Saturday, July 11, 2026

Drug profile · INN

medroxyprogesterone

medroxyprogesterone (RALOVERA) is a progesterone receptor agonist. Associated with Pfizer Australia Pty Ltd.

TGA: approved
Patents linked 0
Pipeline programs 4
News articles 0
Drug details — medroxyprogesterone

Quick answer

medroxyprogesterone (RALOVERA) is a progesterone receptor agonist. Associated with Pfizer Australia Pty Ltd.

Key facts

INN medroxyprogesterone
Brand RALOVERA
Mechanism Progesterone receptor agonist
Target Progesterone receptor

Mechanism of action

Progesterone receptor agonist

Primary target: Progesterone receptor

Approval history

Authority Status Date
TGA approved

Pipeline programs

  1. MK-5684-015 Phase 3 · MSD Merck Sharp · Breast cancer, Ovarian cancer, Endometrial cancer
  2. medroxyprogesterone acetate Phase 1 · Teva Pharma · Healthy
  3. Depo-Medroxyprogesterone Acetate Approved · United Therapeutics Europe · HIV
  4. Subcutaneous depot medroxyprogesterone acetate Approved · Protara Therapeutics · Contraception

Related & competitor drugs

  1. desogestrel Progesterone receptor agonist
  2. medroxyprogesterone acetate Progesterone receptor agonist
  3. megestrol acetate Progesterone receptor agonist
  4. norethindrone Progesterone receptor agonist
  5. norethindrone acetate Progesterone receptor agonist
  6. progesterone Progesterone receptor agonist

Frequently asked questions

What is medroxyprogesterone?

medroxyprogesterone (RALOVERA) is a progesterone receptor agonist. Associated with Pfizer Australia Pty Ltd.

What is the brand name for medroxyprogesterone?

RALOVERA is a marketed brand name for medroxyprogesterone. Check FDA Drugs@FDA for the current US label holder and prescribing information.