Wednesday, July 8, 2026

Drug profile · INN

valdecoxib

valdecoxib (BEXTRA) is a cyclooxygenase-2 inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved EMA: withdrawn Musculo-skeletal system (M01) M01AH03
US status approved
Patents linked 0
Pipeline programs 1
News articles 0
Drug details — valdecoxib
US status
approved
Class
Musculo-skeletal system (M01)
Route
ORAL
Patents
0
Programs
1
Data quality
0.84

Quick answer

valdecoxib (BEXTRA) is a cyclooxygenase-2 inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN valdecoxib
Brand BEXTRA
Mechanism Cyclooxygenase-2 inhibitor
Target Prostaglandin G/H synthase 2
Therapeutic class Musculo-skeletal system (M01)
Route ORAL
Formulation TABLET
ATC code M01AH03

Mechanism of action

Cyclooxygenase-2 inhibitor

Primary target: Prostaglandin G/H synthase 2

Approval history

Authority Status Date
FDA approved
EMA withdrawn

Pipeline programs

  1. valdecoxib Approved · Pfizer · Pain, Postoperative

Related & competitor drugs

  1. allopurinol Musculo-skeletal system (M04)
  2. celecoxib Antineoplastic and immunomodulating agents (L01)
  3. colchicine Musculo-skeletal system (M04)
  4. denosumab Musculo-skeletal system (M05)
  5. eteplirsen Musculo-skeletal system (M09)
  6. etodolac Cyclooxygenase-2 inhibitor

Frequently asked questions

What is valdecoxib?

valdecoxib (BEXTRA) is a cyclooxygenase-2 inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for valdecoxib?

BEXTRA is a marketed brand name for valdecoxib. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of valdecoxib?

valdecoxib has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.