Friday, July 10, 2026

Drug profile · INN

mobocertinib

mobocertinib (EXKIVITY) is a epidermal growth factor receptor erbb1 inhibitor. Associated with Takeda.

EMA: application withdrawn Antineoplastic and immunomodulating agents (L01) L01EB
Patents linked 0
Pipeline programs 4
News articles 1
Drug details — mobocertinib

Quick answer

mobocertinib (EXKIVITY) is a epidermal growth factor receptor erbb1 inhibitor. Associated with Takeda.

Key facts

INN mobocertinib
Brand EXKIVITY
Mechanism Epidermal growth factor receptor erbB1 inhibitor
Target Epidermal growth factor receptor
Therapeutic class Antineoplastic and immunomodulating agents (L01)
ATC code L01EB
Originator Takeda

Mechanism of action

Epidermal growth factor receptor erbB1 inhibitor

Primary target: Epidermal growth factor receptor

Approval history

Authority Status Date
EMA application withdrawn

Recent coverage

Pipeline programs

  1. Mobocertinib Phase 1 · Takeda · Healthy Volunteers
  2. Mobocertinib Phase 1 · Takeda · Hepatic Impairment
  3. Mobocertinib Phase 1 · Takeda · Non-Small Cell Lung Cancer
  4. Mobocertinib Phase 1 · Takeda · Renal Impairment

Related & competitor drugs

  1. abiraterone acetate Antineoplastic and immunomodulating agents (L02)
  2. anagrelide Antineoplastic and immunomodulating agents (L01)
  3. apremilast Antineoplastic and immunomodulating agents (L04)
  4. arsenic trioxide Antineoplastic and immunomodulating agents (L01)
  5. axitinib Antineoplastic and immunomodulating agents (L01)
  6. azacitidine Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is mobocertinib?

mobocertinib (EXKIVITY) is a epidermal growth factor receptor erbb1 inhibitor. Associated with Takeda.

What is the brand name for mobocertinib?

EXKIVITY is a marketed brand name for mobocertinib. Check FDA Drugs@FDA for the current US label holder and prescribing information.