Friday, July 10, 2026

Drug profile · INN

triptorelin pamoate

triptorelin pamoate (TRELSTAR) is a gonadotropin-releasing hormone receptor agonist. Route of administration: intramuscular. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 2
News articles 0
Drug details — triptorelin pamoate
US status
approved
Class
Route
INTRAMUSCULAR
Patents
0
Programs
2
Data quality
0.84

Quick answer

triptorelin pamoate (TRELSTAR) is a gonadotropin-releasing hormone receptor agonist. Route of administration: intramuscular. Current US regulatory status: approved.

Key facts

INN triptorelin pamoate
Brand TRELSTAR
Mechanism Gonadotropin-releasing hormone receptor agonist
Target Gonadotropin-releasing hormone receptor
Route INTRAMUSCULAR
Formulation FOR SUSPENSION, EXTENDED RELEASE

Mechanism of action

Gonadotropin-releasing hormone receptor agonist

Primary target: Gonadotropin-releasing hormone receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. BAY 1841788 for Hormone Naive Prostate Cancer Phase 2 · Ningbo Cancer Hospital · Hormone Naive Prostate Cancer
  2. triptorelin Unknown · Chinese Academy of · Infertility and at High Risk of OHSS

Related & competitor drugs

  1. cetrorelix acetate Gonadotropin-releasing hormone receptor antagonist
  2. elagolix Gonadotropin-releasing hormone receptor antagonist
  3. ganirelix acetate Gonadotropin-releasing hormone receptor antagonist
  4. leuprolide acetate Gonadotropin-releasing hormone receptor agonist
  5. abarelix Gonadotropin-releasing hormone receptor antagonist
  6. degarelix acetate Gonadotropin-releasing hormone receptor antagonist

Frequently asked questions

What is triptorelin pamoate?

triptorelin pamoate (TRELSTAR) is a gonadotropin-releasing hormone receptor agonist. Route of administration: intramuscular. Current US regulatory status: approved.

What is the brand name for triptorelin pamoate?

TRELSTAR is a marketed brand name for triptorelin pamoate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of triptorelin pamoate?

triptorelin pamoate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.