Wednesday, July 8, 2026

Drug profile · INN

mobocertinib succinate

mobocertinib succinate (EXKIVITY) is a epidermal growth factor receptor erbb1 inhibitor. Associated with Takeda. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 4
News articles 0
Drug details — mobocertinib succinate
US status
approved
Class
Route
ORAL
Patents
0
Programs
4
Data quality
0.89

Quick answer

mobocertinib succinate (EXKIVITY) is a epidermal growth factor receptor erbb1 inhibitor. Associated with Takeda. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN mobocertinib succinate
Brand EXKIVITY
Mechanism Epidermal growth factor receptor erbB1 inhibitor
Target Epidermal growth factor receptor
Route ORAL
Formulation CAPSULE
Originator Takeda

Mechanism of action

Epidermal growth factor receptor erbB1 inhibitor

Primary target: Epidermal growth factor receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. Mobocertinib Phase 1 · Takeda · Healthy Volunteers
  2. Mobocertinib Phase 1 · Takeda · Hepatic Impairment
  3. Mobocertinib Phase 1 · Takeda · Non-Small Cell Lung Cancer
  4. Mobocertinib Phase 1 · Takeda · Renal Impairment

Related & competitor drugs

  1. erlotinib hydrochloride Epidermal growth factor receptor erbB1 inhibitor
  2. lapatinib ditosylate Receptor protein-tyrosine kinase erbB-2 inhibitor
  3. mobocertinib Antineoplastic and immunomodulating agents (L01)
  4. neratinib maleate Receptor protein-tyrosine kinase erbB-2 inhibitor
  5. afatinib dimaleate Epidermal growth factor receptor erbB1 inhibitor
  6. amivantamab-vmjw Epidermal growth factor receptor erbB1 inhibitor

Frequently asked questions

What is mobocertinib succinate?

mobocertinib succinate (EXKIVITY) is a epidermal growth factor receptor erbb1 inhibitor. Associated with Takeda. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for mobocertinib succinate?

EXKIVITY is a marketed brand name for mobocertinib succinate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of mobocertinib succinate?

mobocertinib succinate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.