Wednesday, July 8, 2026

Drug profile · INN

sacituzumab govitecan-hziy

sacituzumab govitecan-hziy (TRODELVY) is a dna topoisomerase i inhibitor. Route of administration: injection. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 1
News articles 2
Drug details — sacituzumab govitecan-hziy

Quick answer

sacituzumab govitecan-hziy (TRODELVY) is a dna topoisomerase i inhibitor. Route of administration: injection. Current US regulatory status: approved.

Key facts

INN sacituzumab govitecan-hziy
Brand TRODELVY
Mechanism DNA topoisomerase I inhibitor
Target DNA topoisomerase 1
Route INJECTION
Formulation INJECTABLE

Mechanism of action

DNA topoisomerase I inhibitor

Primary target: DNA topoisomerase 1

Approval history

Authority Status Date
FDA approved

Recent coverage

Pipeline programs

  1. Sacituzumab Govitecan-hziy Phase 3 · Gilead Sciences Ireland · Triple Negative Breast Cancer

Related & competitor drugs

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  2. irinotecan hydrochloride DNA topoisomerase I inhibitor
  3. fam-trastuzumab deruxtecan-nxki DNA topoisomerase I inhibitor
  4. topotecan hydrochloride DNA topoisomerase I, mitochondrial inhibitor
  5. datopotamab deruxtecan Antineoplastic and immunomodulating agents (L01)
  6. irinotecan hydrochloride trihydrate Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is sacituzumab govitecan-hziy?

sacituzumab govitecan-hziy (TRODELVY) is a dna topoisomerase i inhibitor. Route of administration: injection. Current US regulatory status: approved.

What is the brand name for sacituzumab govitecan-hziy?

TRODELVY is a marketed brand name for sacituzumab govitecan-hziy. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of sacituzumab govitecan-hziy?

sacituzumab govitecan-hziy has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.