Wednesday, July 8, 2026

Drug profile · INN

oxymetazoline hydrochloride

oxymetazoline hydrochloride (UPNEEQ) is a adrenergic receptor alpha agonist. Route of administration: ophthalmic. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 1
Pipeline programs 2
News articles 0
Drug details — oxymetazoline hydrochloride
US status
approved
Class
Route
OPHTHALMIC
Patents
1
Programs
2
Data quality
0.84

Quick answer

oxymetazoline hydrochloride (UPNEEQ) is a adrenergic receptor alpha agonist. Route of administration: ophthalmic. Current US regulatory status: approved.

Key facts

INN oxymetazoline hydrochloride
Brand UPNEEQ
Mechanism Adrenergic receptor alpha agonist
Target Adrenergic receptor alpha
Route OPHTHALMIC
Formulation SOLUTION/DROPS

Mechanism of action

Adrenergic receptor alpha agonist

Primary target: Adrenergic receptor alpha

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. 101380003SA Phase 3 · Santen Oy · Acquired Blepharoptosis
  2. Oxymetazoline Hydrochloride Phase 3 · Teva Pharma · Rosacea

Related & competitor drugs

  1. brimonidine tartrate Adrenergic receptor alpha-2 agonist
  2. carvedilol Adrenergic receptor beta antagonist
  3. clonidine hydrochloride Adrenergic receptor alpha-2 agonist
  4. dexmedetomidine hydrochloride Adrenergic receptor alpha-2 agonist
  5. doxazosin mesylate Adrenergic receptor alpha-1 antagonist
  6. guanfacine hydrochloride Adrenergic receptor alpha-2 agonist

Related patents

  1. US 10335391

    Stabilized oxymetazoline formulations and their uses

    Expires Mon Jun 27 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is oxymetazoline hydrochloride?

oxymetazoline hydrochloride (UPNEEQ) is a adrenergic receptor alpha agonist. Route of administration: ophthalmic. Current US regulatory status: approved.

What is the brand name for oxymetazoline hydrochloride?

UPNEEQ is a marketed brand name for oxymetazoline hydrochloride. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of oxymetazoline hydrochloride?

oxymetazoline hydrochloride has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.