Wednesday, June 10, 2026

pharma Β· Renal Transplantation Β· Rheumatoid Arthritis (RA)

Astellas Pharma

Astellas Pharma drug portfolio β€” 12 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

2-5-1, Nihonbashi-Honcho, Chuo-Ku, Tokyo 103-8411, JP HQ
12,378 Employees
NMPA registrant Type
Company details
Status
Public
HQ
2-5-1, Nihonbashi-Honcho, Chuo-Ku, Tokyo 103-8411, JP
Employees
12,378
Programs
20
Drugs
12
Patents
25
Intelligence Β· Drug Pipeline

Astellas Pharma pipeline

Portfolio lens on 12 drugs and development assets β€” regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

Astellas Pharma drug portfolio β€” 12 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

12 compounds
  1. Development asset linked to Astellas Pharma in public FDA and regional records.

  2. enfortumab vedotin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Astellas Pharma's portfolio. Molecular target: Nectin-4.

    Target
    Nectin-4
    Mechanism
    Tubulin inhibitor
  3. enzalutamide

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  4. fezolinetant

    Genito-urinary system and sex hormones (G02)

    US regulatory status: approved. Molecular target: Neuromedin-K receptor.

    Target
    Neuromedin-K receptor
    Mechanism
    Neurokinin 3 receptor antagonist
  5. gilteritinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Astellas Pharma's portfolio. Molecular target: Receptor-type tyrosine-protein kinase FLT3.

    Target
    Receptor-type tyrosine-protein kinase FLT3
    Mechanism
    Tyrosine-protein kinase receptor FLT3 inhibitor
  6. isavuconazole

    Antiinfectives for systemic use (J02)

    Antiinfectives for systemic use (J02) compound in Astellas Pharma's portfolio.

  7. linaclotide

    Alimentary tract and metabolism (A06)

    US regulatory status: approved. Molecular target: Guanylyl cyclase C.

    Target
    Guanylyl cyclase C
    Mechanism
    Heat-stable enterotoxin receptor agonist
  8. mirabegron

    Genito-urinary system and sex hormones (G04)

    US regulatory status: approved. Molecular target: Beta-3 adrenergic receptor.

    Target
    Beta-3 adrenergic receptor
    Mechanism
    Beta-3 adrenergic receptor agonist
  9. US regulatory status: approved. Mechanism: Supplement.

    Mechanism
    Supplement
  10. Development asset linked to Astellas Pharma in public FDA and regional records. Molecular target: Serotonin 3 (5-HT3) receptor.

    Target
    Serotonin 3 (5-HT3) receptor
    Mechanism
    Serotonin 3 (5-HT3) receptor antagonist
  11. tacrolimus

    Dermatologicals (D11)

    US regulatory status: approved. Molecular target: Peptidyl-prolyl cis-trans isomerase FKBP1A.

    Target
    Peptidyl-prolyl cis-trans isomerase FKBP1A
    Mechanism
    FK506-binding protein 1A inhibitor
  12. Development asset linked to Astellas Pharma in public FDA and regional records.