Saturday, July 11, 2026

Drug profile · INN

linerixibat

linerixibat (LYNAVOY) is a ileal bile acid transporter inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 0
News articles 1
Drug details — linerixibat
US status
approved
Class
Route
ORAL
Patents
0
Programs
0
Data quality
0.84

Quick answer

linerixibat (LYNAVOY) is a ileal bile acid transporter inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN linerixibat
Brand LYNAVOY
Mechanism Ileal bile acid transporter inhibitor
Target Ileal sodium/bile acid cotransporter
Route ORAL
Formulation TABLET

Mechanism of action

Ileal bile acid transporter inhibitor

Primary target: Ileal sodium/bile acid cotransporter

Approval history

Authority Status Date
FDA approved

Recent coverage

Related & competitor drugs

  1. maralixibat chloride Alimentary tract and metabolism (A05)
  2. odevixibat Alimentary tract and metabolism (A05)
  3. maralixibat Alimentary tract and metabolism (A05)

Frequently asked questions

What is linerixibat?

linerixibat (LYNAVOY) is a ileal bile acid transporter inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for linerixibat?

LYNAVOY is a marketed brand name for linerixibat. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of linerixibat?

linerixibat has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.