers Squibb Australia Pty Ltd.

Key facts

INN fedratinib
Brand INREBIC
Mechanism Tyrosine-protein kinase JAK2 inhibitor
Target Tyrosine-protein kinase JAK2
Therapeutic class Antineoplastic and immunomodulating agents (L01)
ATC code L01EJ02

Mechanism of action

Tyrosine-protein kinase JAK2 inhibitor

Primary target: Tyrosine-protein kinase JAK2

Approval history

Authority Status Date
EMA approved
TGA approved

Pipeline programs

  1. FEDR-MF-002 Phase 3 · Celgene · Primary myelofibrosis, post-polycythemia vera myelofibrosis
  2. CA011-023 Phase 2 · Bristol-Myers Squibb Australia · DIPSS-Intermediate or High Risk Myelofibrosis
  3. FRACTION_2021 Phase 2 · George Institute for · Primary and secondary Myelofibrosis

Related & competitor drugs

  1. abiraterone acetate Antineoplastic and immunomodulating agents (L02)
  2. anagrelide Antineoplastic and immunomodulating agents (L01)
  3. apremilast Antineoplastic and immunomodulating agents (L04)
  4. arsenic trioxide Antineoplastic and immunomodulating agents (L01)
  5. axitinib Antineoplastic and immunomodulating agents (L01)
  6. azacitidine Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is fedratinib?

fedratinib (INREBIC) is a tyrosine-protein kinase jak2 inhibitor. Associated with Bristol-Myers Squibb Australia Pty Ltd.

What is the brand name for fedratinib?

INREBIC is a marketed brand name for fedratinib. Check FDA Drugs@FDA for the current US label holder and prescribing information.