Friday, July 10, 2026

Drug profile · INN

bosutinib

bosutinib (BOSULIF) is a tyrosine-protein kinase abl inhibitor.

EMA: approved NMPA: clinical trials Antineoplastic and immunomodulating agents (L01) L01EA04
Patents linked 0
Pipeline programs 7
News articles 1
Drug details — bosutinib
Class
Antineoplastic and immunomodulating agents (L01)
Route
Patents
0
Programs
7
Data quality
0.83

Quick answer

bosutinib (BOSULIF) is a tyrosine-protein kinase abl inhibitor.

Key facts

INN bosutinib
Brand BOSULIF
Mechanism Tyrosine-protein kinase ABL inhibitor
Target Tyrosine-protein kinase ABL1
Therapeutic class Antineoplastic and immunomodulating agents (L01)
ATC code L01EA04

Mechanism of action

Tyrosine-protein kinase ABL inhibitor

Primary target: Tyrosine-protein kinase ABL1

Approval history

Authority Status Date
EMA approved
NMPA clinical trials

Recent coverage

Pipeline programs

  1. Bosutinib Phase 3 · Pfizer · Chronic Myeloid Leukemia
  2. CABL001A2001B Phase 3 · Novartis India · chronic myelogenous leukemia (CML) or Philadelphia Chromosom
  3. CABL001J12301 Phase 3 · Novartis India · Chronic Myeloid Leukemia
  4. HQP1351CG301 Phase 3 · Anaxis Pharma · Chronic Phase Chronic Myeloid Leukemia
  5. ITCC-054/AAML1921 Phase 2 · Disc Medicine · Chronic Myeloid Leukemia
  6. BOSUT-09-24 Phase 1 · Anaxis Pharma · myeloid leukemia
  7. IMATINIB for Chronic myeloid leukaemia Approved · Disc Medicine · Chronic myeloid leukaemia

Related & competitor drugs

  1. abiraterone acetate Antineoplastic and immunomodulating agents (L02)
  2. anagrelide Antineoplastic and immunomodulating agents (L01)
  3. apremilast Antineoplastic and immunomodulating agents (L04)
  4. arsenic trioxide Antineoplastic and immunomodulating agents (L01)
  5. axitinib Antineoplastic and immunomodulating agents (L01)
  6. azacitidine Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is bosutinib?

bosutinib (BOSULIF) is a tyrosine-protein kinase abl inhibitor.

What is the brand name for bosutinib?

BOSULIF is a marketed brand name for bosutinib. Check FDA Drugs@FDA for the current US label holder and prescribing information.