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Takeda

Takeda drug portfolio — 200 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Cambridge, USA HQ
1993 Founded
1,617 Employees
NMPA registrant Type
Company details
Intelligence · Drug Pipeline

Takeda pipeline

Portfolio lens on 200 drugs and development assets — regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

Takeda drug portfolio — 200 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

200 compounds
  1. Development asset linked to Takeda in public FDA and regional records.

  2. Development asset linked to Takeda in public FDA and regional records. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  3. Development asset linked to Takeda in public FDA and regional records.

  4. abacavir

    Antiinfectives for systemic use (J05)

    US regulatory status: approved.

  5. US regulatory status: approved. Molecular target: Fatty-acid amide hydrolase 1.

    Target
    Fatty-acid amide hydrolase 1
    Mechanism
    Cyclooxygenase inhibitor
  6. US regulatory status: approved. Molecular target: Bacterial urease.

    Target
    Bacterial urease
    Mechanism
    Bacterial urease inhibitor
  7. US regulatory status: approved. Molecular target: Sodium/potassium-transporting ATPase.

    Target
    Sodium/potassium-transporting ATPase
    Mechanism
    Sodium/potassium-transporting ATPase inhibitor
  8. adalimumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Tumor necrosis factor.

    Target
    Tumor necrosis factor
    Mechanism
    TNF-alpha inhibitor
  9. Development asset linked to Takeda in public FDA and regional records.

  10. Development asset linked to Takeda in public FDA and regional records.

  11. US regulatory status: approved. Molecular target: Placenta growth factor.

    Target
    Placenta growth factor
    Mechanism
    Placenta growth factor inhibitor
  12. agalsidase alfa

    Alimentary tract and metabolism (A16)

    Alimentary tract and metabolism (A16) compound in Takeda's portfolio. Molecular target: Globotriosylceramide.

    Target
    Globotriosylceramide
    Mechanism
    Globotriosylceramide hydrolytic enzyme
  13. agalsidase beta

    Alimentary tract and metabolism (A16)

    US regulatory status: approved. Molecular target: Globotriosylceramide.

    Target
    Globotriosylceramide
    Mechanism
    Globotriosylceramide hydrolytic enzyme
  14. US regulatory status: approved. Molecular target: Beta-2 adrenergic receptor.

    Target
    Beta-2 adrenergic receptor
    Mechanism
    Beta-2 adrenergic receptor agonist
  15. US regulatory status: approved.

  16. alogliptin

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Mechanism: Dipeptidyl peptidase IV inhibitor.

    Mechanism
    Dipeptidyl peptidase IV inhibitor
  17. alogliptin benzoate

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Dipeptidyl peptidase 4.

    Target
    Dipeptidyl peptidase 4
    Mechanism
    Dipeptidyl peptidase IV inhibitor
  18. alpha1-proteinase inhibitor (human)

    Blood and blood forming organs (B02)

    Blood and blood forming organs (B02) compound in Takeda's portfolio. Molecular target: Neutrophil elastase.

    Target
    Neutrophil elastase
    Mechanism
    Leukocyte elastase inhibitor
  19. Development asset linked to Takeda in public FDA and regional records.

  20. amifampridine

    Nervous system (N07)

    US regulatory status: approved. Molecular target: Voltage-gated potassium channel.

    Target
    Voltage-gated potassium channel
    Mechanism
    Voltage-gated potassium channel blocker
  21. US regulatory status: approved. Molecular target: Phosphodiesterase 4.

    Target
    Phosphodiesterase 4
    Mechanism
    Phosphodiesterase 4 inhibitor
  22. amlodipine

    Cardiovascular system (C09)

    Cardiovascular system (C09) compound in Takeda's portfolio. Mechanism: Voltage-gated L-type calcium channel blocker.

    Mechanism
    Voltage-gated L-type calcium channel blocker
  23. US regulatory status: approved. Molecular target: Voltage-gated L-type calcium channel.

    Target
    Voltage-gated L-type calcium channel
    Mechanism
    Voltage-gated L-type calcium channel blocker
  24. US regulatory status: approved. Molecular target: Bacterial penicillin-binding protein.

    Target
    Bacterial penicillin-binding protein
    Mechanism
    Bacterial penicillin-binding protein inhibitor
  25. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter releasing agent
  26. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter releasing agent
  27. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter releasing agent
  28. US regulatory status: approved. Molecular target: Bacterial penicillin-binding protein.

    Target
    Bacterial penicillin-binding protein
    Mechanism
    Bacterial penicillin-binding protein inhibitor
  29. US regulatory status: approved. Mechanism: Removal of necrotic tissue.

    Mechanism
    Removal of necrotic tissue
  30. anagrelide

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Takeda's portfolio. Mechanism: Phosphodiesterase 3 inhibitor.

    Mechanism
    Phosphodiesterase 3 inhibitor
  31. US regulatory status: approved. Molecular target: Phosphodiesterase 3.

    Target
    Phosphodiesterase 3
    Mechanism
    Phosphodiesterase 3 inhibitor
  32. Development asset linked to Takeda in public FDA and regional records.

  33. Development asset linked to Takeda in public FDA and regional records.

  34. Various (V09) compound in Takeda's portfolio. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  35. Development asset linked to Takeda in public FDA and regional records.

  36. apremilast

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Phosphodiesterase 4.

    Target
    Phosphodiesterase 4
    Mechanism
    Phosphodiesterase 4 inhibitor
  37. US regulatory status: approved. Mechanism: Supplement.

    Mechanism
    Supplement
  38. Development asset linked to Takeda in public FDA and regional records.

  39. US regulatory status: approved. Molecular target: Cyclooxygenase.

    Target
    Cyclooxygenase
    Mechanism
    Cyclooxygenase inhibitor
  40. Development asset linked to Takeda in public FDA and regional records. Mechanism: HMG-CoA reductase inhibitor.

    Mechanism
    HMG-CoA reductase inhibitor
  41. atropine sulfate

    Sensory organs (S01)

    US regulatory status: approved. Molecular target: Muscarinic acetylcholine receptor M1.

    Target
    Muscarinic acetylcholine receptor M1
    Mechanism
    Muscarinic acetylcholine receptor M3 antagonist
  42. Development asset linked to Takeda in public FDA and regional records.

  43. azacitidine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA (cytosine-5)-methyltransferase 1.

    Target
    DNA (cytosine-5)-methyltransferase 1
    Mechanism
    DNA (cytosine-5)-methyltransferase 3A inhibitor
  44. US regulatory status: approved. Molecular target: Type-1 angiotensin II receptor.

    Target
    Type-1 angiotensin II receptor
    Mechanism
    Type-1 angiotensin II receptor antagonist
  45. azilsartan medoxomil

    Cardiovascular system (C09)

    US regulatory status: approved. Mechanism: Type-1 angiotensin II receptor antagonist.

    Mechanism
    Type-1 angiotensin II receptor antagonist
  46. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  47. bevacizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Vascular endothelial growth factor A, long form.

    Target
    Vascular endothelial growth factor A, long form
    Mechanism
    Vascular endothelial growth factor A inhibitor
  48. binimetinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Dual specificity mitogen-activated protein kinase kinase 1.

    Target
    Dual specificity mitogen-activated protein kinase kinase 1
    Mechanism
    Dual specificity mitogen-activated protein kinase kinase 1 inhibitor
  49. Development asset linked to Takeda in public FDA and regional records.

  50. blinatumomab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: B-lymphocyte antigen CD19.

    Target
    B-lymphocyte antigen CD19
    Mechanism
    T cell surface glycoprotein CD3 cross-linking agent
  51. bortezomib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  52. Development asset linked to Takeda in public FDA and regional records.

  53. brentuximab vedotin

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  54. brigatinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: ALK tyrosine kinase receptor.

    Target
    ALK tyrosine kinase receptor
    Mechanism
    ALK tyrosine kinase receptor inhibitor
  55. budesonide

    Alimentary tract and metabolism (A07)

    US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  56. Development asset linked to Takeda in public FDA and regional records. Mechanism: Dopamine transporter inhibitor.

    Mechanism
    Dopamine transporter inhibitor
  57. c1 inhibitor (human)

    Blood and blood forming organs (B06)

    Blood and blood forming organs (B06) compound in Takeda's portfolio. Molecular target: Coagulation factor XI.

    Target
    Coagulation factor XI
    Mechanism
    Coagulation factor XI inhibitor
  58. cabozantinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Mechanism: Hepatocyte growth factor receptor inhibitor.

    Mechanism
    Hepatocyte growth factor receptor inhibitor
  59. caffeine

    Nervous system (N06)

    US regulatory status: approved. Molecular target: Adenosine receptor.

    Target
    Adenosine receptor
    Mechanism
    Adenosine receptor antagonist
  60. US regulatory status: approved. Molecular target: Vitamin D3 receptor.

    Target
    Vitamin D3 receptor
    Mechanism
    Vitamin D receptor agonist
  61. US regulatory status: approved.

  62. US regulatory status: approved. Mechanism: Dihydrofolate reductase inhibitor.

    Mechanism
    Dihydrofolate reductase inhibitor
  63. Development asset linked to Takeda in public FDA and regional records. Molecular target: Type-1 angiotensin II receptor.

    Target
    Type-1 angiotensin II receptor
    Mechanism
    Type-1 angiotensin II receptor antagonist
  64. US regulatory status: approved. Molecular target: Type-1 angiotensin II receptor.

    Target
    Type-1 angiotensin II receptor
    Mechanism
    Type-1 angiotensin II receptor antagonist
  65. Development asset linked to Takeda in public FDA and regional records.

  66. Development asset linked to Takeda in public FDA and regional records.

  67. Development asset linked to Takeda in public FDA and regional records.

  68. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  69. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  70. US regulatory status: approved. Molecular target: Bacterial penicillin-binding protein.

    Target
    Bacterial penicillin-binding protein
    Mechanism
    Bacterial penicillin-binding protein inhibitor
  71. US regulatory status: approved. Molecular target: Bacterial penicillin-binding protein.

    Target
    Bacterial penicillin-binding protein
    Mechanism
    Bacterial penicillin-binding protein inhibitor
  72. Development asset linked to Takeda in public FDA and regional records.

  73. Development asset linked to Takeda in public FDA and regional records.

  74. Development asset linked to Takeda in public FDA and regional records.

  75. Development asset linked to Takeda in public FDA and regional records.

  76. US regulatory status: approved. Molecular target: Solute carrier family 12 member 3.

    Target
    Solute carrier family 12 member 3
    Mechanism
    Thiazide-sensitive sodium-chloride cotransporter inhibitor
  77. US regulatory status: approved. Molecular target: Sodium-dependent serotonin transporter.

    Target
    Sodium-dependent serotonin transporter
    Mechanism
    Serotonin transporter substrate
  78. US regulatory status: approved. Molecular target: Solute carrier family 12 member 3.

    Target
    Solute carrier family 12 member 3
    Mechanism
    Thiazide-sensitive sodium-chloride cotransporter inhibitor
  79. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  80. US regulatory status: approved. Molecular target: Bacterial DNA gyrase.

    Target
    Bacterial DNA gyrase
    Mechanism
    Bacterial DNA gyrase inhibitor
  81. US regulatory status: approved. Molecular target: Bacterial DNA gyrase.

    Target
    Bacterial DNA gyrase
    Mechanism
    Bacterial DNA gyrase inhibitor
  82. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  83. Development asset linked to Takeda in public FDA and regional records. Mechanism: Serotonin transporter inhibitor.

    Mechanism
    Serotonin transporter inhibitor
  84. US regulatory status: approved. Molecular target: Bacterial 70S ribosome.

    Target
    Bacterial 70S ribosome
    Mechanism
    Bacterial 70S ribosome inhibitor
  85. clopidogrel

    Blood and blood forming organs (B01)

    Blood and blood forming organs (B01) compound in Takeda's portfolio. Mechanism: Purinergic receptor P2Y12 antagonist.

    Mechanism
    Purinergic receptor P2Y12 antagonist
  86. US regulatory status: approved. Molecular target: P2Y purinoceptor 12.

    Target
    P2Y purinoceptor 12
    Mechanism
    Purinergic receptor P2Y12 antagonist
  87. Development asset linked to Takeda in public FDA and regional records.

  88. colchicine

    Musculo-skeletal system (M04)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  89. Development asset linked to Takeda in public FDA and regional records.

  90. Development asset linked to Takeda in public FDA and regional records.

  91. Development asset linked to Takeda in public FDA and regional records.

  92. covid-19 vaccine (inactivated, adjuvanted, adsorbed)

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in Takeda's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  93. US regulatory status: approved. Molecular target: 5-hydroxytryptamine receptor 2A.

    Target
    5-hydroxytryptamine receptor 2A
    Mechanism
    Serotonin 2c (5-HT2c) receptor antagonist
  94. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  95. US regulatory status: approved. Molecular target: Peptidyl-prolyl cis-trans isomerase A.

    Target
    Peptidyl-prolyl cis-trans isomerase A
    Mechanism
    Cyclophilin A modulator
  96. Development asset linked to Takeda in public FDA and regional records.

  97. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  98. damoctocog alfa pegol

    Blood and blood forming organs (B02)

    Blood and blood forming organs (B02) compound in Takeda's portfolio. Molecular target: Coagulation factor VIII.

    Target
    Coagulation factor VIII
    Mechanism
    Coagulation factor VIII exogenous protein
  99. daratumumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1.

    Target
    ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
    Mechanism
    Lymphocyte differentiation antigen CD38 inhibitor
  100. darbepoetin alfa

    Blood and blood forming organs (B03)

    US regulatory status: approved. Molecular target: Erythropoietin receptor.

    Target
    Erythropoietin receptor
    Mechanism
    Erythropoietin receptor agonist
  101. darvadstrocel

    Antineoplastic and immunomodulating agents (L04)

    Antineoplastic and immunomodulating agents (L04) compound in Takeda's portfolio. Mechanism: Unknown.

    Mechanism
    Unknown
  102. dasatinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Bcr/Abl fusion protein.

    Target
    Bcr/Abl fusion protein
    Mechanism
    SRC inhibitor
  103. dengue tetravalent vaccine (live, attenuated)

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in Takeda's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  104. Development asset linked to Takeda in public FDA and regional records.

  105. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  106. deucravacitinib

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Non-receptor tyrosine-protein kinase TYK2.

    Target
    Non-receptor tyrosine-protein kinase TYK2
    Mechanism
    Tyrosine-protein kinase TYK2 negative allosteric modulator
  107. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  108. Development asset linked to Takeda in public FDA and regional records. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Dopamine transporter releasing agent
  109. US regulatory status: approved. Molecular target: Potassium-transporting ATPase.

    Target
    Potassium-transporting ATPase
    Mechanism
    Potassium-transporting ATPase inhibitor
  110. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter releasing agent
  111. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter releasing agent
  112. US regulatory status: approved. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  113. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter inhibitor
  114. US regulatory status: approved. Molecular target: Sodium/potassium-transporting ATPase.

    Target
    Sodium/potassium-transporting ATPase
    Mechanism
    Sodium/potassium-transporting ATPase inhibitor
  115. docetaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  116. Development asset linked to Takeda in public FDA and regional records.

  117. doxorubicin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Takeda's portfolio. Mechanism: DNA topoisomerase II alpha inhibitor.

    Mechanism
    DNA topoisomerase II alpha inhibitor
  118. doxorubicin hydrochloride

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA topoisomerase II alpha inhibitor
  119. US regulatory status: approved. Molecular target: Plasma kallikrein.

    Target
    Plasma kallikrein
    Mechanism
    Plasma kallikrein inhibitor
  120. emicizumab

    Blood and blood forming organs (B02)

    US regulatory status: approved. Molecular target: Coagulation factor IX and X.

    Target
    Coagulation factor IX and X
    Mechanism
    Coagulation factor IX and X other
  121. enoxaparin sodium

    Blood and blood forming organs (B01)

    US regulatory status: approved. Molecular target: Antithrombin-III.

    Target
    Antithrombin-III
    Mechanism
    Antithrombin-III activator
  122. Development asset linked to Takeda in public FDA and regional records.

  123. US regulatory status: approved. Molecular target: Erythropoietin receptor.

    Target
    Erythropoietin receptor
    Mechanism
    Erythropoietin receptor agonist
  124. epoetin delta

    Blood and blood forming organs (B03)

    Blood and blood forming organs (B03) compound in Takeda's portfolio. Molecular target: Erythropoietin receptor.

    Target
    Erythropoietin receptor
    Mechanism
    Erythropoietin receptor agonist
  125. US regulatory status: approved. Molecular target: Vitamin D3 receptor.

    Target
    Vitamin D3 receptor
    Mechanism
    Vitamin D receptor agonist
  126. Development asset linked to Takeda in public FDA and regional records.

  127. Development asset linked to Takeda in public FDA and regional records. Mechanism: Serotonin transporter inhibitor.

    Mechanism
    Serotonin transporter inhibitor
  128. US regulatory status: approved. Molecular target: Sodium-dependent serotonin transporter.

    Target
    Sodium-dependent serotonin transporter
    Mechanism
    Serotonin transporter inhibitor
  129. US regulatory status: approved. Molecular target: Glutamate [NMDA] receptor.

    Target
    Glutamate [NMDA] receptor
    Mechanism
    Glutamate [NMDA] receptor negative allosteric modulator
  130. esomeprazole

    Alimentary tract and metabolism (A02)

    Alimentary tract and metabolism (A02) compound in Takeda's portfolio. Mechanism: Potassium-transporting ATPase inhibitor.

    Mechanism
    Potassium-transporting ATPase inhibitor
  131. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  132. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  133. everolimus

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Peptidyl-prolyl cis-trans isomerase FKBP1A.

    Target
    Peptidyl-prolyl cis-trans isomerase FKBP1A
    Mechanism
    FK506-binding protein 1A inhibitor
  134. exagamglogene autotemcel

    Blood and blood forming organs (B06)

    Blood and blood forming organs (B06) compound in Takeda's portfolio. Molecular target: BCL11 transcription factor A.

    Target
    BCL11 transcription factor A
    Mechanism
    B-cell lymphoma/leukemia 11A gene editing negative modulator
  135. Development asset linked to Takeda in public FDA and regional records.

  136. febuxostat

    Musculo-skeletal system (M04)

    US regulatory status: approved. Molecular target: Xanthine dehydrogenase/oxidase.

    Target
    Xanthine dehydrogenase/oxidase
    Mechanism
    Xanthine dehydrogenase inhibitor
  137. fenofibrate

    Cardiovascular system (C10)

    US regulatory status: approved. Molecular target: Peroxisome proliferator-activated receptor alpha.

    Target
    Peroxisome proliferator-activated receptor alpha
    Mechanism
    Peroxisome proliferator-activated receptor alpha agonist
  138. US regulatory status: approved. Molecular target: Mu-type opioid receptor.

    Target
    Mu-type opioid receptor
    Mechanism
    Mu opioid receptor agonist
  139. ferumoxytol

    Blood and blood forming organs (B03)

    US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  140. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  141. follitropin beta

    Genito-urinary system and sex hormones (G03)

    Genito-urinary system and sex hormones (G03) compound in Takeda's portfolio. Molecular target: Follicle-stimulating hormone receptor.

    Target
    Follicle-stimulating hormone receptor
    Mechanism
    Follicle stimulating hormone receptor agonist
  142. Development asset linked to Takeda in public FDA and regional records.

  143. fruquintinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Vascular endothelial growth factor receptor.

    Target
    Vascular endothelial growth factor receptor
    Mechanism
    Vascular endothelial growth factor receptor inhibitor
  144. US regulatory status: approved. Molecular target: Voltage-gated calcium channel.

    Target
    Voltage-gated calcium channel
    Mechanism
    Voltage-gated calcium channel modulator
  145. US regulatory status: approved. Molecular target: Peroxisome proliferator-activated receptor alpha.

    Target
    Peroxisome proliferator-activated receptor alpha
    Mechanism
    Peroxisome proliferator-activated receptor alpha agonist
  146. US regulatory status: approved. Molecular target: Sulfonylurea receptor 1, Kir6.2.

    Target
    Sulfonylurea receptor 1, Kir6.2
    Mechanism
    Sulfonylurea receptor 1, Kir6.2 blocker
  147. glucagon

    Systemic hormonal preparations (H04)

    US regulatory status: approved. Molecular target: Glucagon receptor.

    Target
    Glucagon receptor
    Mechanism
    Glucagon receptor agonist
  148. US regulatory status: approved. Molecular target: Sulfonylurea receptor 1, Kir6.2.

    Target
    Sulfonylurea receptor 1, Kir6.2
    Mechanism
    Sulfonylurea receptor 1, Kir6.2 blocker
  149. Development asset linked to Takeda in public FDA and regional records.

  150. Development asset linked to Takeda in public FDA and regional records.

  151. Development asset linked to Takeda in public FDA and regional records.

  152. guanfacine

    Cardiovascular system (C02)

    Cardiovascular system (C02) compound in Takeda's portfolio. Mechanism: Adrenergic receptor alpha-2 agonist.

    Mechanism
    Adrenergic receptor alpha-2 agonist
  153. US regulatory status: approved. Molecular target: Adrenergic receptor alpha-2.

    Target
    Adrenergic receptor alpha-2
    Mechanism
    Adrenergic receptor alpha-2 agonist
  154. Development asset linked to Takeda in public FDA and regional records.

  155. Development asset linked to Takeda in public FDA and regional records.

  156. US regulatory status: approved. Molecular target: Muscarinic acetylcholine receptor M1.

    Target
    Muscarinic acetylcholine receptor M1
    Mechanism
    Muscarinic acetylcholine receptor M1 antagonist
  157. Development asset linked to Takeda in public FDA and regional records.

  158. human fibrinogen

    Blood and blood forming organs (B02)

    Blood and blood forming organs (B02) compound in Takeda's portfolio. Molecular target: Fibrinogen.

    Target
    Fibrinogen
    Mechanism
    Fibrinogen exogenous protein
  159. human normal immunoglobulin

    Antiinfectives for systemic use (J06)

    Antiinfectives for systemic use (J06) compound in Takeda's portfolio. Mechanism: Replacement therapy, immunomodulatory effects.

    Mechanism
    Replacement therapy, immunomodulatory effects
  160. human protein c

    Blood and blood forming organs (B01)

    Blood and blood forming organs (B01) compound in Takeda's portfolio. Molecular target: Vitamin K-dependent protein C.

    Target
    Vitamin K-dependent protein C
    Mechanism
    Vitamin K-dependent protein C exogenous protein
  161. US regulatory status: approved. Molecular target: Hyaluronic acid.

    Target
    Hyaluronic acid
    Mechanism
    Hyaluronic acid hydrolytic enzyme
  162. US regulatory status: approved. Molecular target: Solute carrier family 12 member 3.

    Target
    Solute carrier family 12 member 3
    Mechanism
    Thiazide-sensitive sodium-chloride cotransporter inhibitor
  163. hydrocortisone

    Systemic hormonal preparations (H02)

    US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  164. Development asset linked to Takeda in public FDA and regional records. Mechanism: Mu opioid receptor agonist.

    Mechanism
    Mu opioid receptor agonist
  165. Development asset linked to Takeda in public FDA and regional records.

  166. icatibant

    Blood and blood forming organs (B06)

    Blood and blood forming organs (B06) compound in Takeda's portfolio. Mechanism: Bradykinin B2 receptor antagonist.

    Mechanism
    Bradykinin B2 receptor antagonist
  167. US regulatory status: approved. Molecular target: B2 bradykinin receptor.

    Target
    B2 bradykinin receptor
    Mechanism
    Bradykinin B2 receptor antagonist
  168. idursulfase

    Alimentary tract and metabolism (A16)

    US regulatory status: approved. Molecular target: Heparan sulfate.

    Target
    Heparan sulfate
    Mechanism
    Heparan sulfate hydrolytic enzyme
  169. imatinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Takeda's portfolio. Mechanism: Tyrosine-protein kinase ABL inhibitor.

    Mechanism
    Tyrosine-protein kinase ABL inhibitor
  170. Development asset linked to Takeda in public FDA and regional records.

  171. Development asset linked to Takeda in public FDA and regional records.

  172. infliximab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Tumor necrosis factor.

    Target
    Tumor necrosis factor
    Mechanism
    TNF-alpha inhibitor
  173. Development asset linked to Takeda in public FDA and regional records.

  174. Development asset linked to Takeda in public FDA and regional records.

  175. Development asset linked to Takeda in public FDA and regional records.

  176. Development asset linked to Takeda in public FDA and regional records.

  177. Development asset linked to Takeda in public FDA and regional records. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  178. Development asset linked to Takeda in public FDA and regional records.

  179. interferon beta-1a

    Antineoplastic and immunomodulating agents (L03)

    US regulatory status: approved. Molecular target: Interferon alpha/beta receptor.

    Target
    Interferon alpha/beta receptor
    Mechanism
    Interferon alpha/beta receptor agonist
  180. Development asset linked to Takeda in public FDA and regional records.

  181. Development asset linked to Takeda in public FDA and regional records.

  182. Development asset linked to Takeda in public FDA and regional records.

  183. Development asset linked to Takeda in public FDA and regional records.

  184. ixazomib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Takeda's portfolio. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteasome inhibitor
  185. US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  186. lanadelumab

    Blood and blood forming organs (B06)

    Blood and blood forming organs (B06) compound in Takeda's portfolio. Molecular target: Plasma kallikrein.

    Target
    Plasma kallikrein
    Mechanism
    Plasma kallikrein inhibitor
  187. US regulatory status: approved. Molecular target: Plasma kallikrein.

    Target
    Plasma kallikrein
    Mechanism
    Plasma kallikrein inhibitor