Friday, July 10, 2026

Drug profile · INN

inclisiran

inclisiran (LEQVIO) is a pcsk9 mrna rnai inhibitor. Associated with Novartis Pharmaceuticals.

EMA: approved TGA: approved Cardiovascular system (C10) C10AX
Patents linked 0
Pipeline programs 10
News articles 0
Drug details — inclisiran
Class
Cardiovascular system (C10)
Route
Patents
0
Programs
10
Data quality
0.83

Quick answer

inclisiran (LEQVIO) is a pcsk9 mrna rnai inhibitor. Associated with Novartis Pharmaceuticals.

Key facts

INN inclisiran
Brand LEQVIO
Mechanism PCSK9 mRNA RNAi inhibitor
Target PCSK9 mRNA
Therapeutic class Cardiovascular system (C10)
ATC code C10AX

Mechanism of action

PCSK9 mRNA RNAi inhibitor

Primary target: PCSK9 mRNA

Approval history

Authority Status Date
EMA approved
TGA approved

Pipeline programs

  1. CKJX839A12309 Phase 3 · Novartis India · Acute coronary syndrome (ST-elevation myocardial infarction
  2. CKJX839B12302 Phase 3 · Novartis India · Atherosclerotic cardiovascular disease (ASCVD)
  3. CKJX839C12303 Phase 3 · Novartis India · Heterozygous Familial Hypercholesterolemia
  4. CKJX839C12304 Phase 3 · Novartis India · homozygous familial hypercholesterolemia
  5. CKJX839D12303 Phase 3 · Novartis India · Non-obstructive Coronary Artery Disease
  6. CTQJ230A12304 Phase 3 · Novartis India · Atherosclerotic cardiovascular disease (ASCVD)
  7. INCLISIRAN, - Phase 3 · Novartis India · Familial hypercholsterolemia
  8. Inclisiran Phase 3 · Novartis India · Familial Hypercholesterolemia - Heterozygous

Related & competitor drugs

  1. alirocumab Cardiovascular system (C10)
  2. aliskiren Cardiovascular system (C09)
  3. azilsartan medoxomil Cardiovascular system (C09)
  4. bempedoic acid Cardiovascular system (C10)
  5. bosentan Cardiovascular system (C02)
  6. dofetilide Cardiovascular system (C01)

Frequently asked questions

What is inclisiran?

inclisiran (LEQVIO) is a pcsk9 mrna rnai inhibitor. Associated with Novartis Pharmaceuticals.

What is the brand name for inclisiran?

LEQVIO is a marketed brand name for inclisiran. Check FDA Drugs@FDA for the current US label holder and prescribing information.