Wednesday, July 8, 2026

Drug profile · INN

glycopyrronium tosylate

glycopyrronium tosylate (GLYCOPYRRONIUM TOSYLATE) is a muscarinic acetylcholine receptor inhibitor. Route of administration: topical. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 4
Pipeline programs 1
News articles 0
Drug details — glycopyrronium tosylate
US status
approved
Class
Route
TOPICAL
Patents
4
Programs
1
Data quality
0.84

Quick answer

glycopyrronium tosylate (GLYCOPYRRONIUM TOSYLATE) is a muscarinic acetylcholine receptor inhibitor. Route of administration: topical. Current US regulatory status: approved.

Key facts

INN glycopyrronium tosylate
Brand GLYCOPYRRONIUM TOSYLATE
Mechanism Muscarinic acetylcholine receptor inhibitor
Target Muscarinic acetylcholine receptor
Route TOPICAL
Formulation CLOTH

Mechanism of action

Muscarinic acetylcholine receptor inhibitor

Primary target: Muscarinic acetylcholine receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. Glycopyrronium Approved · Chinese Academy of · Postoperative Nausea and Vomiting

Related & competitor drugs

  1. atropine sulfate Sensory organs (S01)
  2. benztropine mesylate Muscarinic acetylcholine receptor M1 antagonist
  3. bethanechol chloride Muscarinic acetylcholine receptor M3 agonist
  4. dicyclomine hydrochloride Muscarinic acetylcholine receptor M3 antagonist
  5. fesoterodine fumarate Muscarinic acetylcholine receptor M2 antagonist
  6. glycopyrrolate Muscarinic acetylcholine receptor M3 antagonist

Related patents

  1. US 10548875

    Glycopyrrolate salts

    Expires Mon Jan 30 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 10543192

    Glycopyrrolate salts

    Expires Mon Jan 23 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 10004717

    Glycopyrrolate salts

    Expires Mon Jun 21 2038 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. US 9259414

    Glycopyrrolate salts

    Expires Mon Feb 11 2036 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is glycopyrronium tosylate?

glycopyrronium tosylate (GLYCOPYRRONIUM TOSYLATE) is a muscarinic acetylcholine receptor inhibitor. Route of administration: topical. Current US regulatory status: approved.

What is the brand name for glycopyrronium tosylate?

GLYCOPYRRONIUM TOSYLATE is a marketed brand name for glycopyrronium tosylate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of glycopyrronium tosylate?

glycopyrronium tosylate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.