Wednesday, July 8, 2026

Drug profile · INN

aminophylline

aminophylline (AMINOPHYLLINE) is a adenosine receptor antagonist. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: rectal. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 20
Pipeline programs 1
News articles 0
Drug details — aminophylline
US status
approved
Class
Route
RECTAL
Patents
20
Programs
1
Data quality
0.89

Quick answer

aminophylline (AMINOPHYLLINE) is a adenosine receptor antagonist. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: rectal. Current US regulatory status: approved.

Key facts

INN aminophylline
Brand AMINOPHYLLINE
Mechanism Adenosine receptor antagonist
Target Adenosine receptor
Route RECTAL
Formulation TABLET, EXTENDED RELEASE

Mechanism of action

Adenosine receptor antagonist

Primary target: Adenosine receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. SOM 230 / Pasireotide Phase 1 · United Therapeutics Europe · Atypical Ductal Breast Hyperplasia

Related & competitor drugs

  1. adenosine Adenosine receptor agonist
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  4. caffeine Nervous system (N06)
  5. istradefylline Nervous system (N04)
  6. oxtriphylline Phosphodiesterase 3 inhibitor
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Frequently asked questions

What is aminophylline?

aminophylline (AMINOPHYLLINE) is a adenosine receptor antagonist. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: rectal. Current US regulatory status: approved.

What is the brand name for aminophylline?

AMINOPHYLLINE is a marketed brand name for aminophylline. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of aminophylline?

aminophylline has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.