Wednesday, July 8, 2026

Drug profile · INN

netarsudil

netarsudil (RHOKIINSA) is a rho-associated protein kinase inhibitor. Route of administration: drops. Current US regulatory status: approved.

FDA: approved EMA: approved Sensory organs (S01) S01EX05
US status approved
Patents linked 0
Pipeline programs 4
News articles 0
Drug details — netarsudil
US status
approved
Class
Sensory organs (S01)
Route
DROPS
Patents
0
Programs
4
Data quality
0.84

Quick answer

netarsudil (RHOKIINSA) is a rho-associated protein kinase inhibitor. Route of administration: drops. Current US regulatory status: approved.

Key facts

INN netarsudil
Brand RHOKIINSA
Mechanism Rho-associated protein kinase inhibitor
Therapeutic class Sensory organs (S01)
Route DROPS
Formulation SOLUTION
ATC code S01EX05

Mechanism of action

Rho-associated protein kinase inhibitor

Approval history

Authority Status Date
FDA approved
EMA approved

Pipeline programs

  1. 64Cu(II)Cl2 solution for injection Phase 3 · A.C.O.M. - Advanced · Cancer on the prostatic bed
  2. P.64Cu.003.01 Phase 3 · A.C.O.M. - Advanced · Prostate cancer at risk of developing metastatic lesions
  3. FirstHCMU-JBi-PARTOM Phase 2 · Chinese Academy of · Metastatic Castration-resistant Prostate Cancer
  4. PC-IIT-003 Phase 2 · First People's Hospital · Pancreatic Cancer

Related & competitor drugs

  1. aflibercept Sensory organs (S01)
  2. atropine sulfate Sensory organs (S01)
  3. bimatoprost Sensory organs (S01)
  4. atropine Sensory organs (S01)
  5. brinzolamide Sensory organs (S01)
  6. latanoprost Sensory organs (S01)

Frequently asked questions

What is netarsudil?

netarsudil (RHOKIINSA) is a rho-associated protein kinase inhibitor. Route of administration: drops. Current US regulatory status: approved.

What is the brand name for netarsudil?

RHOKIINSA is a marketed brand name for netarsudil. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of netarsudil?

netarsudil has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.