Wednesday, July 8, 2026

Drug profile · INN

cabergoline

cabergoline (CABASER) is a dopamine d2 receptor agonist. Associated with Pfizer Australia Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

FDA: approved TGA: approved NMPA: clinical trials
US status approved
Patents linked 20
Pipeline programs 1
News articles 0
Drug details — cabergoline
US status
approved
Class
Route
ORAL
Patents
20
Programs
1
Data quality
0.89

Quick answer

cabergoline (CABASER) is a dopamine d2 receptor agonist. Associated with Pfizer Australia Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN cabergoline
Brand CABASER
Mechanism Dopamine D2 receptor agonist
Target D(2) dopamine receptor
Route ORAL
Formulation TABLET

Mechanism of action

Dopamine D2 receptor agonist

Primary target: D(2) dopamine receptor

Approval history

Authority Status Date
FDA approved
TGA approved
NMPA clinical trials

Pipeline programs

  1. Cabergoline 1 MG Phase 2 · Monte Rosa Therapeutics · Lactation Suppressed

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Frequently asked questions

What is cabergoline?

cabergoline (CABASER) is a dopamine d2 receptor agonist. Associated with Pfizer Australia Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for cabergoline?

CABASER is a marketed brand name for cabergoline. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of cabergoline?

cabergoline has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.