Friday, July 10, 2026

Drug profile · INN

pirtobrutinib

pirtobrutinib (JAYPIRCA) is a tyrosine-protein kinase btk inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved EMA: approved PMDA: approved NMPA: clinical trials Antineoplastic and immunomodulating agents (L01) L01
US status approved
Patents linked 0
Pipeline programs 11
News articles 2
Drug details — pirtobrutinib

Quick answer

pirtobrutinib (JAYPIRCA) is a tyrosine-protein kinase btk inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN pirtobrutinib
Brand JAYPIRCA
Mechanism Tyrosine-protein kinase BTK inhibitor
Target Tyrosine-protein kinase BTK
Therapeutic class Antineoplastic and immunomodulating agents (L01)
Route ORAL
Formulation TABLET
ATC code L01

Mechanism of action

Tyrosine-protein kinase BTK inhibitor

Primary target: Tyrosine-protein kinase BTK

Approval history

Authority Status Date
FDA approved
EMA approved
PMDA approved
NMPA clinical trials

Recent coverage

Pipeline programs

  1. BGB-16673-304 Phase 3 · BEONE MEDICINES AUS · Chronic lymphocytic leukemia (CLL), Small lymphocytic lympho
  2. LOXO-BTK-20019 Phase 3 · Createrna Science and · Mantle cell lymphoma
  3. LOXO-BTK-20020 Phase 3 · Createrna Science and · Chronic Lymphocytic Leukemia/Small Lymphocytic Lymphoma
  4. LOXO-BTK-20022 Phase 3 · Createrna Science and · Chronic Lymphocytic Leukemia/Small Lymphocytic Lymphoma (BRU
  5. LOXO-BTK-20023 Phase 3 · Createrna Science and · Chronic Lymphocytic Leukemia/Small Lymphocytic Lymphoma
  6. LOXO-BTK-20030 Phase 3 · Createrna Science and · Chronic Lymphocytic Leukemia/Small Lymphocytic Lymphoma
  7. GCT3013-03 Phase 2 · Genmab · Chronic Lymphocytic Leukemia
  8. M22-132 Phase 2 · AbbVie Deutschland GmbH · B-cell Non-Hodgkin's lymphoma, diffuse large B-cell lymphoma

Related & competitor drugs

  1. abiraterone acetate Antineoplastic and immunomodulating agents (L02)
  2. anagrelide Antineoplastic and immunomodulating agents (L01)
  3. apremilast Antineoplastic and immunomodulating agents (L04)
  4. arsenic trioxide Antineoplastic and immunomodulating agents (L01)
  5. axitinib Antineoplastic and immunomodulating agents (L01)
  6. azacitidine Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is pirtobrutinib?

pirtobrutinib (JAYPIRCA) is a tyrosine-protein kinase btk inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for pirtobrutinib?

JAYPIRCA is a marketed brand name for pirtobrutinib. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of pirtobrutinib?

pirtobrutinib has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.