Friday, July 10, 2026

Drug profile · INN

tolebrutinib

tolebrutinib (CENRIFKI) is a tyrosine-protein kinase btk inhibitor.

EMA: unknown
Patents linked 0
Pipeline programs 4
News articles 0
Drug details — tolebrutinib
Class
Route
Patents
0
Programs
4
Data quality
0.83

Quick answer

tolebrutinib (CENRIFKI) is a tyrosine-protein kinase btk inhibitor.

Key facts

INN tolebrutinib
Brand CENRIFKI
Mechanism Tyrosine-protein kinase BTK inhibitor
Target Tyrosine-protein kinase BTK

Mechanism of action

Tyrosine-protein kinase BTK inhibitor

Primary target: Tyrosine-protein kinase BTK

Approval history

Authority Status Date
EMA unknown

Pipeline programs

  1. EFC16035 Phase 3 · Genzyme Europe · Primary Progressive Multiple Sclerosis
  2. LTS17043 Phase 3 · Sanofi-Aventis U.S · Nervous system diseases
  3. LTS17043 Phase 3 · Sanofi-Aventis U.S · Nervous system diseases
  4. Tolebrutinib Phase 3 · Sanofi Pasteur MSD · Non-relapsing Secondary Progressive Multiple Sclerosis

Related & competitor drugs

  1. ibrutinib Antineoplastic and immunomodulating agents (L01)
  2. zanubrutinib Antineoplastic and immunomodulating agents (L01)
  3. acalabrutinib Antineoplastic and immunomodulating agents (L01)
  4. acalabrutinib maleate Tyrosine-protein kinase BTK inhibitor
  5. pirtobrutinib Antineoplastic and immunomodulating agents (L01)
  6. rilzabrutinib Nervous system (NOT)

Frequently asked questions

What is tolebrutinib?

tolebrutinib (CENRIFKI) is a tyrosine-protein kinase btk inhibitor.

What is the brand name for tolebrutinib?

CENRIFKI is a marketed brand name for tolebrutinib. Check FDA Drugs@FDA for the current US label holder and prescribing information.