Wednesday, July 8, 2026

pharma · Non-small Cell Lung Cancer · Epilepsy

Eisai

Eisai drug portfolio — 31 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Tokyo, Japan, JP HQ
41 Employees
NMPA registrant Type
Company details
Intelligence · Drug Pipeline

Eisai pipeline

Portfolio lens on 31 drugs and development assets — regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

Eisai drug portfolio — 31 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

31 compounds
  1. adc

    Development asset linked to Eisai in public FDA and regional records.

  2. Development asset linked to Eisai in public FDA and regional records.

  3. Development asset linked to Eisai in public FDA and regional records.

  4. Development asset linked to Eisai in public FDA and regional records.

  5. bexarotene

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Retinoid X receptor.

    Target
    Retinoid X receptor
    Mechanism
    Retinoid X receptor agonist
  6. Development asset linked to Eisai in public FDA and regional records.

  7. Development asset linked to Eisai in public FDA and regional records.

  8. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  9. carmustine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Glutathione reductase inhibitor
  10. doxorubicin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Eisai's portfolio. Mechanism: DNA topoisomerase II alpha inhibitor.

    Mechanism
    DNA topoisomerase II alpha inhibitor
  11. Development asset linked to Eisai in public FDA and regional records. Molecular target: Fibroblast growth factor receptor 1.

    Target
    Fibroblast growth factor receptor 1
    Mechanism
    Fibroblast growth factor receptor 1 inhibitor
  12. eribulin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Eisai's portfolio. Mechanism: Tubulin inhibitor.

    Mechanism
    Tubulin inhibitor
  13. US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  14. erlotinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Eisai's portfolio. Mechanism: Epidermal growth factor receptor erbB1 inhibitor.

    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  15. Development asset linked to Eisai in public FDA and regional records.

  16. Development asset linked to Eisai in public FDA and regional records.

  17. Development asset linked to Eisai in public FDA and regional records.

  18. lecanemab

    Nervous system (N06)

    Nervous system (N06) compound in Eisai's portfolio. Molecular target: Amyloid-beta precursor protein.

    Target
    Amyloid-beta precursor protein
    Mechanism
    Beta amyloid A4 protein inhibitor
  19. lenvatinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Eisai's portfolio. Mechanism: Vascular endothelial growth factor receptor inhibitor.

    Mechanism
    Vascular endothelial growth factor receptor inhibitor
  20. US regulatory status: approved. Molecular target: Vascular endothelial growth factor receptor.

    Target
    Vascular endothelial growth factor receptor
    Mechanism
    Vascular endothelial growth factor receptor inhibitor
  21. Development asset linked to Eisai in public FDA and regional records.

  22. paclitaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  23. pembrolizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  24. perampanel

    Nervous system (N03)

    US regulatory status: approved. Molecular target: Glutamate receptor ionotropic AMPA.

    Target
    Glutamate receptor ionotropic AMPA
    Mechanism
    Glutamate receptor ionotropic AMPA antagonist
  25. Development asset linked to Eisai in public FDA and regional records.

  26. Development asset linked to Eisai in public FDA and regional records.

  27. Development asset linked to Eisai in public FDA and regional records.

  28. Development asset linked to Eisai in public FDA and regional records.

  29. US regulatory status: approved. Molecular target: Histone-lysine N-methyltransferase EZH2.

    Target
    Histone-lysine N-methyltransferase EZH2
    Mechanism
    Histone-lysine N-methyltransferase EZH2 inhibitor
  30. zonisamide

    Nervous system (N03)

    US regulatory status: approved. Molecular target: Sodium channel alpha subunit.

    Target
    Sodium channel alpha subunit
    Mechanism
    Sodium channel alpha subunit blocker