Wednesday, July 8, 2026

Drug profile · INN

ixazomib citrate

ixazomib citrate (NINLARO) is a 26s proteosome inhibitor. Associated with Takeda. Route of administration: oral. Current US regulatory status: approved.

FDA: approved PMDA: approved
US status approved
Patents linked 2
Pipeline programs 25
News articles 0
Drug details — ixazomib citrate
US status
approved
Class
Route
ORAL
Patents
2
Programs
25
Data quality
0.89

Quick answer

ixazomib citrate (NINLARO) is a 26s proteosome inhibitor. Associated with Takeda. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN ixazomib citrate
Brand NINLARO
Mechanism 26S proteosome inhibitor
Target 26S proteasome
Route ORAL
Formulation CAPSULE
Originator Takeda

Mechanism of action

26S proteosome inhibitor

Primary target: 26S proteasome

Approval history

Authority Status Date
FDA approved
PMDA approved

Pipeline programs

  1. IXAZOMIB Phase 3 · Takeda · Relapsed or Refractory Systemic Light Chain Amyloidosis
  2. Ixazomib Phase 3 · Takeda · Relapsed Multiple Myeloma
  3. Ixazomib Citrate Phase 3 · Takeda · Multiple Myeloma
  4. IXAZOMIB Phase 2 · Takeda · Follicular Lymphoma
  5. Ixazomib Phase 2 · Takeda · Mantle Cell Lymphoma
  6. Ixazomib Phase 2 · Takeda · ALL, Childhood
  7. Ixazomib Phase 2 · Takeda · Leukemia
  8. Ixazomib Phase 2 · Takeda · Multiple Myeloma

Related & competitor drugs

  1. bortezomib Antineoplastic and immunomodulating agents (L01)
  2. carfilzomib Antineoplastic and immunomodulating agents (L01)
  3. ixazomib Antineoplastic and immunomodulating agents (L01)
  1. US 11053261

    Solid state forms of ixazomib citrate

    Expires Mon Jul 01 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 10604537

    Solid state forms of ixazomib citrate

    Expires Mon Mar 26 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is ixazomib citrate?

ixazomib citrate (NINLARO) is a 26s proteosome inhibitor. Associated with Takeda. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for ixazomib citrate?

NINLARO is a marketed brand name for ixazomib citrate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of ixazomib citrate?

ixazomib citrate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.