Wednesday, July 8, 2026

Drug profile · INN

degarelix acetate

degarelix acetate (FIRMAGON) is a gonadotropin-releasing hormone receptor antagonist. Route of administration: subcutaneous. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 3
News articles 0
Drug details — degarelix acetate
US status
approved
Class
Route
SUBCUTANEOUS
Patents
0
Programs
3
Data quality
0.84

Quick answer

degarelix acetate (FIRMAGON) is a gonadotropin-releasing hormone receptor antagonist. Route of administration: subcutaneous. Current US regulatory status: approved.

Key facts

INN degarelix acetate
Brand FIRMAGON
Mechanism Gonadotropin-releasing hormone receptor antagonist
Target Gonadotropin-releasing hormone receptor
Route SUBCUTANEOUS
Formulation POWDER

Mechanism of action

Gonadotropin-releasing hormone receptor antagonist

Primary target: Gonadotropin-releasing hormone receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. CAAA617B12203 Phase 2 · Novartis India · PSMA PET scan positive Castration-Resistant Prostate Cancer
  2. CAAA802A12101 Phase 2 · Novartis India · PSMA-positive metastatic hormone sensitive prostate cancer (
  3. Degarelix Phase 2 · Regeneron UK · Prostate Cancer

Related & competitor drugs

  1. cetrorelix acetate Gonadotropin-releasing hormone receptor antagonist
  2. elagolix Gonadotropin-releasing hormone receptor antagonist
  3. ganirelix acetate Gonadotropin-releasing hormone receptor antagonist
  4. leuprolide acetate Gonadotropin-releasing hormone receptor agonist
  5. abarelix Gonadotropin-releasing hormone receptor antagonist
  6. elagolix sodium Gonadotropin-releasing hormone receptor antagonist

Frequently asked questions

What is degarelix acetate?

degarelix acetate (FIRMAGON) is a gonadotropin-releasing hormone receptor antagonist. Route of administration: subcutaneous. Current US regulatory status: approved.

What is the brand name for degarelix acetate?

FIRMAGON is a marketed brand name for degarelix acetate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of degarelix acetate?

degarelix acetate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.