Wednesday, July 8, 2026

Drug profile · INN

acetylcholine chloride

acetylcholine chloride (MIOCHOL) is a muscarinic acetylcholine receptor m3 agonist. Route of administration: ophthalmic. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 1
Pipeline programs 2
News articles 0
Drug details — acetylcholine chloride
US status
approved
Class
Route
OPHTHALMIC
Patents
1
Programs
2
Data quality
0.84

Quick answer

acetylcholine chloride (MIOCHOL) is a muscarinic acetylcholine receptor m3 agonist. Route of administration: ophthalmic. Current US regulatory status: approved.

Key facts

INN acetylcholine chloride
Brand MIOCHOL
Mechanism Muscarinic acetylcholine receptor M3 agonist
Target Muscarinic acetylcholine receptor M3
Route OPHTHALMIC
Formulation FOR SOLUTION

Mechanism of action

Muscarinic acetylcholine receptor M3 agonist

Primary target: Muscarinic acetylcholine receptor M3

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. Choline Chloride for Injection Phase 3 · Protara Therapeutics · Choline Deficiency
  2. PROMISE Approved · Telethon Foundation · Myocardial infarction with non-obstructive coronary arteries

Related & competitor drugs

  1. ipratropium bromide Muscarinic acetylcholine receptor M3 antagonist
  2. aclidinium bromide Respiratory system (R03)
  3. carbachol Muscarinic acetylcholine receptor M3 agonist
  4. cyclopentolate hydrochloride Muscarinic acetylcholine receptor M3 antagonist
  5. methacholine chloride Muscarinic acetylcholine receptor M3 agonist
  6. revefenacin Muscarinic acetylcholine receptor M3 antagonist

Related patents

  1. US 11472840

    Acetylcholine receptor-binding peptide

    Expires Mon Oct 13 2042 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is acetylcholine chloride?

acetylcholine chloride (MIOCHOL) is a muscarinic acetylcholine receptor m3 agonist. Route of administration: ophthalmic. Current US regulatory status: approved.

What is the brand name for acetylcholine chloride?

MIOCHOL is a marketed brand name for acetylcholine chloride. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of acetylcholine chloride?

acetylcholine chloride has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.