Wednesday, June 10, 2026

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Sanofi-Aventis U.S

Sanofi-Aventis U.S drug portfolio β€” 148 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Bridgewater, USA HQ
177 Employees
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Company details
Status
Public
HQ
Bridgewater, USA
Employees
177
Programs
117
Drugs
148
Patents
0
Intelligence Β· Drug Pipeline

Sanofi-Aventis U.S pipeline

Portfolio lens on 148 drugs and development assets β€” regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

Sanofi-Aventis U.S drug portfolio β€” 148 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

148 compounds
  1. abemaciclib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Cyclin-dependent kinase 4.

    Target
    Cyclin-dependent kinase 4
    Mechanism
    Cyclin-dependent kinase 6 inhibitor
  2. afamelanotide

    Dermatologicals (D02)

    US regulatory status: approved. Molecular target: Melanocyte-stimulating hormone receptor.

    Target
    Melanocyte-stimulating hormone receptor
    Mechanism
    Melanocortin receptor 1 agonist
  3. agalsidase alfa

    Alimentary tract and metabolism (A16)

    Alimentary tract and metabolism (A16) compound in Sanofi-Aventis U.S's portfolio. Molecular target: Globotriosylceramide.

    Target
    Globotriosylceramide
    Mechanism
    Globotriosylceramide hydrolytic enzyme
  4. agalsidase beta

    Alimentary tract and metabolism (A16)

    US regulatory status: approved. Molecular target: Globotriosylceramide.

    Target
    Globotriosylceramide
    Mechanism
    Globotriosylceramide hydrolytic enzyme
  5. US regulatory status: approved. Molecular target: Beta-2 adrenergic receptor.

    Target
    Beta-2 adrenergic receptor
    Mechanism
    Beta-2 adrenergic receptor agonist
  6. US regulatory status: approved. Molecular target: Beta-2 adrenergic receptor.

    Target
    Beta-2 adrenergic receptor
    Mechanism
    Beta-2 adrenergic receptor agonist
  7. alemtuzumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: CAMPATH-1 antigen.

    Target
    CAMPATH-1 antigen
    Mechanism
    CAMPATH-1 antigen inhibitor
  8. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Mechanism: Adrenergic receptor alpha-1 agonist.

    Mechanism
    Adrenergic receptor alpha-1 agonist
  9. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Molecular target: Starch.

    Target
    Starch
    Mechanism
    Starch hydrolytic enzyme
  10. alglucosidase alfa

    Alimentary tract and metabolism (A16)

    US regulatory status: approved. Molecular target: Starch.

    Target
    Starch
    Mechanism
    Starch hydrolytic enzyme
  11. alpha1-proteinase inhibitor (human)

    Blood and blood forming organs (B02)

    Blood and blood forming organs (B02) compound in Sanofi-Aventis U.S's portfolio. Molecular target: Neutrophil elastase.

    Target
    Neutrophil elastase
    Mechanism
    Leukocyte elastase inhibitor
  12. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  13. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  14. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  15. avalglucosidase alfa

    Alimentary tract and metabolism (A16)

    Alimentary tract and metabolism (A16) compound in Sanofi-Aventis U.S's portfolio. Molecular target: Glycogen.

    Target
    Glycogen
    Mechanism
    Glycogen hydrolytic enzyme
  16. beclometasone

    Respiratory system (R03)

    Respiratory system (R03) compound in Sanofi-Aventis U.S's portfolio.

  17. belumosudil

    Antineoplastic and immunomodulating agents (L04)

    Antineoplastic and immunomodulating agents (L04) compound in Sanofi-Aventis U.S's portfolio. Molecular target: Rho-associated protein kinase 2.

    Target
    Rho-associated protein kinase 2
    Mechanism
    Rho-associated protein kinase inhibitor
  18. bevacizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Vascular endothelial growth factor A, long form.

    Target
    Vascular endothelial growth factor A, long form
    Mechanism
    Vascular endothelial growth factor A inhibitor
  19. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  20. bortezomib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  21. budesonide

    Alimentary tract and metabolism (A07)

    US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  22. canakinumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Interleukin-1 beta.

    Target
    Interleukin-1 beta
    Mechanism
    Interleukin-1 beta inhibitor
  23. caplacizumab

    Blood and blood forming organs (B01)

    Blood and blood forming organs (B01) compound in Sanofi-Aventis U.S's portfolio. Molecular target: von Willebrand factor.

    Target
    von Willebrand factor
    Mechanism
    von Willebrand factor inhibitor
  24. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  25. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  26. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  27. carfilzomib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  28. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  29. cemiplimab

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Sanofi-Aventis U.S's portfolio. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  30. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  31. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Mechanism: Histamine H1 receptor antagonist.

    Mechanism
    Histamine H1 receptor antagonist
  32. cetuximab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  33. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  34. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Mechanism: Histamine H1 receptor antagonist.

    Mechanism
    Histamine H1 receptor antagonist
  35. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  36. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Molecular target: Bile acids.

    Target
    Bile acids
    Mechanism
    Bile acids sequestering agent
  37. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  38. covid-19 vaccine (inactivated, adjuvanted, adsorbed)

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in Sanofi-Aventis U.S's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  39. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  40. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  41. dexamethasone phosphate

    Systemic hormonal preparations (H02)

    Systemic hormonal preparations (H02) compound in Sanofi-Aventis U.S's portfolio.

  42. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  43. US regulatory status: approved. Molecular target: Sodium-dependent dopamine transporter.

    Target
    Sodium-dependent dopamine transporter
    Mechanism
    Norepinephrine transporter inhibitor
  44. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Mechanism: Voltage-gated L-type calcium channel blocker.

    Mechanism
    Voltage-gated L-type calcium channel blocker
  45. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Mechanism: Histamine H1 receptor antagonist.

    Mechanism
    Histamine H1 receptor antagonist
  46. US regulatory status: approved. Molecular target: Histamine H1 receptor.

    Target
    Histamine H1 receptor
    Mechanism
    Histamine H1 receptor antagonist
  47. docetaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  48. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  49. dupilumab

    Dermatologicals (D11)

    US regulatory status: approved. Molecular target: Interleukin-4 receptor subunit alpha.

    Target
    Interleukin-4 receptor subunit alpha
    Mechanism
    Interleukin-4 receptor subunit alpha antagonist
  50. emicizumab

    Blood and blood forming organs (B02)

    US regulatory status: approved. Molecular target: Coagulation factor IX and X.

    Target
    Coagulation factor IX and X
    Mechanism
    Coagulation factor IX and X other
  51. enoxaparin sodium

    Blood and blood forming organs (B01)

    US regulatory status: approved. Molecular target: Antithrombin-III.

    Target
    Antithrombin-III
    Mechanism
    Antithrombin-III activator
  52. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  53. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  54. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Mechanism: Histamine H1 receptor antagonist.

    Mechanism
    Histamine H1 receptor antagonist
  55. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  56. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  57. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  58. US regulatory status: approved. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  59. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  60. glibenclamide

    Alimentary tract and metabolism (A10)

    Alimentary tract and metabolism (A10) compound in Sanofi-Aventis U.S's portfolio. Molecular target: Sulfonylurea receptor 1, Kir6.2.

    Target
    Sulfonylurea receptor 1, Kir6.2
    Mechanism
    Sulfonylurea receptor 1, Kir6.2 blocker
  61. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Molecular target: Soluble guanylate cyclase.

    Target
    Soluble guanylate cyclase
    Mechanism
    Soluble guanylate cyclase activator
  62. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  63. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  64. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  65. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  66. human heterologous liver cells

    Alimentary tract and metabolism (A16)

    Alimentary tract and metabolism (A16) compound in Sanofi-Aventis U.S's portfolio.

  67. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Mechanism: Toll-like receptor 7 antagonist.

    Mechanism
    Toll-like receptor 7 antagonist
  68. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  69. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  70. imiglucerase

    Alimentary tract and metabolism (A16)

    US regulatory status: approved. Molecular target: Glucocerebroside.

    Target
    Glucocerebroside
    Mechanism
    Glucocerebroside hydrolytic enzyme
  71. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  72. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  73. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  74. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  75. insulin glargine

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  76. insulin glulisine

    Alimentary tract and metabolism (A10)

    Alimentary tract and metabolism (A10) compound in Sanofi-Aventis U.S's portfolio. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  77. isatuximab

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Sanofi-Aventis U.S's portfolio. Molecular target: ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1.

    Target
    ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
    Mechanism
    Lymphocyte differentiation antigen CD38 inhibitor
  78. lenalidomide

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: CRL4(CRBN) E3 ubiquitin ligase.

    Target
    CRL4(CRBN) E3 ubiquitin ligase
    Mechanism
    CRL4(CRBN) E3 ubiquitin ligase inhibitor
  79. US regulatory status: approved. Molecular target: Progesterone receptor.

    Target
    Progesterone receptor
    Mechanism
    Progesterone receptor agonist
  80. US regulatory status: approved. Molecular target: Histamine H1 receptor.

    Target
    Histamine H1 receptor
    Mechanism
    Histamine H1 receptor antagonist
  81. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  82. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  83. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  84. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  85. methotrexate

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Dihydrofolate reductase.

    Target
    Dihydrofolate reductase
    Mechanism
    Dihydrofolate reductase inhibitor
  86. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  87. migalastat

    Alimentary tract and metabolism (A16)

    Alimentary tract and metabolism (A16) compound in Sanofi-Aventis U.S's portfolio. Molecular target: Alpha-galactosidase A.

    Target
    Alpha-galactosidase A
    Mechanism
    Alpha-galactosidase A stabiliser
  88. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  89. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  90. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Mechanism: Cysteinyl leukotriene receptor 1 antagonist.

    Mechanism
    Cysteinyl leukotriene receptor 1 antagonist
  91. US regulatory status: approved. Molecular target: Cannabinoid receptor 1.

    Target
    Cannabinoid receptor 1
    Mechanism
    Cannabinoid CB1 receptor agonist
  92. US regulatory status: approved. Molecular target: Progesterone receptor.

    Target
    Progesterone receptor
    Mechanism
    Progesterone receptor agonist
  93. oxybutynin

    Genito-urinary system and sex hormones (G04)

    US regulatory status: approved. Molecular target: Muscarinic acetylcholine receptor M2.

    Target
    Muscarinic acetylcholine receptor M2
    Mechanism
    Muscarinic acetylcholine receptor M2 antagonist
  94. palbociclib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: CDK6/cyclin D1.

    Target
    CDK6/cyclin D1
    Mechanism
    Cyclin-dependent kinase 4/cyclin D1 inhibitor
  95. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Molecular target: Fatty-acid amide hydrolase 1.

    Target
    Fatty-acid amide hydrolase 1
    Mechanism
    Anandamide amidohydrolase inhibitor
  96. pembrolizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  97. US regulatory status: approved. Molecular target: Dihydrofolate reductase.

    Target
    Dihydrofolate reductase
    Mechanism
    Thymidylate synthase inhibitor
  98. US regulatory status: approved. Molecular target: Peptidyl-prolyl cis-trans isomerase FKBP1A.

    Target
    Peptidyl-prolyl cis-trans isomerase FKBP1A
    Mechanism
    FK506-binding protein 1A inhibitor
  99. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  100. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  101. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  102. pomalidomide

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: CRL4(CRBN) E3 ubiquitin ligase.

    Target
    CRL4(CRBN) E3 ubiquitin ligase
    Mechanism
    CRL4(CRBN) E3 ubiquitin ligase inhibitor
  103. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  104. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  105. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  106. US regulatory status: approved. Molecular target: Histamine H1 receptor.

    Target
    Histamine H1 receptor
    Mechanism
    Histamine H1 receptor antagonist
  107. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  108. riluzole

    Nervous system (N07)

    US regulatory status: approved. Molecular target: Sodium channel alpha subunit.

    Target
    Sodium channel alpha subunit
    Mechanism
    Sodium channel alpha subunit blocker
  109. rilzabrutinib

    Nervous system (NOT)

    US regulatory status: approved. Molecular target: Tyrosine-protein kinase BTK.

    Target
    Tyrosine-protein kinase BTK
    Mechanism
    Tyrosine-protein kinase BTK inhibitor
  110. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  111. rotavirus vaccine

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in Sanofi-Aventis U.S's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  112. rotavirus vaccine, live

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in Sanofi-Aventis U.S's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  113. salmeterol

    Respiratory system (R03)

    Respiratory system (R03) compound in Sanofi-Aventis U.S's portfolio. Mechanism: Beta-2 adrenergic receptor agonist.

    Mechanism
    Beta-2 adrenergic receptor agonist
  114. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  115. sarilumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Interleukin-6 receptor subunit alpha.

    Target
    Interleukin-6 receptor subunit alpha
    Mechanism
    Interleukin-6 receptor alpha subunit antagonist
  116. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  117. sevelamer

    Various (V03)

    Various (V03) compound in Sanofi-Aventis U.S's portfolio.

  118. US regulatory status: approved. Molecular target: Potassium.

    Target
    Potassium
    Mechanism
    Potassium sequestering agent
  119. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  120. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  121. spesolimab

    Antineoplastic and immunomodulating agents (L04)

    Antineoplastic and immunomodulating agents (L04) compound in Sanofi-Aventis U.S's portfolio. Molecular target: IL36 receptor.

    Target
    IL36 receptor
    Mechanism
    IL36 receptor antagonist
  122. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  123. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  124. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  125. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  126. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  127. tacrolimus

    Dermatologicals (D11)

    US regulatory status: approved. Molecular target: Peptidyl-prolyl cis-trans isomerase FKBP1A.

    Target
    Peptidyl-prolyl cis-trans isomerase FKBP1A
    Mechanism
    FK506-binding protein 1A inhibitor
  128. teplizumab

    Alimentary tract and metabolism (A10)

    Alimentary tract and metabolism (A10) compound in Sanofi-Aventis U.S's portfolio. Molecular target: T-cell surface glycoprotein CD3 epsilon chain.

    Target
    T-cell surface glycoprotein CD3 epsilon chain
    Mechanism
    T-cell surface glycoprotein CD3 epsilon chain other
  129. teriflunomide

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Dihydroorotate dehydrogenase (quinone), mitochondrial.

    Target
    Dihydroorotate dehydrogenase (quinone), mitochondrial
    Mechanism
    Dihydroorotate dehydrogenase inhibitor
  130. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  131. thyrotropin alfa

    Systemic hormonal preparations (H01)

    US regulatory status: approved. Molecular target: Thyrotropin receptor.

    Target
    Thyrotropin receptor
    Mechanism
    Thyroid stimulating hormone receptor agonist
  132. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records. Molecular target: Tyrosine-protein kinase BTK.

    Target
    Tyrosine-protein kinase BTK
    Mechanism
    Tyrosine-protein kinase BTK inhibitor
  133. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  134. Development asset linked to Sanofi-Aventis U.S in public FDA and regional records.

  135. vigabatrin

    Nervous system (N03)

    US regulatory status: approved. Molecular target: 4-aminobutyrate aminotransferase, mitochondrial.

    Target
    4-aminobutyrate aminotransferase, mitochondrial
    Mechanism
    Gamma-amino-N-butyrate transaminase inhibitor