Wednesday, July 8, 2026

Drug profile · INN

fam-trastuzumab deruxtecan-nxki

fam-trastuzumab deruxtecan-nxki (ENHERTU) is a dna topoisomerase i inhibitor. Route of administration: injection. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 0
News articles 2
Drug details — fam-trastuzumab deruxtecan-nxki

Quick answer

fam-trastuzumab deruxtecan-nxki (ENHERTU) is a dna topoisomerase i inhibitor. Route of administration: injection. Current US regulatory status: approved.

Key facts

INN fam-trastuzumab deruxtecan-nxki
Brand ENHERTU
Mechanism DNA topoisomerase I inhibitor
Target DNA topoisomerase 1
Route INJECTION
Formulation INJECTABLE

Mechanism of action

DNA topoisomerase I inhibitor

Primary target: DNA topoisomerase 1

Approval history

Authority Status Date
FDA approved

Recent coverage

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Frequently asked questions

What is fam-trastuzumab deruxtecan-nxki?

fam-trastuzumab deruxtecan-nxki (ENHERTU) is a dna topoisomerase i inhibitor. Route of administration: injection. Current US regulatory status: approved.

What is the brand name for fam-trastuzumab deruxtecan-nxki?

ENHERTU is a marketed brand name for fam-trastuzumab deruxtecan-nxki. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of fam-trastuzumab deruxtecan-nxki?

fam-trastuzumab deruxtecan-nxki has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.