Wednesday, July 8, 2026

Drug profile · INN

lapatinib ditosylate

lapatinib ditosylate (LAPATINIB DITOSYLATE) is a receptor protein-tyrosine kinase erbb-2 inhibitor. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 13
News articles 0
Drug details — lapatinib ditosylate
US status
approved
Class
Route
ORAL
Patents
0
Programs
13
Data quality
0.89

Quick answer

lapatinib ditosylate (LAPATINIB DITOSYLATE) is a receptor protein-tyrosine kinase erbb-2 inhibitor. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN lapatinib ditosylate
Brand LAPATINIB DITOSYLATE
Mechanism Receptor protein-tyrosine kinase erbB-2 inhibitor
Target Epidermal growth factor receptor
Route ORAL
Formulation TABLET

Mechanism of action

Receptor protein-tyrosine kinase erbB-2 inhibitor

Primary target: Epidermal growth factor receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. Apatinib Phase 2 · First People's Hospital · Thyroid
  2. Apatinib Phase 2 · First People's Hospital · Advanced Solid Tumors
  3. Apatinib Phase 2 · Chinese Academy of · Breast Cancer Metastatic
  4. Apatinib Phase 2 · Chinese Academy of · Lung Cancer
  5. Apatinib Phase 2 · Chinese Academy of · Metastatic Gastric Adenocarcinoma
  6. Apatinib Phase 2 · First People's Hospital · Advanced Esophageal Squamous Carcinoma
  7. Apatinib Phase 2 · First People's Hospital · Breast Cancer
  8. Apatinib Phase 2 · First People's Hospital · Intrahepatic Cholangiocarcinoma

Related & competitor drugs

  1. erlotinib hydrochloride Epidermal growth factor receptor erbB1 inhibitor
  2. mobocertinib Antineoplastic and immunomodulating agents (L01)
  3. mobocertinib succinate Epidermal growth factor receptor erbB1 inhibitor
  4. neratinib maleate Receptor protein-tyrosine kinase erbB-2 inhibitor
  5. afatinib dimaleate Epidermal growth factor receptor erbB1 inhibitor
  6. amivantamab-vmjw Epidermal growth factor receptor erbB1 inhibitor

Frequently asked questions

What is lapatinib ditosylate?

lapatinib ditosylate (LAPATINIB DITOSYLATE) is a receptor protein-tyrosine kinase erbb-2 inhibitor. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for lapatinib ditosylate?

LAPATINIB DITOSYLATE is a marketed brand name for lapatinib ditosylate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of lapatinib ditosylate?

lapatinib ditosylate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.