Saturday, July 11, 2026

Patent directory · USPTO A61K / A61P

Patents matching “derivative”

1,342 pharma patents match "derivative" in our USPTO index (A61K/A61P) — applicant, grant date, expiration, and drug links.

Matches 1,342
Index total 30,257
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This filtered view shows 1,342 pharmaceutical patents matching "derivative" in our USPTO PatentsView index (CPC A61K/A61P). Search matches patent number, title, applicant, and CPC classification codes.

Patent results

1,342 results for “derivative” · 30,257 patents in full index Clear search

  1. US 8329687

    Pyridooxazepine derivative and use thereof

    Takeda Pharmaceutical Company Limited · Granted Dec 11, 2012 · Expires Dec 6, 2032

    granted
  2. US 8329664

    Anti-viral pyrimidine nucleoside derivatives

    University College Cardiff Consultants Limited · Granted Dec 11, 2012 · Expires Dec 6, 2032

    granted
  3. US 8324201

    Pyrazinooxazepine derivatives

    Takeda Pharmaceutical Company Limited · Granted Dec 4, 2012 · Expires Nov 29, 2032

    granted
  4. US 8318765

    3-carboxypropyl-aminotetralin derivatives and related compounds as mu opioid receptor antagonists

    Theravance, Inc. · Granted Nov 27, 2012 · Expires Nov 22, 2032

    granted
  5. US 8318722

    Pyrazinooxazepine derivatives

    Takeda Pharmaceutical Company Limited · Granted Nov 27, 2012 · Expires Nov 22, 2032

    granted
  6. US 8314125

    Bicyclic derivatives as modulators of ion channels

    Vertex Pharmaceuticals Incorporated · Granted Nov 20, 2012 · Expires Nov 15, 2032

    granted
  7. US 8314088

    Pyrazinooxazepine derivatives

    Takeda Pharmaceutical Company Limited · Granted Nov 20, 2012 · Expires Nov 15, 2032

    granted
  8. US 8309766

    Phenyl-containing n-acyl amine and aminoacid derivatives, methods for the production thereof, a pharmaceutical composition and the use thereof

    OBSCHESTVO S OGRANICHENNOI OTVETSTVENNOSTIYU “PHARMENTERPRISES” · Granted Nov 13, 2012 · Expires Nov 8, 2032

    granted
  9. US 8304511

    Maleamic acid polymer derivatives and their bioconjugates

    Nektar Therapeutics · Granted Nov 6, 2012 · Expires Nov 1, 2032

    granted
  10. US 8304557

    Fused heterocycle derivatives and use thereof

    Takeda Pharmaceutical Company Limited · Granted Nov 6, 2012 · Expires Nov 1, 2032

    granted
  11. US 8299261

    1-heterocyclylsulfonyl, 3-aminomethyl, 5-(hetero-) aryl substituted 1-H-pyrrole derivatives as acid secretion inhibitors

    Takeda Pharmaceutical Company Limited · Granted Oct 30, 2012 · Expires Oct 25, 2032

    granted
  12. US 8299101

    1,4-disubstituted 3-cyano-pyridone derivatives and their use as positive mGluR2-receptor modulators

    Addex Pharma, S.A. · Granted Oct 30, 2012 · Expires Oct 25, 2032

    granted
  13. US 8299099

    Heteroaryl derivatives as CFTR modulators

    Vertex Pharmaceuticals Incorporated · Granted Oct 30, 2012 · Expires Oct 25, 2032

    granted
  14. US 8293800

    Quinone derivative 2,3-dimethoxy-5-methyl-6-(10-hydroxydecyl)-1,4-benzoquinone for the treatment of primary progressive multiple sclerosis

    The United States of America, as represented by the Secretary, Department of Health and Human Services · Granted Oct 23, 2012 · Expires Oct 18, 2032

    granted
  15. US 8288390

    Benzofuran derivatives

    Takeda Pharmaceutical Company Limited · Granted Oct 16, 2012 · Expires Oct 11, 2032

    granted
  16. US 8283370

    Imidazolidinedione derivatives as antimalarial agents, preparation thereof, and methods of use

    The United States of America as represented by the Secretary of the Army · Granted Oct 9, 2012 · Expires Oct 4, 2032

    granted
  17. US 8269026

    Lupane derivatives useful for treating HIV

    Vertex Pharmaceuticals Incorporated · Granted Sep 18, 2012 · Expires Sep 13, 2032

    granted
  18. US 8268777

    Oximyl macrocyclic derivatives

    Enanta Pharmaceuticals, Inc. · Granted Sep 18, 2012 · Expires Sep 13, 2032

    granted
  19. US 8263632

    Aminopyridine derivatives having Aurora A selective inhibitory action

    Vertex Pharmaceuticals Incorporated · Granted Sep 11, 2012 · Expires Sep 6, 2032

    granted
  20. US 8263762

    Alkoxy-carbonyl-amino-alkynyl-adenosine compounds and derivatives thereof as A2AR agonists

    Dogwood Pharmaceuticals, Inc. · Granted Sep 11, 2012 · Expires Sep 6, 2032

    granted
  21. US 8258308

    Amino nicotinic and isonicotinic acid derivatives as DHODH inhibitors

    Laboratories Almirall, S.A. · Granted Sep 4, 2012 · Expires Aug 30, 2032

    granted
  22. US 8258122

    3-([1,2,4]triazolo[4,3-a]pyridin-7-yl)benzamide derivatives

    Almirall, S.A. · Granted Sep 4, 2012 · Expires Aug 30, 2032

    granted
  23. US 8247421

    5-cyano-4-(pyrrolo [2,3B] pyridine-3-yl)-pyrimidine derivatives useful as protein kinase inhibitors

    Vertex Pharmaceuticals Incorporated · Granted Aug 21, 2012 · Expires Aug 16, 2032

    granted
  24. US 8247410

    Pyrimidine substituted purine derivatives

    VERASTEM, INC. · Granted Aug 21, 2012 · Expires Aug 16, 2032

    granted