Friday, July 10, 2026

Drug profile · INN

furmonertinib

furmonertinib is a epidermal growth factor receptor erbb1 inhibitor.

NMPA: clinical trials
Patents linked 0
Pipeline programs 10
News articles 0
Drug details — furmonertinib
Class
Route
Patents
0
Programs
10
Data quality
0.70

Quick answer

furmonertinib is a epidermal growth factor receptor erbb1 inhibitor.

Key facts

INN furmonertinib
Mechanism Epidermal growth factor receptor erbB1 inhibitor
Target Epidermal growth factor receptor

Mechanism of action

Epidermal growth factor receptor erbB1 inhibitor

Primary target: Epidermal growth factor receptor

Approval history

Authority Status Date
NMPA clinical trials

Pipeline programs

  1. FURMO-006 Phase 3 · ArriVent BioPharma · Advanced or Metastatic Non-Small-Cell Lung Cancer With Epide
  2. furmonertinib 240 mg oral, daily Phase 3 · ArriVent BioPharma · Metastatic Non-Small Cell Lung Cancer
  3. Furmonertinib Phase 2 · Peking University Biologics · Adenocarcinoma of Lung
  4. Furmonertinib Phase 2 · Shanghai University of · Lung Adenocarcinoma Stage III
  5. Furmonertinib Phase 2 · Chinese Academy of · Lung Adenocarcinoma Stage III
  6. Furmonertinib Phase 2 · First People's Hospital · Non-Small Cell Lung Cancer
  7. Furmonertinib in combination with Anrotinib and chemotherapy Phase 2 · Chinese Academy of · Lung Cancer (NSCLC)
  8. furmonertinib Phase 2 · Sun Yat-sen University · Non-small Cell Lung Cancer Metastatic

Related & competitor drugs

  1. erlotinib hydrochloride Epidermal growth factor receptor erbB1 inhibitor
  2. lapatinib ditosylate Receptor protein-tyrosine kinase erbB-2 inhibitor
  3. mobocertinib Antineoplastic and immunomodulating agents (L01)
  4. mobocertinib succinate Epidermal growth factor receptor erbB1 inhibitor
  5. neratinib maleate Receptor protein-tyrosine kinase erbB-2 inhibitor
  6. afatinib dimaleate Epidermal growth factor receptor erbB1 inhibitor

Frequently asked questions

What is furmonertinib?

furmonertinib is a epidermal growth factor receptor erbb1 inhibitor.