Saturday, July 11, 2026

Drug profile · INN

reboxetine

reboxetine (EDRONAX) is a norepinephrine transporter inhibitor. Associated with Pfizer Australia Pty Ltd.

TGA: approved
Patents linked 9
Pipeline programs 3
News articles 0
Drug details — reboxetine

Quick answer

reboxetine (EDRONAX) is a norepinephrine transporter inhibitor. Associated with Pfizer Australia Pty Ltd.

Key facts

INN reboxetine
Brand EDRONAX
Mechanism Norepinephrine transporter inhibitor
Target Sodium-dependent noradrenaline transporter

Mechanism of action

Norepinephrine transporter inhibitor

Primary target: Sodium-dependent noradrenaline transporter

Approval history

Authority Status Date
TGA approved

Pipeline programs

  1. AXS-12 (Reboxetine) Phase 3 · Axsome Therapeutics · Narcolepsy
  2. AXS-14 (Esreboxetine) Phase 3 · Axsome Therapeutics · Fibromyalgia
  3. INTENSIFY MDD Phase 3 · Disc Medicine · Major depressive disorder

Related & competitor drugs

  1. amitriptyline hydrochloride Norepinephrine transporter inhibitor
  2. atomoxetine hydrochloride Norepinephrine transporter inhibitor
  3. desipramine hydrochloride Norepinephrine transporter inhibitor
  4. desvenlafaxine fumarate Norepinephrine transporter inhibitor
  5. doxepin hydrochloride Norepinephrine transporter inhibitor
  6. duloxetine hydrochloride Norepinephrine transporter inhibitor
  1. US 12246023

    Use of reboxetine to treat narcolepsy

    Expires 2045-03-06T00:00:00.000Z

    granted
  2. US 12115165

    Use of reboxetine to treat narcolepsy

    Expires 2044-10-10T00:00:00.000Z

    granted
  3. US 11957686

    Compositions for delivery of reboxetine

    Expires 2044-04-11T00:00:00.000Z

    granted
  4. US 11883408

    Reboxetine to treat narcolepsy

    Expires 2044-01-25T00:00:00.000Z

    granted
  5. US 11364245

    Use of reboxetine to treat narcolepsy

    Expires 2042-06-16T00:00:00.000Z

    granted
  6. US 11351175

    Use of reboxetine to treat narcolepsy

    Expires 2042-06-02T00:00:00.000Z

    granted
  7. US 11185547

    Use of reboxetine to treat narcolepsy

    Expires 2041-11-25T00:00:00.000Z

    granted
  8. US 11135226

    Use of reboxetine to treat narcolepsy

    Expires 2041-09-30T00:00:00.000Z

    granted
  9. US 11020402

    Use of reboxetine to treat narcolepsy

    Expires 2041-05-27T00:00:00.000Z

    granted

Frequently asked questions

What is reboxetine?

reboxetine (EDRONAX) is a norepinephrine transporter inhibitor. Associated with Pfizer Australia Pty Ltd.

What is the brand name for reboxetine?

EDRONAX is a marketed brand name for reboxetine. Check FDA Drugs@FDA for the current US label holder and prescribing information.