Wednesday, July 8, 2026

Drug profile · INN

granisetron

granisetron (SANCUSO) is a serotonin 3a (5-ht3a) receptor antagonist. Associated with Heron Therapeutics. Route of administration: subcutaneous. Current US regulatory status: approved.

FDA: approved EMA: approved Alimentary tract and metabolism (A04) A04AA02
US status approved
Patents linked 3
Pipeline programs 5
News articles 0
Drug details — granisetron
US status
approved
Class
Alimentary tract and metabolism (A04)
Route
SUBCUTANEOUS
Patents
3
Programs
5
Data quality
0.89

Quick answer

granisetron (SANCUSO) is a serotonin 3a (5-ht3a) receptor antagonist. Associated with Heron Therapeutics. Route of administration: subcutaneous. Current US regulatory status: approved.

Key facts

INN granisetron
Brand SANCUSO
Mechanism Serotonin 3a (5-HT3a) receptor antagonist
Target 5-hydroxytryptamine receptor 3A
Therapeutic class Alimentary tract and metabolism (A04)
Route SUBCUTANEOUS
Formulation INJECTABLE
ATC code A04AA02

Mechanism of action

Serotonin 3a (5-HT3a) receptor antagonist

Primary target: 5-hydroxytryptamine receptor 3A

Approval history

Authority Status Date
FDA approved
EMA approved

Pipeline programs

  1. ALL3024 Phase 2 · Telethon Foundation · Very High-Risk T-Lineage Acute Lymphoblastic Leukemia (ALL)
  2. GRANISETRON EXTENDED RELEASE INJECTION (GERSC) Phase 2 · Heron Therapeutics · Chemotherapy-induced Nausea and Vomiting
  3. J2R-MC-YAAD Phase 2 · Eli Lilly and · Nausea, Drug-Related Side Effects and Adverse Reactions, Vom
  4. Granisetron hydrochloride 1 mg tablets Phase 1 · Teva Pharma · Healthy
  5. SUSTOL Approved · Heron Therapeutics · Chemotherapy-Induced Nausea and Vomiting (CINV)

Related & competitor drugs

  1. agalsidase alfa Alimentary tract and metabolism (A16)
  2. alogliptin Alimentary tract and metabolism (A10)
  3. alogliptin benzoate Alimentary tract and metabolism (A10)
  4. alosetron hydrochloride Serotonin 3a (5-HT3a) receptor antagonist
  5. aprepitant Alimentary tract and metabolism (A04)
  6. budesonide Alimentary tract and metabolism (A07)
  1. US 10357570

    Methods of treating nausea utilizing semi-solid delivery vehicle compositions comprising granisetron

    Expires Mon Jul 18 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 9913910

    Methods of treating nausea utilizing semi-solid delivery vehicle compositions comprising granisetron

    Expires Mon Mar 08 2038 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 8715710

    Semi-solid delivery vehicle and pharmaceutical compositions for delivery of granisetron

    Expires Mon May 01 2034 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is granisetron?

granisetron (SANCUSO) is a serotonin 3a (5-ht3a) receptor antagonist. Associated with Heron Therapeutics. Route of administration: subcutaneous. Current US regulatory status: approved.

What is the brand name for granisetron?

SANCUSO is a marketed brand name for granisetron. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of granisetron?

granisetron has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.