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Novartis India

Novartis India drug portfolio β€” 200 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Mumbai, IN HQ
1996 Founded
2,240 Employees
NMPA registrant Type
Company details
Status
Public
HQ
Mumbai, IN
Founded
1996
Employees
2,240
Programs
341
Drugs
317
Patents
0
Intelligence Β· Drug Pipeline

Novartis India pipeline

Portfolio lens on 200 drugs and development assets β€” regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

Novartis India drug portfolio β€” 200 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

200 compounds
  1. abacavir

    Antiinfectives for systemic use (J05)

    US regulatory status: approved.

  2. abiraterone

    Antineoplastic and immunomodulating agents (L02)

    Antineoplastic and immunomodulating agents (L02) compound in Novartis India's portfolio. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Steroid 5-alpha-reductase inhibitor
  3. abiraterone acetate

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Steroid 17-alpha-hydroxylase/17,20 lyase.

    Target
    Steroid 17-alpha-hydroxylase/17,20 lyase
    Mechanism
    Cytochrome P450 17A1 inhibitor
  4. Development asset linked to Novartis India in public FDA and regional records. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  5. US regulatory status: approved. Molecular target: Fatty-acid amide hydrolase 1.

    Target
    Fatty-acid amide hydrolase 1
    Mechanism
    Cyclooxygenase inhibitor
  6. Development asset linked to Novartis India in public FDA and regional records.

  7. US regulatory status: approved. Molecular target: Beta-2 adrenergic receptor.

    Target
    Beta-2 adrenergic receptor
    Mechanism
    Beta-2 adrenergic receptor agonist
  8. US regulatory status: approved.

  9. US regulatory status: approved. Molecular target: Interleukin-2 receptor.

    Target
    Interleukin-2 receptor
    Mechanism
    Interleukin-2 receptor agonist
  10. aliskiren

    Cardiovascular system (C09)

    Cardiovascular system (C09) compound in Novartis India's portfolio. Mechanism: Renin inhibitor.

    Mechanism
    Renin inhibitor
  11. alpelisib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform.

    Target
    Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
    Mechanism
    PI3-kinase p110-alpha subunit inhibitor
  12. Development asset linked to Novartis India in public FDA and regional records.

  13. Development asset linked to Novartis India in public FDA and regional records.

  14. US regulatory status: approved. Mechanism: Glutamate [NMDA] receptor antagonist.

    Mechanism
    Glutamate [NMDA] receptor antagonist
  15. US regulatory status: approved. Molecular target: Aromatase.

    Target
    Aromatase
    Mechanism
    Cytochrome P450 19A1 inhibitor
  16. Development asset linked to Novartis India in public FDA and regional records.

  17. Various (V09) compound in Novartis India's portfolio. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  18. Development asset linked to Novartis India in public FDA and regional records.

  19. apalutamide

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  20. Development asset linked to Novartis India in public FDA and regional records.

  21. arginine

    Various (V03)

    Various (V03) compound in Novartis India's portfolio.

  22. asciminib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Novartis India's portfolio. Molecular target: Tyrosine-protein kinase ABL1.

    Target
    Tyrosine-protein kinase ABL1
    Mechanism
    Bcr/Abl fusion protein inhibitor
  23. US regulatory status: approved. Molecular target: Bcr/Abl fusion protein.

    Target
    Bcr/Abl fusion protein
    Mechanism
    Bcr/Abl fusion protein inhibitor
  24. asenapine

    Nervous system (N05)

    US regulatory status: approved. Mechanism: Serotonin 2a (5-HT2a) receptor antagonist.

    Mechanism
    Serotonin 2a (5-HT2a) receptor antagonist
  25. atezolizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death 1 ligand 1.

    Target
    Programmed cell death 1 ligand 1
    Mechanism
    Programmed cell death 1 ligand 1 inhibitor
  26. Development asset linked to Novartis India in public FDA and regional records. Mechanism: HMG-CoA reductase inhibitor.

    Mechanism
    HMG-CoA reductase inhibitor
  27. Development asset linked to Novartis India in public FDA and regional records.

  28. atropine sulfate

    Sensory organs (S01)

    US regulatory status: approved. Molecular target: Muscarinic acetylcholine receptor M1.

    Target
    Muscarinic acetylcholine receptor M1
    Mechanism
    Muscarinic acetylcholine receptor M3 antagonist
  29. azacitidine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA (cytosine-5)-methyltransferase 1.

    Target
    DNA (cytosine-5)-methyltransferase 1
    Mechanism
    DNA (cytosine-5)-methyltransferase 3A inhibitor
  30. azathioprine

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Amidophosphoribosyltransferase.

    Target
    Amidophosphoribosyltransferase
    Mechanism
    Amidophosphoribosyltransferase inhibitor
  31. US regulatory status: approved. Molecular target: Amidophosphoribosyltransferase.

    Target
    Amidophosphoribosyltransferase
    Mechanism
    Amidophosphoribosyltransferase inhibitor
  32. US regulatory status: approved. Molecular target: Type-1 angiotensin II receptor.

    Target
    Type-1 angiotensin II receptor
    Mechanism
    Type-1 angiotensin II receptor antagonist
  33. belimumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Tumor necrosis factor ligand superfamily member 13B.

    Target
    Tumor necrosis factor ligand superfamily member 13B
    Mechanism
    Tumor necrosis factor ligand superfamily member 13B inhibitor
  34. bempedoic acid

    Cardiovascular system (C10)

    US regulatory status: approved. Molecular target: ATP-citrate synthase.

    Target
    ATP-citrate synthase
    Mechanism
    ATP-citrate synthase inhibitor
  35. Development asset linked to Novartis India in public FDA and regional records. Mechanism: Angiotensin-converting enzyme inhibitor.

    Mechanism
    Angiotensin-converting enzyme inhibitor
  36. Development asset linked to Novartis India in public FDA and regional records.

  37. US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  38. blinatumomab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: B-lymphocyte antigen CD19.

    Target
    B-lymphocyte antigen CD19
    Mechanism
    T cell surface glycoprotein CD3 cross-linking agent
  39. bosutinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Novartis India's portfolio. Molecular target: Tyrosine-protein kinase ABL1.

    Target
    Tyrosine-protein kinase ABL1
    Mechanism
    Tyrosine-protein kinase ABL inhibitor
  40. brimonidine

    Dermatologicals (D11)

    Dermatologicals (D11) compound in Novartis India's portfolio. Mechanism: Adrenergic receptor alpha-2 agonist.

    Mechanism
    Adrenergic receptor alpha-2 agonist
  41. brinzolamide

    Sensory organs (S01)

    US regulatory status: approved. Molecular target: Carbonic anhydrase 2.

    Target
    Carbonic anhydrase 2
    Mechanism
    Carbonic anhydrase II inhibitor
  42. brolucizumab

    Sensory organs (S01)

    Sensory organs (S01) compound in Novartis India's portfolio. Molecular target: Vascular endothelial growth factor A, long form.

    Target
    Vascular endothelial growth factor A, long form
    Mechanism
    Vascular endothelial growth factor A inhibitor
  43. cabazitaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  44. US regulatory status: approved. Molecular target: Vitamin D3 receptor.

    Target
    Vitamin D3 receptor
    Mechanism
    Vitamin D receptor agonist
  45. US regulatory status: approved.

  46. canakinumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Interleukin-1 beta.

    Target
    Interleukin-1 beta
    Mechanism
    Interleukin-1 beta inhibitor
  47. Development asset linked to Novartis India in public FDA and regional records. Molecular target: Type-1 angiotensin II receptor.

    Target
    Type-1 angiotensin II receptor
    Mechanism
    Type-1 angiotensin II receptor antagonist
  48. capecitabine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  49. capmatinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Novartis India's portfolio. Molecular target: Hepatocyte growth factor receptor.

    Target
    Hepatocyte growth factor receptor
    Mechanism
    Hepatocyte growth factor receptor inhibitor
  50. Development asset linked to Novartis India in public FDA and regional records.

  51. Development asset linked to Novartis India in public FDA and regional records.

  52. US regulatory status: approved. Molecular target: Angiotensin-converting enzyme.

    Target
    Angiotensin-converting enzyme
    Mechanism
    Angiotensin-converting enzyme inhibitor
  53. Development asset linked to Novartis India in public FDA and regional records.

  54. US regulatory status: approved. Molecular target: Sodium channel alpha subunit.

    Target
    Sodium channel alpha subunit
    Mechanism
    Sodium channel alpha subunit blocker
  55. US regulatory status: approved. Molecular target: Aromatic-L-amino-acid decarboxylase.

    Target
    Aromatic-L-amino-acid decarboxylase
    Mechanism
    DOPA decarboxylase inhibitor
  56. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  57. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  58. carmustine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Glutathione reductase inhibitor
  59. Development asset linked to Novartis India in public FDA and regional records.

  60. ceritinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: ALK tyrosine kinase receptor.

    Target
    ALK tyrosine kinase receptor
    Mechanism
    EML4-ALK
  61. cetuximab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  62. Development asset linked to Novartis India in public FDA and regional records.

  63. Development asset linked to Novartis India in public FDA and regional records.

  64. ciclosporin

    Sensory organs (S01)

    Sensory organs (S01) compound in Novartis India's portfolio. Molecular target: Peptidyl-prolyl cis-trans isomerase A.

    Target
    Peptidyl-prolyl cis-trans isomerase A
    Mechanism
    Cyclophilin A modulator
  65. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  66. Development asset linked to Novartis India in public FDA and regional records.

  67. clopidogrel

    Blood and blood forming organs (B01)

    Blood and blood forming organs (B01) compound in Novartis India's portfolio. Mechanism: Purinergic receptor P2Y12 antagonist.

    Mechanism
    Purinergic receptor P2Y12 antagonist
  68. Development asset linked to Novartis India in public FDA and regional records. Mechanism: Opioid receptors; mu/kappa/delta agonist.

    Mechanism
    Opioid receptors; mu/kappa/delta agonist
  69. US regulatory status: approved. Molecular target: Opioid receptors; mu/kappa/delta.

    Target
    Opioid receptors; mu/kappa/delta
    Mechanism
    Opioid receptors; mu/kappa/delta agonist
  70. Development asset linked to Novartis India in public FDA and regional records. Molecular target: Bile acids.

    Target
    Bile acids
    Mechanism
    Bile acids sequestering agent
  71. Development asset linked to Novartis India in public FDA and regional records.

  72. Development asset linked to Novartis India in public FDA and regional records.

  73. Development asset linked to Novartis India in public FDA and regional records.

  74. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  75. US regulatory status: approved. Molecular target: Peptidyl-prolyl cis-trans isomerase A.

    Target
    Peptidyl-prolyl cis-trans isomerase A
    Mechanism
    Cyclophilin A modulator
  76. cytarabine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA polymerase (alpha/delta/epsilon) inhibitor
  77. dabrafenib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Novartis India's portfolio. Mechanism: Serine/threonine-protein kinase B-raf inhibitor.

    Mechanism
    Serine/threonine-protein kinase B-raf inhibitor
  78. US regulatory status: approved. Molecular target: Serine/threonine-protein kinase B-raf.

    Target
    Serine/threonine-protein kinase B-raf
    Mechanism
    Serine/threonine-protein kinase B-raf inhibitor
  79. US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Progesterone receptor agonist
  80. darolutamide

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  81. dasatinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Bcr/Abl fusion protein.

    Target
    Bcr/Abl fusion protein
    Mechanism
    SRC inhibitor
  82. daunorubicin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Novartis India's portfolio. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA topoisomerase II alpha inhibitor
  83. deferasirox

    Various (V03)

    US regulatory status: approved. Molecular target: Iron.

    Target
    Iron
    Mechanism
    Iron chelating agent
  84. degarelix

    Antineoplastic and immunomodulating agents (L02)

    Antineoplastic and immunomodulating agents (L02) compound in Novartis India's portfolio. Mechanism: Gonadotropin-releasing hormone receptor antagonist.

    Mechanism
    Gonadotropin-releasing hormone receptor antagonist
  85. US regulatory status: approved. Molecular target: Gonadotropin-releasing hormone receptor.

    Target
    Gonadotropin-releasing hormone receptor
    Mechanism
    Gonadotropin-releasing hormone receptor antagonist
  86. dengue tetravalent vaccine (live, attenuated)

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in Novartis India's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  87. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  88. Development asset linked to Novartis India in public FDA and regional records.

  89. dimethyl fumarate

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Kelch-like ECH-associated protein 1.

    Target
    Kelch-like ECH-associated protein 1
    Mechanism
    Kelch-like ECH-associated protein 1 inhibitor
  90. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  91. diroximel fumarate

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Kelch-like ECH-associated protein 1.

    Target
    Kelch-like ECH-associated protein 1
    Mechanism
    Kelch-like ECH-associated protein 1 inhibitor
  92. docetaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  93. dolutegravir

    Antiinfectives for systemic use (J05)

    US regulatory status: approved.

  94. Development asset linked to Novartis India in public FDA and regional records.

  95. doxorubicin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Novartis India's portfolio. Mechanism: DNA topoisomerase II alpha inhibitor.

    Mechanism
    DNA topoisomerase II alpha inhibitor
  96. doxorubicin hydrochloride

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA topoisomerase II alpha inhibitor
  97. US regulatory status: approved. Molecular target: Mineralocorticoid receptor.

    Target
    Mineralocorticoid receptor
    Mechanism
    Progesterone receptor agonist
  98. eltrombopag

    Blood and blood forming organs (B02)

    US regulatory status: approved. Mechanism: Thrombopoietin receptor agonist.

    Mechanism
    Thrombopoietin receptor agonist
  99. Development asset linked to Novartis India in public FDA and regional records. Mechanism: Angiotensin-converting enzyme inhibitor.

    Mechanism
    Angiotensin-converting enzyme inhibitor
  100. Development asset linked to Novartis India in public FDA and regional records.

  101. entacapone

    Nervous system (N04)

    US regulatory status: approved. Molecular target: Catechol O-methyltransferase.

    Target
    Catechol O-methyltransferase
    Mechanism
    Catechol O-methyltransferase inhibitor
  102. entecavir

    Antiinfectives for systemic use (J05)

    US regulatory status: approved. Molecular target: DNA polymerase/reverse transcriptase.

    Target
    DNA polymerase/reverse transcriptase
    Mechanism
    DNA polymerase/reverse transcriptase inhibitor
  103. Development asset linked to Novartis India in public FDA and regional records.

  104. enzalutamide

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  105. Development asset linked to Novartis India in public FDA and regional records.

  106. Development asset linked to Novartis India in public FDA and regional records. Mechanism: Type-1 angiotensin II receptor antagonist.

    Mechanism
    Type-1 angiotensin II receptor antagonist
  107. US regulatory status: approved. Molecular target: Bacterial 70S ribosome.

    Target
    Bacterial 70S ribosome
    Mechanism
    Bacterial 70S ribosome inhibitor
  108. Development asset linked to Novartis India in public FDA and regional records.

  109. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  110. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  111. US regulatory status: approved. Molecular target: DNA topoisomerase II.

    Target
    DNA topoisomerase II
    Mechanism
    DNA topoisomerase II inhibitor
  112. everolimus

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Peptidyl-prolyl cis-trans isomerase FKBP1A.

    Target
    Peptidyl-prolyl cis-trans isomerase FKBP1A
    Mechanism
    FK506-binding protein 1A inhibitor
  113. US regulatory status: approved. Molecular target: Aromatase.

    Target
    Aromatase
    Mechanism
    Cytochrome P450 19A1 inhibitor
  114. US regulatory status: approved. Molecular target: NPC1-like intracellular cholesterol transporter 1.

    Target
    NPC1-like intracellular cholesterol transporter 1
    Mechanism
    Niemann-Pick C1-like protein 1 inhibitor
  115. fingolimod

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Mechanism: Sphingosine 1-phosphate receptor binding agent.

    Mechanism
    Sphingosine 1-phosphate receptor binding agent
  116. US regulatory status: approved. Molecular target: Sphingosine 1-phosphate receptor.

    Target
    Sphingosine 1-phosphate receptor
    Mechanism
    Sphingosine 1-phosphate receptor agonist
  117. florbetaben (18f)

    Various (V09)

    Various (V09) compound in Novartis India's portfolio. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  118. US regulatory status: approved. Molecular target: Lanosterol 14-alpha demethylase.

    Target
    Lanosterol 14-alpha demethylase
    Mechanism
    Cytochrome P450 51 inhibitor
  119. Development asset linked to Novartis India in public FDA and regional records.

  120. US regulatory status: approved. Molecular target: DNA polymerase (alpha/delta/epsilon).

    Target
    DNA polymerase (alpha/delta/epsilon)
    Mechanism
    DNA polymerase (alpha/delta/epsilon) inhibitor
  121. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  122. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  123. US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  124. Development asset linked to Novartis India in public FDA and regional records.

  125. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  126. Development asset linked to Novartis India in public FDA and regional records.

  127. Development asset linked to Novartis India in public FDA and regional records. Mechanism: Angiotensin-converting enzyme inhibitor.

    Mechanism
    Angiotensin-converting enzyme inhibitor
  128. fulvestrant

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor antagonist
  129. gefitinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  130. US regulatory status: approved. Mechanism: DNA polymerase (alpha/delta/epsilon) inhibitor.

    Mechanism
    DNA polymerase (alpha/delta/epsilon) inhibitor
  131. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  132. glycopyrronium

    Respiratory system (R03)

    Respiratory system (R03) compound in Novartis India's portfolio. Mechanism: Muscarinic acetylcholine receptor inhibitor.

    Mechanism
    Muscarinic acetylcholine receptor inhibitor
  133. glycopyrronium bromide

    Respiratory system (R03)

    Respiratory system (R03) compound in Novartis India's portfolio. Molecular target: Muscarinic acetylcholine receptor M1.

    Target
    Muscarinic acetylcholine receptor M1
    Mechanism
    Muscarinic acetylcholine receptor M1 antagonist
  134. US regulatory status: approved. Mechanism: Gonadotropin-releasing hormone receptor agonist.

    Mechanism
    Gonadotropin-releasing hormone receptor agonist
  135. US regulatory status: approved. Molecular target: Gonadotropin-releasing hormone receptor.

    Target
    Gonadotropin-releasing hormone receptor
    Mechanism
    Gonadotropin-releasing hormone receptor agonist
  136. gozetotide

    Various (V09)

    Various (V09) compound in Novartis India's portfolio. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  137. Development asset linked to Novartis India in public FDA and regional records.

  138. Development asset linked to Novartis India in public FDA and regional records.

  139. US regulatory status: approved. Molecular target: Enoyl-[acyl-carrier-protein] reductase [NADH] FabI.

    Target
    Enoyl-[acyl-carrier-protein] reductase [NADH] FabI
    Mechanism
    Bacterial enoyl-[acyl-carrier-protein] reductase inhibitor
  140. US regulatory status: approved. Molecular target: Muscarinic acetylcholine receptor M1.

    Target
    Muscarinic acetylcholine receptor M1
    Mechanism
    Muscarinic acetylcholine receptor M1 antagonist
  141. hydrocortisone

    Systemic hormonal preparations (H02)

    US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  142. Development asset linked to Novartis India in public FDA and regional records. Molecular target: Tumor necrosis factor receptor superfamily member 13C.

    Target
    Tumor necrosis factor receptor superfamily member 13C
    Mechanism
    Tumor necrosis factor receptor superfamily member 13C binding agent
  143. ibrutinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tyrosine-protein kinase BTK.

    Target
    Tyrosine-protein kinase BTK
    Mechanism
    Tyrosine-protein kinase BTK inhibitor
  144. Development asset linked to Novartis India in public FDA and regional records. Mechanism: DNA topoisomerase II alpha inhibitor.

    Mechanism
    DNA topoisomerase II alpha inhibitor
  145. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  146. imatinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Novartis India's portfolio. Mechanism: Tyrosine-protein kinase ABL inhibitor.

    Mechanism
    Tyrosine-protein kinase ABL inhibitor
  147. Development asset linked to Novartis India in public FDA and regional records.

  148. inclisiran

    Cardiovascular system (C10)

    Cardiovascular system (C10) compound in Novartis India's portfolio. Molecular target: PCSK9 mRNA.

    Target
    PCSK9 mRNA
    Mechanism
    PCSK9 mRNA RNAi inhibitor
  149. US regulatory status: approved. Molecular target: PCSK9 mRNA.

    Target
    PCSK9 mRNA
    Mechanism
    PCSK9 mRNA rnai inhibitor
  150. indacaterol

    Respiratory system (R03)

    Respiratory system (R03) compound in Novartis India's portfolio. Mechanism: Beta-2 adrenergic receptor agonist.

    Mechanism
    Beta-2 adrenergic receptor agonist
  151. Development asset linked to Novartis India in public FDA and regional records.

  152. Development asset linked to Novartis India in public FDA and regional records.

  153. Development asset linked to Novartis India in public FDA and regional records.

  154. Development asset linked to Novartis India in public FDA and regional records.

  155. Development asset linked to Novartis India in public FDA and regional records.

  156. Development asset linked to Novartis India in public FDA and regional records.

  157. insulin lispro

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  158. interferon alfa-2b

    Antineoplastic and immunomodulating agents (L03)

    US regulatory status: approved. Molecular target: Interferon alpha/beta receptor.

    Target
    Interferon alpha/beta receptor
    Mechanism
    Interferon alpha/beta receptor agonist
  159. interferon beta-1b

    Antineoplastic and immunomodulating agents (L03)

    US regulatory status: approved. Molecular target: Interferon alpha/beta receptor.

    Target
    Interferon alpha/beta receptor
    Mechanism
    Interferon alpha/beta receptor agonist
  160. Development asset linked to Novartis India in public FDA and regional records.

  161. iptacopan

    Antineoplastic and immunomodulating agents (L04)

    Antineoplastic and immunomodulating agents (L04) compound in Novartis India's portfolio. Molecular target: Complement factor B.

    Target
    Complement factor B
    Mechanism
    Complement factor B inhibitor
  162. US regulatory status: approved. Molecular target: Complement factor B.

    Target
    Complement factor B
    Mechanism
    Complement factor B inhibitor
  163. irbesartan

    Cardiovascular system (C09)

    US regulatory status: approved. Molecular target: Type-1 angiotensin II receptor.

    Target
    Type-1 angiotensin II receptor
    Mechanism
    Type-1 angiotensin II receptor antagonist
  164. Development asset linked to Novartis India in public FDA and regional records. Mechanism: DNA topoisomerase I inhibitor.

    Mechanism
    DNA topoisomerase I inhibitor
  165. US regulatory status: approved. Molecular target: Cyclooxygenase.

    Target
    Cyclooxygenase
    Mechanism
    Cyclooxygenase inhibitor
  166. lamivudine

    Antiinfectives for systemic use (J05)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  167. lapatinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Novartis India's portfolio. Mechanism: Receptor protein-tyrosine kinase erbB-2 inhibitor.

    Mechanism
    Receptor protein-tyrosine kinase erbB-2 inhibitor
  168. lenalidomide

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: CRL4(CRBN) E3 ubiquitin ligase.

    Target
    CRL4(CRBN) E3 ubiquitin ligase
    Mechanism
    CRL4(CRBN) E3 ubiquitin ligase inhibitor
  169. US regulatory status: approved. Molecular target: Aromatase.

    Target
    Aromatase
    Mechanism
    Cytochrome P450 19A1 inhibitor
  170. Development asset linked to Novartis India in public FDA and regional records.

  171. levodopa

    Nervous system (N04)

    US regulatory status: approved. Molecular target: D(3) dopamine receptor.

    Target
    D(3) dopamine receptor
    Mechanism
    Dopamine D3 receptor agonist
  172. Development asset linked to Novartis India in public FDA and regional records.

  173. US regulatory status: approved. Molecular target: Angiotensin-converting enzyme.

    Target
    Angiotensin-converting enzyme
    Mechanism
    Angiotensin-converting enzyme inhibitor
  174. Various (V10) compound in Novartis India's portfolio. Molecular target: Somatostatin receptor.

    Target
    Somatostatin receptor
    Mechanism
    Somatostatin receptor binding agent
  175. Development asset linked to Novartis India in public FDA and regional records.

  176. US regulatory status: approved. Molecular target: Acetylcholinesterase.

    Target
    Acetylcholinesterase
    Mechanism
    Acetylcholinesterase inhibitor
  177. Development asset linked to Novartis India in public FDA and regional records.

  178. Development asset linked to Novartis India in public FDA and regional records.

  179. melphalan

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  180. methotrexate

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Dihydrofolate reductase.

    Target
    Dihydrofolate reductase
    Mechanism
    Dihydrofolate reductase inhibitor
  181. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter inhibitor