Friday, July 10, 2026

Drug profile · INN

ivabradine

ivabradine (APO-IVABRADINE) is a potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 blocker. Associated with Servier Laboratories (Aust.) Pty.. Route of administration: oral. Current US regulatory status: approved.

FDA: approved EMA: approved TGA: approved Cardiovascular system (C01) C01EB17
US status approved
Patents linked 0
Pipeline programs 3
News articles 0
Drug details — ivabradine
US status
approved
Class
Cardiovascular system (C01)
Route
ORAL
Patents
0
Programs
3
Data quality
0.84

Quick answer

ivabradine (APO-IVABRADINE) is a potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 blocker. Associated with Servier Laboratories (Aust.) Pty.. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN ivabradine
Brand APO-IVABRADINE
Mechanism Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 blocker
Target Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4
Therapeutic class Cardiovascular system (C01)
Route ORAL
Formulation SOLUTION
ATC code C01EB17

Mechanism of action

Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 blocker

Primary target: Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4

Approval history

Authority Status Date
FDA approved
EMA approved
TGA approved

Pipeline programs

  1. P160925J Phase 3 · PARItec · Septic shock
  2. PREVENT-MINS Phase 3 · COLLEGIUM PHARMACEUTICAL · Myocardial Injury after Noncardiac Surgery
  3. Ivabradine + Usual Care Approved · University of Hong · Atrial Fibrillation (Permanent)

Related & competitor drugs

  1. alirocumab Cardiovascular system (C10)
  2. aliskiren Cardiovascular system (C09)
  3. azilsartan medoxomil Cardiovascular system (C09)
  4. bempedoic acid Cardiovascular system (C10)
  5. bosentan Cardiovascular system (C02)
  6. dofetilide Cardiovascular system (C01)

Frequently asked questions

What is ivabradine?

ivabradine (APO-IVABRADINE) is a potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 blocker. Associated with Servier Laboratories (Aust.) Pty.. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for ivabradine?

APO-IVABRADINE is a marketed brand name for ivabradine. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of ivabradine?

ivabradine has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.