Wednesday, July 8, 2026

Drug profile · INN

lutetium lu-177 vipivotide tetraxetan

lutetium lu-177 vipivotide tetraxetan (PLUVICTO) is a glutamate carboxypeptidase ii binding agent. Route of administration: intravenous. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 1
News articles 3
Drug details — lutetium lu-177 vipivotide tetraxetan

Quick answer

lutetium lu-177 vipivotide tetraxetan (PLUVICTO) is a glutamate carboxypeptidase ii binding agent. Route of administration: intravenous. Current US regulatory status: approved.

Key facts

INN lutetium lu-177 vipivotide tetraxetan
Brand PLUVICTO
Mechanism Glutamate carboxypeptidase II binding agent
Target DNA
Route INTRAVENOUS
Formulation SOLUTION

Mechanism of action

Glutamate carboxypeptidase II binding agent

Primary target: DNA

Approval history

Authority Status Date
FDA approved

Recent coverage

Pipeline programs

  1. 177Lu-PSMA-617 Phase 2 · United Therapeutics Europe · Metastatic Hormone Naive Prostate Cancer

Related & competitor drugs

  1. acyclovir Human herpesvirus 1 DNA polymerase inhibitor
  2. acyclovir sodium Human herpesvirus 1 DNA polymerase inhibitor
  3. azacitidine Antineoplastic and immunomodulating agents (L01)
  4. bleomycin sulfate DNA inhibitor
  5. busulfan Antineoplastic and immunomodulating agents (L01)
  6. capecitabine Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is lutetium lu-177 vipivotide tetraxetan?

lutetium lu-177 vipivotide tetraxetan (PLUVICTO) is a glutamate carboxypeptidase ii binding agent. Route of administration: intravenous. Current US regulatory status: approved.

What is the brand name for lutetium lu-177 vipivotide tetraxetan?

PLUVICTO is a marketed brand name for lutetium lu-177 vipivotide tetraxetan. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of lutetium lu-177 vipivotide tetraxetan?

lutetium lu-177 vipivotide tetraxetan has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.