Saturday, July 11, 2026

Drug profile · INN

umeclidinium bromide/ vilanterol trifenatate

umeclidinium bromide/ vilanterol trifenatate (ANORO ELLIPTA) is a muscarinic acetylcholine receptor m3 antagonist.

PMDA: approved
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Drug details — umeclidinium bromide/ vilanterol trifenatate
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Quick answer

umeclidinium bromide/ vilanterol trifenatate (ANORO ELLIPTA) is a muscarinic acetylcholine receptor m3 antagonist.

Key facts

INN umeclidinium bromide/ vilanterol trifenatate
Brand ANORO ELLIPTA
Mechanism Muscarinic acetylcholine receptor M3 antagonist
Target Muscarinic acetylcholine receptor M3

Mechanism of action

Muscarinic acetylcholine receptor M3 antagonist

Primary target: Muscarinic acetylcholine receptor M3

Approval history

Authority Status Date
PMDA approved

Related & competitor drugs

  1. ipratropium bromide Muscarinic acetylcholine receptor M3 antagonist
  2. acetylcholine chloride Muscarinic acetylcholine receptor M3 agonist
  3. aclidinium bromide Respiratory system (R03)
  4. carbachol Muscarinic acetylcholine receptor M3 agonist
  5. cyclopentolate hydrochloride Muscarinic acetylcholine receptor M3 antagonist
  6. methacholine chloride Muscarinic acetylcholine receptor M3 agonist

Frequently asked questions

What is umeclidinium bromide/ vilanterol trifenatate?

umeclidinium bromide/ vilanterol trifenatate (ANORO ELLIPTA) is a muscarinic acetylcholine receptor m3 antagonist.

What is the brand name for umeclidinium bromide/ vilanterol trifenatate?

ANORO ELLIPTA is a marketed brand name for umeclidinium bromide/ vilanterol trifenatate. Check FDA Drugs@FDA for the current US label holder and prescribing information.