Friday, July 10, 2026

Drug profile · INN

margetuximab-cmkb

margetuximab-cmkb (MARGENZA) is a receptor protein-tyrosine kinase erbb-2 inhibitor. Route of administration: injection. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — margetuximab-cmkb
US status
approved
Class
Route
INJECTION
Patents
0
Programs
0
Data quality
0.84

Quick answer

margetuximab-cmkb (MARGENZA) is a receptor protein-tyrosine kinase erbb-2 inhibitor. Route of administration: injection. Current US regulatory status: approved.

Key facts

INN margetuximab-cmkb
Brand MARGENZA
Mechanism Receptor protein-tyrosine kinase erbB-2 inhibitor
Target Receptor tyrosine-protein kinase erbB-2
Route INJECTION
Formulation INJECTABLE

Mechanism of action

Receptor protein-tyrosine kinase erbB-2 inhibitor

Primary target: Receptor tyrosine-protein kinase erbB-2

Approval history

Authority Status Date
FDA approved

Related & competitor drugs

  1. zanidatamab Antineoplastic and immunomodulating agents (L01)
  2. zanidatamab-hrii Receptor protein-tyrosine kinase erbB-2 inhibitor
  3. ado-trastuzumab emtansine Receptor protein-tyrosine kinase erbB-2 binding agent
  4. pertuzumab Antineoplastic and immunomodulating agents (L01)
  5. trastuzumab Antineoplastic and immunomodulating agents (L01)
  6. trastuzumab-anns Receptor protein-tyrosine kinase erbB-2 inhibitor

Frequently asked questions

What is margetuximab-cmkb?

margetuximab-cmkb (MARGENZA) is a receptor protein-tyrosine kinase erbb-2 inhibitor. Route of administration: injection. Current US regulatory status: approved.

What is the brand name for margetuximab-cmkb?

MARGENZA is a marketed brand name for margetuximab-cmkb. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of margetuximab-cmkb?

margetuximab-cmkb has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.