Wednesday, July 8, 2026

Drug profile · INN

glycopyrrolate

glycopyrrolate (GLYCOPYRROLATE) is a muscarinic acetylcholine receptor m3 antagonist. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 6
Pipeline programs 0
News articles 0
Drug details — glycopyrrolate
US status
approved
Class
Route
ORAL
Patents
6
Programs
0
Data quality
0.89

Quick answer

glycopyrrolate (GLYCOPYRROLATE) is a muscarinic acetylcholine receptor m3 antagonist. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: oral. Current US regulatory status: approved.

Key facts

INN glycopyrrolate
Brand GLYCOPYRROLATE
Mechanism Muscarinic acetylcholine receptor M3 antagonist
Target Muscarinic acetylcholine receptor M1
Route ORAL
Formulation TABLET, ORALLY DISINTEGRATING

Mechanism of action

Muscarinic acetylcholine receptor M3 antagonist

Primary target: Muscarinic acetylcholine receptor M1

Approval history

Authority Status Date
FDA approved

Related & competitor drugs

  1. atropine sulfate Sensory organs (S01)
  2. benztropine mesylate Muscarinic acetylcholine receptor M1 antagonist
  3. dicyclomine hydrochloride Muscarinic acetylcholine receptor M3 antagonist
  4. pilocarpine hydrochloride Muscarinic acetylcholine receptor M3 agonist
  5. scopolamine Muscarinic acetylcholine receptor M1 antagonist
  6. anisotropine methylbromide Muscarinic acetylcholine receptor M1 antagonist
  1. US 10548875

    Glycopyrrolate salts

    Expires Mon Jan 30 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 10543192

    Glycopyrrolate salts

    Expires Mon Jan 23 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 10004717

    Glycopyrrolate salts

    Expires Mon Jun 21 2038 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. US 9610278

    Glycopyrrolate salts

    Expires Mon Mar 30 2037 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  5. US 9259414

    Glycopyrrolate salts

    Expires Mon Feb 11 2036 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  6. US 9006462

    Glycopyrrolate salts

    Expires Mon Apr 09 2035 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is glycopyrrolate?

glycopyrrolate (GLYCOPYRROLATE) is a muscarinic acetylcholine receptor m3 antagonist. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: oral. Current US regulatory status: approved.

What is the brand name for glycopyrrolate?

GLYCOPYRROLATE is a marketed brand name for glycopyrrolate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of glycopyrrolate?

glycopyrrolate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.