Wednesday, July 8, 2026

Drug profile · INN

methscopolamine bromide

methscopolamine bromide (METHSCOPOLAMINE BROMIDE) is a muscarinic acetylcholine receptor m1 antagonist. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 20
Pipeline programs 2
News articles 0
Drug details — methscopolamine bromide
US status
approved
Class
Route
ORAL
Patents
20
Programs
2
Data quality
0.84

Quick answer

methscopolamine bromide (METHSCOPOLAMINE BROMIDE) is a muscarinic acetylcholine receptor m1 antagonist. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN methscopolamine bromide
Brand METHSCOPOLAMINE BROMIDE
Mechanism Muscarinic acetylcholine receptor M1 antagonist
Target Muscarinic acetylcholine receptor M1
Route ORAL
Formulation TABLET

Mechanism of action

Muscarinic acetylcholine receptor M1 antagonist

Primary target: Muscarinic acetylcholine receptor M1

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. Evaluation of the safety and efficacy of Cont... for Parkinson's disease Phase 2 · Anaxis Pharma · Parkinson's disease
  2. dopamine Unknown · First People's Hospital · Renal Artery Stenosis Atherosclerotic

Related & competitor drugs

  1. atropine sulfate Sensory organs (S01)
  2. benztropine mesylate Muscarinic acetylcholine receptor M1 antagonist
  3. dicyclomine hydrochloride Muscarinic acetylcholine receptor M3 antagonist
  4. glycopyrrolate Muscarinic acetylcholine receptor M3 antagonist
  5. pilocarpine hydrochloride Muscarinic acetylcholine receptor M3 agonist
  6. scopolamine Muscarinic acetylcholine receptor M1 antagonist

Related patents

  1. US 12162861

    Dopamine D3 receptor selective antagonists/partial agonists; method of making; and use thereof

    Expires Mon Dec 05 2044 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 12145922

    Selective D3 dopamine receptor agonists and methods of their use

    Expires Mon Nov 14 2044 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 12102640

    Use of dopamine and serotonin receptor antagonists for treatment in a subject with retinal degeneration

    Expires Mon Sep 26 2044 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. US 12097196

    Dopamine D3 receptor selective antagonists/partial agonists and uses thereof

    Expires Mon Sep 19 2044 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  5. US 11634404

    Selective D3 dopamine receptor agonists and methods of their use

    Expires Mon Apr 20 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  6. US 11337971

    Dopamine D3 receptor selective antagonists/partial agonists and uses thereof

    Expires Mon May 19 2042 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  7. US 11299476

    Dopamine D3 receptor selective antagonists/partial agonists; method of making; and use thereof

    Expires Mon Apr 07 2042 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  8. US 11261461

    Methods and compositions for selective generation of dopaminergic precursors

    Expires Mon Feb 24 2042 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  9. US 11033554

    Use of dopamine and serotonin receptor antagonists for treatment in a subject with retinal degeneration

    Expires Mon Jun 10 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  10. WO 2020246903

    INHIBITEURS DE DOPAMINE-B-HYDROXYLASE

    Expires Wed Dec 05 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  11. CA 3142348

    INHIBITEURS DE DOPAMINE-B-HYDROXYLASE

    Expires Wed Dec 05 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  12. AU 2018379646

    Dopamine-B-hydroxylase inhibitors

    Expires Wed Jun 06 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  13. US 10654842

    Dopamine D3 receptor antagonist compounds

    Expires Mon May 14 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  14. US 10577361

    Dopamine D3 receptor antagonists having a morpholine moiety

    Expires Mon Feb 27 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  15. CA 3103212

    FORMULATIONS COMPRENANT DES INHIBITEURS DE LA DOPAMINE-S-HYDROXYLASE ET LEURS PROCEDES DE PREPARATION

    Expires Wed Dec 28 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  16. US 2019337950

    BLOOD-BRAIN BARRIER-PENETRANT DOPAMINE-B-HYDROXYLASE INHIBITORS

    Expires Wed Nov 02 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  17. CA 3082337

    INHIBITEURS DE DOPAMINE-B-HYDROXYLASE

    Expires Wed Jun 08 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  18. US 10273244

    Substituted hexahydropyrrolo[3,4-b]pyrroles and hexahydrocyclopenta[c]pyrroles as dopamine receptor modulators

    Expires Mon Apr 25 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  19. US 10239870

    Dopamine D3 receptor antagonists

    Expires Mon Mar 21 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  20. US 10016499

    Multifunctional metal nanoparticles having a polydopamine-based surface and methods of making and using the same

    Expires Mon Jul 05 2038 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is methscopolamine bromide?

methscopolamine bromide (METHSCOPOLAMINE BROMIDE) is a muscarinic acetylcholine receptor m1 antagonist. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for methscopolamine bromide?

METHSCOPOLAMINE BROMIDE is a marketed brand name for methscopolamine bromide. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of methscopolamine bromide?

methscopolamine bromide has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.