Wednesday, July 8, 2026

Drug profile · INN

netarsudil mesylate

netarsudil mesylate (RHOPRESSA) is a rho-associated protein kinase inhibitor. Route of administration: ophthalmic. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — netarsudil mesylate
US status
approved
Class
Route
OPHTHALMIC
Patents
0
Programs
0
Data quality
0.84

Quick answer

netarsudil mesylate (RHOPRESSA) is a rho-associated protein kinase inhibitor. Route of administration: ophthalmic. Current US regulatory status: approved.

Key facts

INN netarsudil mesylate
Brand RHOPRESSA
Mechanism Rho-associated protein kinase inhibitor
Target Rho-associated protein kinase
Route OPHTHALMIC
Formulation SOLUTION/DROPS

Mechanism of action

Rho-associated protein kinase inhibitor

Primary target: Rho-associated protein kinase

Approval history

Authority Status Date
FDA approved

Related & competitor drugs

  1. belumosudil mesylate Rho-associated protein kinase inhibitor
  2. belumosudil Antineoplastic and immunomodulating agents (L04)

Frequently asked questions

What is netarsudil mesylate?

netarsudil mesylate (RHOPRESSA) is a rho-associated protein kinase inhibitor. Route of administration: ophthalmic. Current US regulatory status: approved.

What is the brand name for netarsudil mesylate?

RHOPRESSA is a marketed brand name for netarsudil mesylate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of netarsudil mesylate?

netarsudil mesylate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.