Friday, July 10, 2026

Drug profile · INN

carvedilol phosphate

carvedilol phosphate (COREG CR) is a adrenergic receptor beta antagonist. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 2
Pipeline programs 0
News articles 0
Drug details — carvedilol phosphate
US status
approved
Class
Route
ORAL
Patents
2
Programs
0
Data quality
0.84

Quick answer

carvedilol phosphate (COREG CR) is a adrenergic receptor beta antagonist. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN carvedilol phosphate
Brand COREG CR
Mechanism Adrenergic receptor beta antagonist
Target Adrenergic receptor alpha-1
Route ORAL
Formulation CAPSULE, EXTENDED RELEASE

Mechanism of action

Adrenergic receptor beta antagonist

Primary target: Adrenergic receptor alpha-1

Approval history

Authority Status Date
FDA approved

Related & competitor drugs

  1. carvedilol Adrenergic receptor beta antagonist
  2. doxazosin mesylate Adrenergic receptor alpha-1 antagonist
  3. midodrine hydrochloride Adrenergic receptor alpha-1 agonist
  4. phenylephrine hydrochloride Adrenergic receptor alpha-1 agonist
  5. prazosin hydrochloride Adrenergic receptor alpha-1 antagonist
  6. tamsulosin hydrochloride Adrenergic receptor alpha-1 antagonist

Related patents

  1. US 8124644

    Carvedilol phosphate

    Expires Mon Feb 23 2032 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 8022094

    Carvedilol phosphate

    Expires Mon Sep 15 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is carvedilol phosphate?

carvedilol phosphate (COREG CR) is a adrenergic receptor beta antagonist. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for carvedilol phosphate?

COREG CR is a marketed brand name for carvedilol phosphate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of carvedilol phosphate?

carvedilol phosphate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.